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Year of Publication 28.06.2024
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Year of Publication 21.06.2024
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Year of Publication 21.06.2024
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Year of Publication 28.06.2024
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Year of Publication 28.06.2024
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ZHU YEHENG, ORWAT MICHAEL J, DILGER ANDREW K, EWING WILLIAM R, PINTO DONALD J.P
Year of Publication 02.04.2018
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Year of Publication 02.04.2018
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Discovery of Milvexian, a High-Affinity, Orally Bioavailable Inhibitor of Factor XIa in Clinical Studies for Antithrombotic Therapy
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XIa PYRIMIDINONES AS FACTOR XIA INHIBITORS
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Year of Publication 27.11.2018
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Year of Publication 27.11.2018
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SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS AS FACTOR XIA INHIBITORS
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Year of Publication 17.07.2014
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Year of Publication 17.07.2014
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Factor XIa Inhibitors as New Anticoagulants
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Preclinical discovery of apixaban, a direct and orally bioavailable factor Xa inhibitor
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XIa PYRIMIDINONES AS FACTOR XIA INHIBITORS
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Year of Publication 24.05.2017
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Year of Publication 24.05.2017
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Factor Xa Inhibitors: Next-Generation Antithrombotic Agents
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Discovery of 1-(4-Methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro- 1H-pyrazolo[3,4-c]pyridine-3-carboxamide (Apixaban, BMS-562247), a Highly Potent, Selective, Efficacious, and Orally Bioavailable Inhibitor of Blood Coagulation Factor Xa
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Potent, Orally Bioavailable, and Efficacious Macrocyclic Inhibitors of Factor XIa. Discovery of Pyridine-Based Macrocycles Possessing Phenylazole Carboxamide P1 Groups
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Published in Journal of medicinal chemistry (23.01.2020)
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Structure-Based Design of Macrocyclic Factor XIa Inhibitors: Discovery of the Macrocyclic Amide Linker
Corte, James R, Fang, Tianan, Osuna, Honey, Pinto, Donald J. P, Rossi, Karen A, Myers, Joseph E, Sheriff, Steven, Lou, Zhen, Zheng, Joanna J, Harper, Timothy W, Bozarth, Jeffrey M, Wu, Yiming, Luettgen, Joseph M, Seiffert, Dietmar A, Decicco, Carl P, Wexler, Ruth R, Quan, Mimi L
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Discovery of a Parenteral Small Molecule Coagulation Factor XIa Inhibitor Clinical Candidate (BMS-962212)
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Published in Journal of medicinal chemistry (14.12.2017)
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Chemistry and pharmacokinetics of diarylthiophenes and terphenyls as selective COX-2 inhibitors
Pinto, Donald J.P., Copeland, Robert A., Covington, Maryanne B., Pitts, William J., Batt, Douglas G., Orwat, Michael J., Lam, Gilbert N., Joshi, Amita, Chan, Yuk-Charn, Wang, Shuaige, Trzaskos, James M., Magolda, Ronald L., Kornhauser, David M.
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
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