Developing a transition-metal-free green protocol for the electrophilic hydrazination of silyl enol ethers using diazo electrophiles with EtOH-H2O as a safe solvent
Polimera, Subba Rao, Ilangovan, Andivelu, Subbaiah, Murugaiah A. M.
Published in Green chemistry : an international journal and green chemistry resource : GC (20.03.2023)
Published in Green chemistry : an international journal and green chemistry resource : GC (20.03.2023)
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Journal Article
IRAK4 억제제로서 유용한 비시클릭 헤테로아릴 화합물
WU HONG, SANTELLA JOSEPH B, PAIDI VENKATRAM REDDY, POLIMERA SUBBA RAO, HYNES JOHN, NAIR SATHEESH KESAVAN
Year of Publication 15.04.2022
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Year of Publication 15.04.2022
Patent
Developing a transition-metal-free green protocol for the electrophilic hydrazination of silyl enol ethers using diazo electrophiles with EtOH–H 2 O as a safe solvent
Polimera, Subba Rao, Ilangovan, Andivelu, Subbaiah, Murugaiah A. M.
Published in Green chemistry : an international journal and green chemistry resource : GC (20.03.2023)
Published in Green chemistry : an international journal and green chemistry resource : GC (20.03.2023)
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Journal Article
Developing a transition-metal-free green protocol for the electrophilic hydrazination of silyl enol ethers using diazo electrophiles with EtOH-HO as a safe solvent
Polimera, Subba Rao, Ilangovan, Andivelu, Subbaiah, Murugaiah A. M
Published in Green chemistry : an international journal and green chemistry resource : GC (20.03.2023)
Published in Green chemistry : an international journal and green chemistry resource : GC (20.03.2023)
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Journal Article
Examining the Scope of Deriving β‑Aryl Enones from Enol Silanes as Ketone Equivalents via Pd(II)-Mediated Sequential Dehydrosilylation and Arylation
Polimera, Subba Rao, Ilangovan, Andivelu, Subbaiah, Murugaiah A. M.
Published in Journal of organic chemistry (02.06.2023)
Published in Journal of organic chemistry (02.06.2023)
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Journal Article
The Ligand Free Palladium(II)-Catalyzed Regioselective 1,2-Addition of Enol Silanes to Quinones to Access 4‑Hydroxy-4-(2-oxo-2-arylethyl)cyclohexadien-1-ones and Synthetic Applications
Polimera, Subba Rao, A. M. Subbaiah, Murugaiah, Ilangovan, Andivelu
Published in Journal of organic chemistry (05.11.2021)
Published in Journal of organic chemistry (05.11.2021)
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Journal Article
헤테로아릴 치환된 아미노피리딘 화합물
DUNCIA JOHN V, SANTELLA JOSEPH B, WU HONG, POLIMERA SUBBA RAO, MACOR JOHN E, NAIR SATHEESH KESAVAN, SISTLA RAMESH KUMAR, RATNA KUMAR SREEKANTHA, SARKUNAM KANDHASAMY, PAIDI VENKATRAM REDDY, GARDNER DANIEL S, MURUGESAN NATESSAN, HYNES JOHN, KANTHETI DURGARAO
Year of Publication 26.02.2019
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Year of Publication 26.02.2019
Patent
Synthetic Access to α‑Oxoketene Aminals by the Nucleophilic Addition of Enol Silane-Derived Palladium(II) Enolates to Carbodiimides
Polimera, Subba Rao, Ilangovan, Andivelu, Meanwell, Nicholas A., Subbaiah, Murugaiah A. M.
Published in Journal of organic chemistry (04.11.2022)
Published in Journal of organic chemistry (04.11.2022)
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Journal Article
Optimization of Nicotinamides as Potent and Selective IRAK4 Inhibitors with Efficacy in a Murine Model of Psoriasis
Nair, Satheesh, Kumar, Sreekantha Ratna, Paidi, Venkatram Reddy, Sistla, Ramesh, Kantheti, Durgarao, Polimera, Subba Rao, Thangavel, Soodamani, Mukherjee, Amrita Jha, Das, Mitalee, Bhide, Rajeev S, Pitts, William J, Murugesan, Natesan, Dudhgoankar, Shailesh, Nagar, Jignesh, Subramani, Siva, Mazumder, Debarati, Carman, Julie A, Holloway, Deborah A, Li, Xin, Fereshteh, Mark P, Ruepp, Stefan, Palanisamy, Kamalavenkatesh, Mariappan, T. Thanga, Maddi, Srinivas, Saxena, Ajay, Elzinga, Paul, Chimalakonda, Anjaneya, Ruan, Qian, Ghosh, Kaushik, Bose, Sucharita, Sack, John, Yan, Chunhong, Kiefer, Susan E, Xie, Dianlin, Newitt, John A, Saravanakumar, S. Pon, Rampulla, Richard A, Barrish, Joel C, Carter, Percy H, Hynes, John
Published in ACS medicinal chemistry letters (09.07.2020)
Published in ACS medicinal chemistry letters (09.07.2020)
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Journal Article
BICYCLIC HETEROARYL COMPOUNDS USEFUL AS IRAK4 INHIBITORS
Nair, Satheesh Kesavan, Santella, Joseph B, Hynes, John, Wu, Hong, Polimera, Subba Rao, Paidi, Venkatram Reddy
Year of Publication 01.12.2022
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Year of Publication 01.12.2022
Patent
BICYCLIC HETEROARYL COMPOUNDS USEFUL AS IRAK4 INHIBITORS
POLIMERA, Subba Rao, PAIDI, Venkatram Reddy, WU, Hong, SANTELLA, Joseph B, NAIR, Satheesh Kesavan, HYNES, John
Year of Publication 22.06.2022
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Year of Publication 22.06.2022
Patent
BICYCLIC HETEROARYL COMPOUNDS USEFUL AS IRAK4 INHIBITORS
POLIMERA, Subba Rao, PAIDI, Venkatram Reddy, WU, Hong, SANTELLA, Joseph B, NAIR, Satheesh Kesavan, HYNES, John
Year of Publication 24.03.2022
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Year of Publication 24.03.2022
Patent
HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS
SARKUNAM, Kandhasamy, POLIMERA, Subba Rao, PAIDI, Venkatram Reddy, DUNCIA, John V, SANTELLA, Joseph B, WU, Hong, GARDNER, Daniel S, NAIR, Satheesh Kesavan, MACOR, John E, HYNES, John, SISTLA, Ramesh Kumar
Year of Publication 26.08.2020
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Year of Publication 26.08.2020
Patent
Heteroaryl substituted aminopyridine compounds
Santella, Joseph B, Sarkunam, Kandhasamy, Murugesan, Natesan, Kumar, Sreekantha Ratna, Sistla, Ramesh Kumar, Nair, Satheesh Kesavan, Hynes, John, Gardner, Daniel S, Wu, Hong, Polimera, Subba Rao, Paidi, Venkatram Reddy, Macor, John E, Duncia, John V, Kantheti, Durgarao
Year of Publication 14.04.2020
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Year of Publication 14.04.2020
Patent
HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS
POLIMERA, Subba Rao, SANTELLA, Joseph B, WU, Hong, NAIR, Satheesh Kesavan, MURUGESAN, Natessan, SISTLA, Ramesh Kumar, SARKUNAM, Kandhasamy, PAIDI, Venkatram Reddy, DUNCIA, John V, GARDNER, Daniel S, KANTHETI, Durgarao, RATNA KUMAR, Sreekantha, MACOR, John E, HYNES, John
Year of Publication 26.02.2020
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Year of Publication 26.02.2020
Patent
HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS
Santella, Joseph B, Sarkunam, Kandhasamy, Murugesan, Natesan, Kumar, Sreekantha Ratna, Sistla, Ramesh Kumar, Nair, Satheesh Kesavan, Hynes, John, Gardner, Daniel S, Wu, Hong, Polimera, Subba Rao, Paidi, Venkatram Reddy, Macor, John E, Duncia, John V, Kantheti, Durgarao
Year of Publication 26.09.2019
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Year of Publication 26.09.2019
Patent
HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS
POLIMERA, Subba Rao, SANTELLA, Joseph B, WU, Hong, NAIR, Satheesh Kesavan, MURUGESAN, Natessan, SISTLA, Ramesh Kumar, SARKUNAM, Kandhasamy, PAIDI, Venkatram Reddy, DUNCIA, John V, GARDNER, Daniel S, KANTHETI, Durgarao, RATNA KUMAR, Sreekantha, MACOR, John E, HYNES, John
Year of Publication 01.05.2019
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Year of Publication 01.05.2019
Patent
Bicyclic heteroaryl compounds useful as IRAK4 inhibitors
WU HONG, SANTELLA JOSEPH B, PAIDI VENKATRAM REDDY, POLIMERA SUBBA RAO, HYNES JOHN, NAIR SATHEESH KESAVAN
Year of Publication 18.03.2022
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Year of Publication 18.03.2022
Patent
Heteroaryl substituted aminopyridine compounds
Nair, Satheesh Kesavan, Santella, Joseph B, Sarkunam, Kandhasamy, Hynes, John, Gardner, Daniel S, Polimera, Subba Rao, Wu, Hong, Paidi, Venkatram Reddy, Sistla, Ramesh Kumar, Macor, John E, Duncia, John V
Year of Publication 12.02.2019
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Year of Publication 12.02.2019
Patent
HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS
Nair, Satheesh Kesavan, Santella, Joseph B, Sarkunam, Kandhasamy, Hynes, John, DUNCIA, John V, Gardner, Daniel S, Polimera, Subba Rao, Wu, Hong, Paidi, Venkatram Reddy, Sistla, Ramesh Kumar, Macor, John E
Year of Publication 28.06.2018
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Year of Publication 28.06.2018
Patent