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Gorski, Judith N, Pachanski, Michele J, Mane, Joel, Plummer, Christopher W, Souza, Sarah, Thomas-Fowlkes, Brande S, Ogawa, Aimie M, Weinglass, Adam B, Di Salvo, Jerry, Cheewatrakoolpong, Boonlert, Howard, Andrew D, Colletti, Steven L, Trujillo, Maria E
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Published in American journal of physiology: endocrinology and metabolism (01.07.2017)
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Structure–Activity Relationship of Novel and Selective Biaryl-Chroman GPR40 AgoPAMs
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Published in ACS medicinal chemistry letters (12.07.2018)
Published in ACS medicinal chemistry letters (12.07.2018)
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Design, Development, Mechanistic Elucidation, and Rational Optimization of a Tandem Ireland Claisen/Cope Rearrangement Reaction for Rapid Access to the (Iso)Cyclocitrinol Core
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Enantioselective Synthesis of α‑Methyl-β-cyclopropyldihydrocinnamates
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Published in Journal of organic chemistry (05.02.2016)
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GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent
Pachanski, Michele J, Kirkland, Melissa E, Kosinski, Daniel T, Mane, Joel, Cheewatrakoolpong, Boonlert, Xue, Jiyan, Szeto, Daphne, Forrest, Gail, Miller, Corin, Bunzel, Michelle, Plummer, Christopher W, Chobanian, Harry R, Miller, Michael W, Souza, Sarah, Thomas-Fowlkes, Brande S, Ogawa, Aimie M, Weinglass, Adam B, Di Salvo, Jerry, Li, Xiaoyan, Feng, Yue, Tatosian, Daniel A, Howard, Andrew D, Colletti, Steven L, Trujillo, Maria E
Published in PloS one (20.10.2017)
Published in PloS one (20.10.2017)
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Correction to “Design, Development, Mechanistic Elucidation, and Rational Optimization of a Tandem Ireland Claisen/Cope Rearrangement Reaction for Rapid Access to the (Iso)Cyclocitrinol Core”
Plummer, Christopher W, Wei, Carolyn S, Yozwiak, Carrie E, Soheili, Arash, Smithback, Sara O, Leighton, James L
Published in Journal of the American Chemical Society (28.10.2015)
Published in Journal of the American Chemical Society (28.10.2015)
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Design and Synthesis of Novel, Selective GPR40 AgoPAMs
Plummer, Christopher W., Clements, Matthew J., Chen, Helen, Rajagopalan, Murali, Josien, Hubert, Hagmann, William K., Miller, Michael, Trujillo, Maria E., Kirkland, Melissa, Kosinski, Daniel, Mane, Joel, Pachanski, Michele, Cheewatrakoolpong, Boonlert, Nolting, Andrew F., Orr, Robert, Christensen, Melodie, Campeau, Louis-Charles, Wright, Michael J., Bugianesi, Randal, Souza, Sarah, Zhang, Xiaoping, Di Salvo, Jerry, Weinglass, Adam B., Tschirret-Guth, Richard, Nargund, Ravi, Howard, Andrew D., Colletti, Steven L.
Published in ACS medicinal chemistry letters (09.02.2017)
Published in ACS medicinal chemistry letters (09.02.2017)
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Synthesis and activity of 4,5-diarylimidazoles as human CB1 receptor inverse agonists
Plummer, Christopher W., Finke, Paul E., Mills, Sander G., Wang, Junying, Tong, Xinchun, Doss, George A., Fong, Tung M., Lao, Julie Z., Schaeffer, Marie-Therese, Chen, Jing, Shen, Chun-Pyn, Stribling, D. Sloan, Shearman, Lauren P., Strack, Alison M., Van der Ploeg, Lex H.T.
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
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Characterization of a novel and selective cannabinoid CB1 receptor inverse agonist, Imidazole 24b, in rodents
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Published in European journal of pharmacology (28.01.2008)
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Year of Publication 06.08.2021
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WANG HUIJUN, SWAMINATHAN UMA, ALI AMJAD, LARSEN MATTHEW A, LIU PING, PAN JIANPING, DENG QIAOLIN, MANSOOR UMAR FARUK, LIU KUN, CUMMING JARED, DEMONG DUANE, PLUMMER CHRISTOPHER W, SATHER AARON, ZHANG YONGLIAN, GRAHAM THOMAS H, HOOVER ANDREW J, HENNESSY ELISABETH
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Year of Publication 04.08.2021
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치환된 아미노 트리아졸로피리미딘 및 아미노 트리아졸로피라진 아데노신 수용체 길항제, 제약 조성물 및 그의 용도
WANG HUIJUN, ALI AMJAD, DENG QIAOLIN, CUMMING JARED, KUANG RONGZE, DEMONG DUANE, RICO DUQUE JENNY LORENA, BRILL ZACHARY G, PLUMMER CHRISTOPHER W, ZHANG YONGLIAN, GRAHAM THOMAS H, LIM YEON HEE, ZHAO KAKE
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Year of Publication 28.07.2021
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PAN WEIDONG, LIU WEIGUO, BROCKUNIER LINDA, ZANG YI, JIANG JINLONG, TANG HAIFENG, BIFTU TESFAYE, WANG HONGWU, HUANG XIANHAI, OGAWA ANTHONY, PARK MIN, CHEN HELEN, PLUMMER CHRISTOPHER W, MAL RUDRAJIT, GUO YAN, DING FA XIANG, SUN WANYING
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Year of Publication 22.08.2018
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Structural basis for the cooperative allosteric activation of the free fatty acid receptor GPR40
Lu, Jun, Byrne, Noel, Wang, John, Bricogne, Gerard, Brown, Frank K, Chobanian, Harry R, Colletti, Steven L, Di Salvo, Jerry, Thomas-Fowlkes, Brande, Guo, Yan, Hall, Dawn L, Hadix, Jennifer, Hastings, Nicholas B, Hermes, Jeffrey D, Ho, Thu, Howard, Andrew D, Josien, Hubert, Kornienko, Maria, Lumb, Kevin J, Miller, Michael W, Patel, Sangita B, Pio, Barbara, Plummer, Christopher W, Sherborne, Bradley S, Sheth, Payal, Souza, Sarah, Tummala, Srivanya, Vonrhein, Clemens, Webb, Maria, Allen, Samantha J, Johnston, Jennifer M, Weinglass, Adam B, Sharma, Sujata, Soisson, Stephen M
Published in Nature structural & molecular biology (01.07.2017)
Published in Nature structural & molecular biology (01.07.2017)
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ANTIDIABETIC TRICYCLIC COMPOUNDS
BLIZZARD TIMOTHY A, HAGMANN WILLIAM K, NAIR ANILKUMAR G, FRIE JESSICA L, CHEN ZHENGXIA, BIFU TESFAYE, JOSIEN HUBERT, ZHU CHENG, CUI MINGXIANG, BIJU PURAKKATTLE, PLUMMER CHRISTOPHER W, CLEMENTS MATTHEW J, HU BIN
Year of Publication 16.01.2017
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Year of Publication 16.01.2017
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ANTIDIABETIC BICYCLIC COMPOUNDS
CHOBANIAN HARRY R, HAGMANN WILLIAM K, MARCANTONIO KAREN M, XIAO DONG, CRESPO ALEJANDRO, DEMONG DUANE E, MILLER MICHAEL, PIO BARBARA, BROCKUNIER LINDA L, CHEN HELEN, PLUMMER CHRISTOPHER W, GUO YAN, CLEMENTS MATTHEW J
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Year of Publication 21.10.2015
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A Modular Synthesis of 2-Alkyl- and 2-Arylchromans via a Three-Step Sequence
Orr, Robert K., Campeau, Louis-Charles, Chobanian, Harry R., Dunn, Jamie M. McCabe, Pio, Barbara, Plummer, Christopher W., Nolting, Andrew, Ruck, Rebecca T.
Published in Synthesis (Stuttgart) (01.02.2017)
Published in Synthesis (Stuttgart) (01.02.2017)
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ChemInform Abstract: Design, Development, Mechanistic Elucidation, and Rational Optimization of a Tandem Ireland Claisen/Cope Rearrangement Reaction for Rapid Access to the (Iso)Cyclocitrinol Core
Plummer, Christopher W., Wei, Carolyn S., Yozwiak, Carrie E., Soheili, Arash, Smithback, Sara O., Leighton, James L.
Published in ChemInform (01.02.2015)
Published in ChemInform (01.02.2015)
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Characterization of a novel and selective cannabinoid CB 1 receptor inverse agonist, Imidazole 24b, in rodents
Shearman, Lauren P., Stribling, D. Sloan, Camacho, Ramon E., Rosko, Kimberly M., Wang, Junying, Tong, Sharon, Feng, Yue, Marsh, Donald J., Yu, Hong, Guan, Xiaoming, Spann, Stephanie K., MacNeil, Douglas J., Fong, Tung M., Metzger, Joseph M., Goulet, Mark T., Hagmann, William K., Plummer, Christopher W., Finke, Paul E., Mills, Sander G., Shah, Shrenik K., Truong, Quang, Van der Ploeg, L.H.T., MacIntyre, D. Euan, Strack, Alison M.
Published in European journal of pharmacology (2008)
Published in European journal of pharmacology (2008)
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