Diverse drug-resistance mechanisms can emerge from drug-tolerant cancer persister cells
Ramirez, Michael, Rajaram, Satwik, Steininger, Robert J, Osipchuk, Daria, Roth, Maike A, Morinishi, Leanna S, Evans, Louise, Ji, Weiyue, Hsu, Chien-Hsiang, Thurley, Kevin, Wei, Shuguang, Zhou, Anwu, Koduru, Prasad R, Posner, Bruce A, Wu, Lani F, Altschuler, Steven J
Published in Nature communications (19.02.2016)
Published in Nature communications (19.02.2016)
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Journal Article
Systematic Identification of Molecular Subtype-Selective Vulnerabilities in Non-Small-Cell Lung Cancer
Kim, Hyun Seok, Mendiratta, Saurabh, Kim, Jiyeon, Pecot, Chad Victor, Larsen, Jill E., Zubovych, Iryna, Seo, Bo Yeun, Kim, Jimi, Eskiocak, Banu, Chung, Hannah, McMillan, Elizabeth, Wu, Sherry, De Brabander, Jef, Komurov, Kakajan, Toombs, Jason E., Wei, Shuguang, Peyton, Michael, Williams, Noelle, Gazdar, Adi F., Posner, Bruce A., Brekken, Rolf A., Sood, Anil K., Deberardinis, Ralph J., Roth, Michael G., Minna, John D., White, Michael A.
Published in Cell (24.10.2013)
Published in Cell (24.10.2013)
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Journal Article
Small-molecule TFEB pathway agonists that ameliorate metabolic syndrome in mice and extend C. elegans lifespan
Wang, Chensu, Niederstrasser, Hanspeter, Douglas, Peter M, Lin, Rueyling, Jaramillo, Juan, Li, Yang, Oswald, Nathaniel W, Zhou, Anwu, McMillan, Elizabeth A, Mendiratta, Saurabh, Wang, Zhaohui, Zhao, Tian, Lin, Zhiqaing, Luo, Min, Huang, Gang, Brekken, Rolf A, Posner, Bruce A, MacMillan, John B, Gao, Jinming, White, Michael A
Published in Nature communications (22.12.2017)
Published in Nature communications (22.12.2017)
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Journal Article
ZNF281 enhances cardiac reprogramming by modulating cardiac and inflammatory gene expression
Zhou, Huanyu, Morales, Maria Gabriela, Hashimoto, Hisayuki, Dickson, Matthew E, Song, Kunhua, Ye, Wenduo, Kim, Min S, Niederstrasser, Hanspeter, Wang, Zhaoning, Chen, Beibei, Posner, Bruce A, Bassel-Duby, Rhonda, Olson, Eric N
Published in Genes & development (01.09.2017)
Published in Genes & development (01.09.2017)
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Journal Article
SMARCA4-inactivating mutations increase sensitivity to Aurora kinase A inhibitor VX-680 in non-small cell lung cancers
Tagal, Vural, Wei, Shuguang, Zhang, Wei, Brekken, Rolf A, Posner, Bruce A, Peyton, Michael, Girard, Luc, Hwang, TaeHyun, Wheeler, David A, Minna, John D, White, Michael A, Gazdar, Adi F, Roth, Michael G
Published in Nature communications (19.01.2017)
Published in Nature communications (19.01.2017)
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Benzoxazole-derivatives enhance progranulin expression and reverse the aberrant lysosomal proteome caused by GRN haploinsufficiency
Tesla, Rachel, Guhl, Charlotte, Werthmann, Gordon C, Dixon, Danielle, Cenik, Basar, Addepalli, Yesu, Liang, Jue, Fass, Daniel M, Rosenthal, Zachary, Haggarty, Stephen J, Williams, Noelle S, Posner, Bruce A, Ready, Joseph M, Herz, Joachim
Published in Nature communications (20.07.2024)
Published in Nature communications (20.07.2024)
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Journal Article
HORMAD1 Is a Negative Prognostic Indicator in Lung Adenocarcinoma and Specifies Resistance to Oxidative and Genotoxic Stress
Nichols, Brandt A, Oswald, Nathaniel W, McMillan, Elizabeth A, McGlynn, Kathleen, Yan, Jingsheng, Kim, Min S, Saha, Janapriya, Mallipeddi, Prema L, LaDuke, Sydnie A, Villalobos, Pamela A, Rodriguez-Canales, Jaime, Wistuba, Ignacio I, Posner, Bruce A, Davis, Anthony J, Minna, John D, MacMillan, John B, Whitehurst, Angelique W
Published in Cancer research (Chicago, Ill.) (01.11.2018)
Published in Cancer research (Chicago, Ill.) (01.11.2018)
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Journal Article
Discovery of tumor-specific irreversible inhibitors of stearoyl CoA desaturase
Theodoropoulos, Panayotis C, Gonzales, Stephen S, Winterton, Sarah E, Rodriguez-Navas, Carlos, McKnight, John S, Morlock, Lorraine K, Hanson, Jordan M, Cross, Bethany, Owen, Amy E, Duan, Yingli, Moreno, Jose R, Lemoff, Andrew, Mirzaei, Hamid, Posner, Bruce A, Williams, Noelle S, Ready, Joseph M, Nijhawan, Deepak
Published in Nature chemical biology (01.04.2016)
Published in Nature chemical biology (01.04.2016)
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Precursor-Directed Generation of Amidine Containing Ammosamide Analogs: Ammosamides E-P
Pan, Ende, Oswald, Nathaniel W, Legako, Aaron G, Life, Janie M, Posner, Bruce A, Macmillan, John B
Published in Chemical science (Cambridge) (01.01.2013)
Published in Chemical science (Cambridge) (01.01.2013)
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Journal Article
A highly-sensitive high throughput assay for dynamin's basal GTPase activity
Mohanakrishnan, Aparna, Tran, Triet Vincent M, Kumar, Meera, Chen, Hong, Posner, Bruce A, Schmid, Sandra L
Published in PloS one (28.09.2017)
Published in PloS one (28.09.2017)
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Journal Article
Small molecule glucagon release inhibitors with activity in human islets
Kalwat, Michael A, Rodrigues-Dos-Santos, Karina, Binns, Derk D, Wei, Shuguang, Zhou, Anwu, Evans, Matthew R, Posner, Bruce A, Roth, Michael G, Cobb, Melanie H
Published in Frontiers in endocrinology (Lausanne) (19.04.2023)
Published in Frontiers in endocrinology (Lausanne) (19.04.2023)
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Journal Article
Interaction between the autophagy protein Beclin 1 and Na+,K+-ATPase during starvation, exercise, and ischemia
Fernández, Álvaro F, Liu, Yang, Ginet, Vanessa, Shi, Mingjun, Nah, Jihoon, Zou, Zhongju, Zhou, Anwu, Posner, Bruce A, Xiao, Guanghua, Tanguy, Marion, Paradis, Valérie, Sadoshima, Junichi, Rautou, Pierre-Emmanuel, Puyal, Julien, Hu, Ming Chang, Levine, Beth
Published in JCI insight (16.01.2020)
Published in JCI insight (16.01.2020)
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Journal Article
Author Correction: Small-molecule TFEB pathway agonists that ameliorate metabolic syndrome in mice and extend C. elegans lifespan
Wang, Chensu, Niederstrasser, Hanspeter, Douglas, Peter M, Lin, Rueyling, Jaramillo, Juan, Li, Yang, Oswald, Nathaniel W, Zhou, Anwu, McMillan, Elizabeth A, Mendiratta, Saurabh, Wang, Zhaohui, Zhao, Tian, Lin, Zhiqaing, Luo, Min, Huang, Gang, Brekken, Rolf A, Posner, Bruce A, MacMillan, John B, Gao, Jinming, White, Michael A
Published in Nature communications (21.05.2018)
Published in Nature communications (21.05.2018)
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Journal Article
Enhanced HTS Hit Selection via a Local Hit Rate Analysis
Posner, Bruce A, Xi, Hualin, Mills, James E. J
Published in Journal of Chemical Information and Modeling (26.10.2009)
Published in Journal of Chemical Information and Modeling (26.10.2009)
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Journal Article
Targeting ESR1 mutation–induced transcriptional addiction in breast cancer with BET inhibition
Udden, Sm N., Wang, Qian, Kumar, Sunil, Malladi, Venkat S., Wu, Shwu-Yuan, Wei, Shuguang, Posner, Bruce A., Geboers, Sophie, Williams, Noelle S., Liu, Yulun, Sharma, Jayesh K., Mani, Ram S., Malladi, Srinivas, Parra, Karla, Hofstad, Mia, Raj, Ganesh V., Larios, Jose M., Jagsi, Reshma, Wicha, Max S., Park, Ben Ho, Gupta, Gaorav P., Chinnaiyan, Arul M., Chiang, Cheng-Ming, Alluri, Prasanna G.
Published in JCI insight (08.09.2022)
Published in JCI insight (08.09.2022)
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Journal Article
Chromomycin SA analogs from a marine-derived Streptomyces sp
Hu, Youcai, Espindola, Ana Paula D.M., Stewart, Nathan A., Wei, Shuguang, Posner, Bruce A., MacMillan, John B.
Published in Bioorganic & medicinal chemistry (01.09.2011)
Published in Bioorganic & medicinal chemistry (01.09.2011)
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Journal Article
XPO1-dependent nuclear export is a druggable vulnerability in KRAS-mutant lung cancer
Kim, Jimi, McMillan, Elizabeth, Kim, Hyun Seok, Venkateswaran, Niranjan, Makkar, Gurbani, Rodriguez-Canales, Jaime, Villalobos, Pamela, Neggers, Jasper Edgar, Mendiratta, Saurabh, Wei, Shuguang, Landesman, Yosef, Senapedis, William, Baloglu, Erkan, Chow, Chi-Wan B, Frink, Robin E, Gao, Boning, Roth, Michael, Minna, John D, Daelemans, Dirk, Wistuba, Ignacio I, Posner, Bruce A, Scaglioni, Pier Paolo, White, Michael A
Published in Nature (London) (06.10.2016)
Published in Nature (London) (06.10.2016)
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Journal Article
A cholesterol-binding bacterial toxin provides a strategy for identifying a specific Scap inhibitor that blocks lipid synthesis in animal cells
Xu, Shimeng, Smothers, Jared C, Rye, Daphne, Endapally, Shreya, Chen, Hong, Li, Shili, Liang, Guosheng, Kinnebrew, Maia, Rohatgi, Rajat, Posner, Bruce A, Radhakrishnan, Arun
Published in Proceedings of the National Academy of Sciences - PNAS (13.02.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (13.02.2024)
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Journal Article
1,25-Dihydroxyvitamin D 3 enhances glucose-stimulated insulin secretion in mouse and human islets: a role for transcriptional regulation of voltage-gated calcium channels by the vitamin D receptor
Kjalarsdottir, Lilja, Tersey, Sarah A, Vishwanath, Mridula, Chuang, Jen-Chieh, Posner, Bruce A, Mirmira, Raghavendra G, Repa, Joyce J
Published in The Journal of steroid biochemistry and molecular biology (01.01.2019)
Published in The Journal of steroid biochemistry and molecular biology (01.01.2019)
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Journal Article
Improving drug discovery with high-content phenotypic screens by systematic selection of reporter cell lines
Kang, Jungseog, Hsu, Chien-Hsiang, Wu, Qi, Liu, Shanshan, Coster, Adam D, Posner, Bruce A, Altschuler, Steven J, Wu, Lani F
Published in Nature biotechnology (01.01.2016)
Published in Nature biotechnology (01.01.2016)
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