Peptide Ligands Stabilized by Small Molecules
Chen, Shiyu, Bertoldo, Davide, Angelini, Alessandro, Pojer, Florence, Heinis, Christian
Published in Angewandte Chemie (International ed.) (03.02.2014)
Published in Angewandte Chemie (International ed.) (03.02.2014)
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Journal Article
Internalization and vacuolar targeting of the brassinosteroid hormone receptor BRI1 are regulated by ubiquitination
Martins, Sara, Dohmann, Esther M N, Cayrel, Anne, Johnson, Alexander, Fischer, Wolfgang, Pojer, Florence, Satiat-Jeunemaître, Béatrice, Jaillais, Yvon, Chory, Joanne, Geldner, Niko, Vert, Grégory
Published in Nature communications (21.01.2015)
Published in Nature communications (21.01.2015)
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Cryo-EM structures and binding of mouse and human ACE2 to SARS-CoV-2 variants of concern indicate that mutations enabling immune escape could expand host range
Ni, Dongchun, Turelli, Priscilla, Beckert, Bertrand, Nazarov, Sergey, Uchikawa, Emiko, Myasnikov, Alexander, Pojer, Florence, Trono, Didier, Stahlberg, Henning, Lau, Kelvin
Published in PLoS pathogens (01.04.2023)
Published in PLoS pathogens (01.04.2023)
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Journal Article
Selective inhibition of STAT3 signaling using monobodies targeting the coiled-coil and N-terminal domains
La Sala, Grégory, Michiels, Camille, Kükenshöner, Tim, Brandstoetter, Tania, Maurer, Barbara, Koide, Akiko, Lau, Kelvin, Pojer, Florence, Koide, Shohei, Sexl, Veronika, Dumoutier, Laure, Hantschel, Oliver
Published in Nature communications (17.08.2020)
Published in Nature communications (17.08.2020)
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Journal Article
Palmitoylated acyl protein thioesterase APT2 deforms membranes to extract substrate acyl chains
Abrami, Laurence, Audagnotto, Martina, Ho, Sylvia, Marcaida, Maria Jose, Mesquita, Francisco S, Anwar, Muhammad U, Sandoz, Patrick A, Fonti, Giulia, Pojer, Florence, Dal Peraro, Matteo, van der Goot, F Gisou
Published in Nature chemical biology (01.04.2021)
Published in Nature chemical biology (01.04.2021)
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A high-throughput cell- and virus-free assay shows reduced neutralization of SARS-CoV-2 variants by COVID-19 convalescent plasma
Fenwick, Craig, Turelli, Priscilla, Pellaton, Céline, Farina, Alex, Campos, Jérémy, Raclot, Charlène, Pojer, Florence, Cagno, Valeria, Nusslé, Semira Gonseth, D'Acremont, Valerie, Fehr, Jan, Puhan, Milo, Pantaleo, Giuseppe, Trono, Didier
Published in Science Translational Medicine (04.08.2021)
Published in Science Translational Medicine (04.08.2021)
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Towards a new combination therapy for tuberculosis with next generation benzothiazinones
Makarov, Vadim, Lechartier, Benoit, Zhang, Ming, Neres, João, Sar, Astrid M, Raadsen, Susanne A, Hartkoorn, Ruben C, Ryabova, Olga B, Vocat, Anthony, Decosterd, Laurent A, Widmer, Nicolas, Buclin, Thierry, Bitter, Wilbert, Andries, Koen, Pojer, Florence, Dyson, Paul J, Cole, Stewart T
Published in EMBO molecular medicine (01.03.2014)
Published in EMBO molecular medicine (01.03.2014)
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Journal Article
Btk SH2-kinase interface is critical for allosteric kinase activation and its targeting inhibits B-cell neoplasms
Duarte, Daniel P, Lamontanara, Allan J, La Sala, Giuseppina, Jeong, Sukyo, Sohn, Yoo-Kyoung, Panjkovich, Alejandro, Georgeon, Sandrine, Kükenshöner, Tim, Marcaida, Maria J, Pojer, Florence, De Vivo, Marco, Svergun, Dmitri, Kim, Hak-Sung, Dal Peraro, Matteo, Hantschel, Oliver
Published in Nature communications (08.05.2020)
Published in Nature communications (08.05.2020)
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Evolution of the chalcone―isomerase fold from fatty―acid binding to stereospecific catalysis
NGAKI, Micheline N, LOUIE, Gordon V, PHILIPPE, Ryan N, MANNING, Gerard, POJER, Florence, BOWMAN, Marianne E, LING LI, LARSEN, Elise, SYRKIN WURTELE, Eve, NOEL, Joseph P
Published in Nature (London) (24.05.2012)
Published in Nature (London) (24.05.2012)
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Journal Article
Dithiol amino acids can structurally shape and enhance the ligand-binding properties of polypeptides
Chen, Shiyu, Gopalakrishnan, Ranganath, Schaer, Tifany, Marger, Fabrice, Hovius, Ruud, Bertrand, Daniel, Pojer, Florence, Heinis, Christian
Published in Nature chemistry (01.11.2014)
Published in Nature chemistry (01.11.2014)
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Journal Article
Author Correction: Internalization and vacuolar targeting of the brassinosteroid hormone receptor BRI1 are regulated by ubiquitination
Martins, Sara, Dohmann, Esther M N, Cayrel, Anne, Johnson, Alexander, Fischer, Wolfgang, Pojer, Florence, Satiat-Jeunemaître, Béatrice, Jaillais, Yvon, Chory, Joanne, Geldner, Niko, Vert, Grégory
Published in Nature communications (17.05.2021)
Published in Nature communications (17.05.2021)
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Journal Article
Rapid Synthesis of Auxin via a New Tryptophan-Dependent Pathway Is Required for Shade Avoidance in Plants
Tao, Yi, Ferrer, Jean-Luc, Ljung, Karin, Pojer, Florence, Hong, Fangxin, Long, Jeff A., Li, Lin, Moreno, Javier E., Bowman, Marianne E., Ivans, Lauren J., Cheng, Youfa, Lim, Jason, Zhao, Yunde, Ballaré, Carlos L., Sandberg, Göran, Noel, Joseph P., Chory, Joanne
Published in Cell (04.04.2008)
Published in Cell (04.04.2008)
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Discovery and characterization of a marine bacterial SAM-dependent chlorinase
Moore, Bradley S, Eustáquio, Alessandra S, Pojer, Florence, Noel, Joseph P
Published in Nature chemical biology (01.01.2008)
Published in Nature chemical biology (01.01.2008)
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Journal Article
Towards a new tuberculosis drug: pyridomycin – nature's isoniazid
Hartkoorn, Ruben C., Sala, Claudia, Neres, João, Pojer, Florence, Magnet, Sophie, Mukherjee, Raju, Uplekar, Swapna, Boy‐Röttger, Stefanie, Altmann, Karl‐Heinz, Cole, Stewart T.
Published in EMBO molecular medicine (01.10.2012)
Published in EMBO molecular medicine (01.10.2012)
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Journal Article
A highly potent antibody effective against SARS-CoV-2 variants of concern
Fenwick, Craig, Turelli, Priscilla, Perez, Laurent, Pellaton, Céline, Esteves-Leuenberger, Line, Farina, Alex, Campos, Jérémy, Lana, Erica, Fiscalini, Flurin, Raclot, Charlène, Pojer, Florence, Lau, Kelvin, Demurtas, Davide, Descatoire, Marc, Joo, Victor S., Foglierini, Mathilde, Noto, Alessandra, Abdelnabi, Rana, Foo, Caroline S., Vangeel, Laura, Neyts, Johan, Du, Wenjuan, Bosch, Berend-Jan, Veldman, Geertruida, Leyssen, Pieter, Thiel, Volker, LeGrand, Roger, Lévy, Yves, Trono, Didier, Pantaleo, Giuseppe
Published in Cell reports (Cambridge) (12.10.2021)
Published in Cell reports (Cambridge) (12.10.2021)
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Structural and functional dissection of the DH and PH domains of oncogenic Bcr-Abl tyrosine kinase
Reckel, Sina, Gehin, Charlotte, Tardivon, Delphine, Georgeon, Sandrine, Kükenshöner, Tim, Löhr, Frank, Koide, Akiko, Buchner, Lena, Panjkovich, Alejandro, Reynaud, Aline, Pinho, Sara, Gerig, Barbara, Svergun, Dmitri, Pojer, Florence, Güntert, Peter, Dötsch, Volker, Koide, Shohei, Gavin, Anne-Claude, Hantschel, Oliver
Published in Nature communications (13.12.2017)
Published in Nature communications (13.12.2017)
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Journal Article
A rheostat mechanism governs the bifurcation of carbon flux in mycobacteria
Murima, Paul, Zimmermann, Michael, Chopra, Tarun, Pojer, Florence, Fonti, Giulia, Dal Peraro, Matteo, Alonso, Sylvie, Sauer, Uwe, Pethe, Kevin, McKinney, John D
Published in Nature communications (24.08.2016)
Published in Nature communications (24.08.2016)
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Journal Article
Structure-based optimization of type III indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors
Röhrig, Ute F., Majjigapu, Somi Reddy, Vogel, Pierre, Reynaud, Aline, Pojer, Florence, Dilek, Nahzli, Reichenbach, Patrick, Ascenção, Kelly, Irving, Melita, Coukos, George, Michielin, Olivier, Zoete, Vincent
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2022)
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2022)
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