In-vitro profile and ex-vivo anticoagulant activity of the direct thrombin inhibitor dabigatran and its orally active prodrug, dabigatran etexilate
Wienen, Wolfgang, Stassen, Jean-Marie, Priepke, Henning, Ries, Uwe Joerg, Hauel, Norbert
Published in Thrombosis and haemostasis (01.07.2007)
Published in Thrombosis and haemostasis (01.07.2007)
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Structure-Based Design of Novel Potent Nonpeptide Thrombin Inhibitors
Hauel, Norbert H, Nar, Herbert, Priepke, Henning, Ries, Uwe, Stassen, Jean-Marie, Wienen, Wolfgang
Published in Journal of medicinal chemistry (25.04.2002)
Published in Journal of medicinal chemistry (25.04.2002)
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Effects of the direct thrombin inhibitor dabigatran and its orally active prodrug, dabigatran etexilate, on thrombus formation and bleeding time in rats
Wienen, Wolfgang, Stassen, Jean-Marie, Priepke, Henning, Ries, Uwe Joerg, Hauel, Norbert
Published in Thrombosis and haemostasis (01.08.2007)
Published in Thrombosis and haemostasis (01.08.2007)
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Mechanism of Human Telomerase Inhibition by BIBR1532, a Synthetic, Non-nucleosidic Drug Candidate
Pascolo, Emanuelle, Wenz, Christian, Lingner, Joachim, Hauel, Norbert, Priepke, Henning, Kauffmann, Iris, Garin-Chesa, Pilar, Rettig, Wolfgang J., Damm, Klaus, Schnapp, Andreas
Published in The Journal of biological chemistry (03.05.2002)
Published in The Journal of biological chemistry (03.05.2002)
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1,2-Diacetals: A New Opportunity for Organic Synthesis
Ley, Steven V, Baeschlin, Daniel K, Dixon, Darren J, Foster, Alison C, Ince, Stuart J, Priepke, Henning W. M, Reynolds, Dominic J
Published in Chemical reviews (01.01.2001)
Published in Chemical reviews (01.01.2001)
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Heterocyclic thrombin inhibitors. Part 2: quinoxalinone derivatives as novel, potent antithrombotic agents
Ries, Uwe J., Priepke, Henning W.M., Hauel, Norbert H., Handschuh, Sandra, Mihm, Gerhard, Stassen, Jean M., Wienen, Wolfgang, Nar, Herbert
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
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A new strategy for oligosaccharide assembly exploiting cyclohexane-1,2-diacetal methodology: An efficient synthesis of a high mannose type nonasaccharide
Grice, P, Ley, SV, Pietruszka, J, Osborn, HMI, Priepke, HWM, Warriner, SL
Published in Chemistry : a European journal (01.03.1997)
Published in Chemistry : a European journal (01.03.1997)
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Structural Basis for Inhibition Promiscuity of Dual Specific Thrombin and Factor Xa Blood Coagulation Inhibitors
Nar, Herbert, Bauer, Margit, Schmid, Angela, Stassen, Jean-Marie, Wienen, Wolfgang, Priepke, Henning W.M, Kauffmann, Iris K, Ries, Uwe J, Hauel, Norbert H
Published in Structure (London) (10.01.2001)
Published in Structure (London) (10.01.2001)
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Heterocyclic thrombin inhibitors. Part 1: design and synthesis of amidino-phenoxy quinoline derivatives
Ries, Uwe J., Priepke, Henning W.M., Hauel, Norbert H., Haaksma, Eric E.J., Stassen, Jean M., Wienen, Wolfgang, Nar, Herbert
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
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Direct protection of 1,2-diols from alpha-diketones
Douglas, NL, Ley, SV, Osborn, HMI, Owen, DR, Priepke, HWM, Warriner, SL
Published in Synlett (01.08.1996)
Published in Synlett (01.08.1996)
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Synthesis of the nonamannan residue of a glycoprotein with high mannose content
Grice, P, Ley, SV, Pietruszka, J, Priepke, HWM
Published in Angewandte Chemie International Edition (02.02.1996)
Published in Angewandte Chemie International Edition (02.02.1996)
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The discovery of dabigatran etexilate
van Ryn, Joanne, Goss, Ashley, Hauel, Norbert, Wienen, Wolfgang, Priepke, Henning, Nar, Herbert, Clemens, Andreas
Published in Frontiers in pharmacology (01.01.2013)
Published in Frontiers in pharmacology (01.01.2013)
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A highly selective telomerase inhibitor limiting human cancer cell proliferation
Damm, Klaus, Hemmann, Ulrike, Garin-Chesa, Pilar, Hauel, Norbert, Kauffmann, Iris, Priepke, Henning, Niestroj, Claudia, Daiber, Christine, Enenkel, Barbara, Guilliard, Bernd, Lauritsch, Ines, Müller, Elfriede, Pascolo, Emanuelle, Sauter, Gabriele, Pantic, Milena, Martens, Uwe M., Wenz, Christian, Lingner, Joachim, Kraut, Norbert, Rettig, Wolfgang J., Schnapp, Andreas
Published in The EMBO journal (17.12.2001)
Published in The EMBO journal (17.12.2001)
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Effects of Dabigatran, a Direct Thrombin Inhibitor, as Compared to the Direct Factor Xa Inhibitors, Rivaroxaban and Apixaban, on Tissue Factor-Induced Human Platelet Aggregation in Platelet Rich Plasma
van Ryn, Joanne, Kink-Eiband, Monika, Hauel, Norbert, Priepke, Henning, Wienen, Wolfgang
Published in Blood (16.11.2007)
Published in Blood (16.11.2007)
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Comparison of the Antithrombotic Effectiveness of the Direct Thrombin Inhibitor, Dabigatran Etexilate, and Two Factor Xa Inhibitors in an A-V Shunt Model of Thrombosis in Rabbits
van Ryn, Joanne, Hauel, Norbert, Priepke, Henning, Gerlach, Kai, Schuler-Metz, Annette, Wienen, Wolfgang
Published in Blood (16.11.2007)
Published in Blood (16.11.2007)
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Dabigatran Inhibits Arterial Thrombosis in a Porcine Model of Cyclic Flow Reduction
van Ryn, Joanne, Priepke, Henning, Ries, Uwe J., Hauel, Norbert, Stassen, Jean-Marie, Wienen, Wolfgang
Published in Blood (16.11.2006)
Published in Blood (16.11.2006)
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