Deorphanization of a G protein-coupled receptor for oleoylethanolamide and its use in the discovery of small-molecule hypophagic agents
Overton, Hilary A., Babbs, Adam J., Doel, Sheila M., Fyfe, Matthew C.T., Gardner, Lisa S., Griffin, Graeme, Jackson, Helen C., Procter, Martin J., Rasamison, Chrystelle M., Tang-Christensen, Mads, Widdowson, Peter S., Williams, Geoffery M., Reynet, Christine
Published in Cell metabolism (01.03.2006)
Published in Cell metabolism (01.03.2006)
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SAR, Pharmacokinetics, Safety, and Efficacy of Glucokinase Activating 2-(4-Sulfonylphenyl)-N-thiazol-2-ylacetamides: Discovery of PSN-GK1
Bertram, Lisa S, Black, Daniel, Briner, Paul H, Chatfield, Rosemary, Cooke, Andrew, Fyfe, Matthew C. T, Murray, P. John, Naud, Frédéric, Nawano, Masao, Procter, Martin J, Rakipovski, Günaj, Rasamison, Chrystelle M, Reynet, Christine, Schofield, Karen L, Shah, Vilas K, Spindler, Felix, Taylor, Amanda, Turton, Roy, Williams, Geoffrey M, Wong-Kai-In, Philippe, Yasuda, Kosuke
Published in Journal of medicinal chemistry (24.07.2008)
Published in Journal of medicinal chemistry (24.07.2008)
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Design and synthesis of potent carboxylic acid DGAT1 inhibitors with high cell permeability
Bali, Ustav, Barba, Oscar, Dawson, Graham, Gattrell, William T., Horswill, James G., Pan, David A., Procter, Martin J., Rasamison, Chrystelle M., Sambrook Smith, Colin P., Taylor-Warne, Amanda, Wong-Kai-In, Philippe
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Glucokinase-activating ureas
Castelhano, Arlindo L., Dong, Hanqing, Fyfe, Matthew C.T., Gardner, Lisa S., Kamikozawa, Yukari, Kurabayashi, Satomi, Nawano, Masao, Ohashi, Rikiya, Procter, Martin J., Qiu, Li, Rasamison, Chrystelle M., Schofield, Karen L., Shah, Vilas K., Ueta, Kiichiro, Williams, Geoffrey M., Witter, David, Yasuda, Kosuke
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
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Practical Synthesis of 2-Amino-5-fluorothiazole Hydrochloride
Briner, Paul H, Fyfe, Matthew C. T, Martin, Pierre, Murray, P. John, Naud, Frédéric, Procter, Martin J
Published in Organic process research & development (01.03.2006)
Published in Organic process research & development (01.03.2006)
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Structures of synaptic vesicle protein 2A and 2B bound to anticonvulsants
Mittal, Anshumali, Martin, Matthew F, Levin, Elena J, Adams, Christopher, Yang, Meng, Provins, Laurent, Hall, Adrian, Procter, Martin, Ledecq, Marie, Hillisch, Alexander, Wolff, Christian, Gillard, Michel, Horanyi, Peter S, Coleman, Jonathan A
Published in Nature structural & molecular biology (19.06.2024)
Published in Nature structural & molecular biology (19.06.2024)
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A simple route to 6- and 7-fluoro-substituted naphthalene-1-carboxylic acids
Krülle, Thomas M., Barba, Oscar, Davis, Susan H., Dawson, Graham, Procter, Martin J., Staroske, Thomas, Thomas, Gerard H.
Published in Tetrahedron letters (26.02.2007)
Published in Tetrahedron letters (26.02.2007)
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COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS
JEEVARATNAM REVATHY PERPETUA, SAMBROOK SMITH COLIN PETER, SWAIN SIMON ANDREW, STEWART ALAN JOHN WILLIAM, SCHOFIELD KAREN LESLEY, FRY PETER TIMOTHY, FYFE MATTHEW COLIN THOR, BARBA OSCAR, PROCTER MARTIN JAMES, SMYTH DONALD, STONEHOUSE DAVID FRENCH, GATTRELL WILLIAM, KRULLE THOMAS MARTIN
Year of Publication 09.12.2011
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Year of Publication 09.12.2011
Patent
Synthesis of salinomycin
Kocienski, PJ, Brown, RCD, Pommier, A, Procter, M, Schmidt, B
Published in Journal of the Chemical Society, Perkin Transactions 1 (07.01.1998)
Published in Journal of the Chemical Society, Perkin Transactions 1 (07.01.1998)
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