In vitro and in vivo biological activities of SR140333, a novel potent non-peptide tachykinin NK1 receptor antagonist
EMONDS-ALT, X, DOUTREMEPUICH, J.-D, VAN BROECK, D, SOUBRIE, P, LE FUR, G, BRELIERE, J.-C, HEAULME, M, NELIAT, G, SANTUCCI, V, STEINBERG, R, VILAIN, P, BICHON, D, DUCOUX, J.-P, PROIETTO, V
Published in European journal of pharmacology (21.12.1993)
Published in European journal of pharmacology (21.12.1993)
Get full text
Journal Article
SSR240600 [(R)-2-(1-{2-[4-{2-[3,5-Bis(trifluoromethyl)phenyl]acetyl}-2-(3,4-dichlorophenyl)-2-morpholinyl]ethyl}- 4-piperidinyl)-2-methylpropanamide], a Centrally Active Nonpeptide Antagonist of the Tachykinin Neurokinin-1 Receptor: I. Biochemical and Pharmacological Characterization
Emonds-Alt, Xavier, Proietto, Vincenzo, Steinberg, Régis, Oury-Donat, Florence, Vigé, Xavier, Vilain, Pol, Naline, Emmanuel, Daoui, Samira, Advenier, Charles, Le Fur, Gérard, Maffrand, Jean-Pierre, Soubrié, Philippe, Pascal, Marc
Published in The Journal of pharmacology and experimental therapeutics (01.12.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2002)
Get full text
Journal Article
POLYCYCLIC AMINE COMPOUND AND ENANTIOMER THEREOF
GUEULE PATRICK, EMONDSALT XAVIER, GOULAOUIC PIERRE, PROIETTO VINCENZO
Year of Publication 29.01.2003
Get full text
Year of Publication 29.01.2003
Patent
Biochemical and pharmacological activities of SSR 146977, a new potent nonpeptide tachykinin NK3 receptor antagonist
Emonds-Alt, Xavier, Proietto, Vincenzo, Steinberg, Régis, Advenier, Charles, Daoui, Samira, Naline, Emmanuel, Gueudet, Christiane, Michaud, Jean-Claude, Oury-Donat, Florence, Poncelet, Martine, Vilain, Pol, Fur, Gérard Le, Maffrand, Jean-Pierre, Soubrié, Philippe, Pascal, Marc
Published in Canadian journal of physiology and pharmacology (01.05.2002)
Published in Canadian journal of physiology and pharmacology (01.05.2002)
Get full text
Journal Article
Biochemical and pharmacological activities of SSR 146977, a new potent nonpeptide tachykinin NK 3 receptor antagonist
Emonds-Alt, Xavier, Proietto, Vincenzo, Steinberg, Régis, Advenier, Charles, Daoui, Samira, Naline, Emmanuel, Gueudet, Christiane, Michaud, Jean-Claude, Oury-Donat, Florence, Poncelet, Martine, Vilain, Pol, Fur, Gérard Le, Maffrand, Jean-Pierre, Soubrié, Philippe, Pascal, Marc
Published in Canadian journal of physiology and pharmacology (01.05.2002)
Published in Canadian journal of physiology and pharmacology (01.05.2002)
Get full text
Journal Article
Pharmacological profile and chemical synthesis of SR 48968, a non-peptide antagonist of the neurokinin A (NK 2) receptor
Emonds-Alt, Xavier, Proietto, Vincenzo, Van Broeck, Didier, Vilain, Pol, Advenier, Charles, Neliat, Gervais, Le Fur, Gérard, Brelère, Jean-Claude
Published in Bioorganic & medicinal chemistry letters (1993)
Published in Bioorganic & medicinal chemistry letters (1993)
Get full text
Journal Article