Regulation of pulmonary surfactant by the adhesion GPCR GPR116/ADGRF5 requires a tethered agonist-mediated activation mechanism
Bridges, James P, Safina, Caterina, Pirard, Bernard, Brown, Kari, Filuta, Alyssa, Panchanathan, Ravichandran, Bouhelal, Rochdi, Reymann, Nicole, Patel, Sejal, Seuwen, Klaus, Miller, William E, Ludwig, Marie-Gabrielle
Published in eLife (08.09.2022)
Published in eLife (08.09.2022)
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Binding site of a novel Kv1.5 blocker: a "foot in the door" against atrial fibrillation
Decher, Niels, Kumar, Pradeep, Gonzalez, Teresa, Pirard, Bernard, Sanguinetti, Michael C
Published in Molecular pharmacology (01.10.2006)
Published in Molecular pharmacology (01.10.2006)
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Molecular Basis for Kv1.5 Channel Block
Decher, Niels, Pirard, Bernard, Bundis, Florian, Peukert, Stefan, Baringhaus, Karl-Heinz, Busch, Andreas E., Steinmeyer, Klaus, Sanguinetti, Michael C.
Published in The Journal of biological chemistry (02.01.2004)
Published in The Journal of biological chemistry (02.01.2004)
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5,5- and 5,6-Membered Spirocyclic Indolinone Hit-Finding Libraries
Meier, Peter, Battaglia, Nicole, Ertl, Peter, Pirard, Bernard
Published in ACS combinatorial science (08.07.2019)
Published in ACS combinatorial science (08.07.2019)
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Structural Basis for the Highly Selective Inhibition of MMP-13
Engel, Christian K., Pirard, Bernard, Schimanski, Sandra, Kirsch, Reinhard, Habermann, Jörg, Klingler, Otmar, Schlotte, Volkhard, Weithmann, Klaus Ulrich, Wendt, K. Ulrich
Published in Chemistry & biology (01.02.2005)
Published in Chemistry & biology (01.02.2005)
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Building Compound Archives for the Future
Lewis, Richard, Deheuvels, Joakim, Ertl, Peter, Pirard, Bernard, Sirockin, Finton
Published in Molecular informatics (01.12.2016)
Published in Molecular informatics (01.12.2016)
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New pyrazolo[1,5a]pyrimidines as orally active inhibitors of Lck
Gommermann, Nina, Buehlmayer, Peter, von Matt, Anette, Breitenstein, Werner, Masuya, Keiichi, Pirard, Bernard, Furet, Pascal, Cowan-Jacob, Sandra W., Weckbecker, Gisbert
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
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Molecular basis for Kv1.5 channel block: conservation of drug binding sites among voltage-gated K+ channels
Decher, Niels, Pirard, Bernard, Bundis, Florian, Peukert, Stefan, Baringhaus, Karl-Heinz, Busch, Andreas E, Steinmeyer, Klaus, Sanguinetti, Michael C
Published in The Journal of biological chemistry (02.01.2004)
Published in The Journal of biological chemistry (02.01.2004)
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Identification, Synthesis, and Activity of Novel Blockers of the Voltage-Gated Potassium Channel Kv1.5
Peukert, Stefan, Brendel, Joachim, Pirard, Bernard, Brüggemann, Andrea, Below, Peter, Kleemann, Heinz-Werner, Hemmerle, Horst, Schmidt, Wolfgang
Published in Journal of medicinal chemistry (13.02.2003)
Published in Journal of medicinal chemistry (13.02.2003)
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Pharmacophore-based search, synthesis, and biological evaluation of anthranilic amides as novel blockers of the Kv1.5 channel
Peukert, Stefan, Brendel, Joachim, Pirard, Bernard, Strübing, Carsten, Kleemann, Heinz-Werner, Böhme, Thomas, Hemmerle, Horst
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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