new approach to analyze cell surface protein complexes reveals specific heterodimeric metabotropic glutamate receptors
Doumazane, Etienne, Scholler, Pauline, Zwier, Jurriaan M, Eric, Trinquet, Rondard, Philippe, Pin, Jean-Philippe
Published in The FASEB journal (01.01.2011)
Published in The FASEB journal (01.01.2011)
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SGIP1 modulates kinetics and interactions of the cannabinoid receptor 1 and G protein‐coupled receptor kinase 3 signalosome
Gazdarica, Matej, Noda, Judith, Durydivka, Oleh, Novosadova, Vendula, Mackie, Ken, Pin, Jean‐Philippe, Prezeau, Laurent, Blahos, Jaroslav
Published in Journal of neurochemistry (01.03.2022)
Published in Journal of neurochemistry (01.03.2022)
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G protein-coupled receptor oligomerization revisited: functional and pharmacological perspectives
Ferré, Sergi, Casadó, Vicent, Devi, Lakshmi A, Filizola, Marta, Jockers, Ralf, Lohse, Martin J, Milligan, Graeme, Pin, Jean-Philippe, Guitart, Xavier
Published in Pharmacological reviews (01.04.2014)
Published in Pharmacological reviews (01.04.2014)
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Sensing of Amino Acids in a Dopaminergic Circuitry Promotes Rejection of an Incomplete Diet in Drosophila
Bjordal, Marianne, Arquier, Nathalie, Kniazeff, Julie, Pin, Jean Philippe, Léopold, Pierre
Published in Cell (30.01.2014)
Published in Cell (30.01.2014)
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Structural basis of the activation of a metabotropic GABA receptor
Shaye, Hamidreza, Ishchenko, Andrii, Lam, Jordy Homing, Han, Gye Won, Xue, Li, Rondard, Philippe, Pin, Jean-Philippe, Katritch, Vsevolod, Gati, Cornelius, Cherezov, Vadim
Published in Nature (London) (13.08.2020)
Published in Nature (London) (13.08.2020)
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Allosteric modulators enhance agonist efficacy by increasing the residence time of a GPCR in the active state
Cao, Anne-Marinette, Quast, Robert B., Fatemi, Fataneh, Rondard, Philippe, Pin, Jean-Philippe, Margeat, Emmanuel
Published in Nature communications (14.09.2021)
Published in Nature communications (14.09.2021)
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Generic GPCR residue numbers – aligning topology maps while minding the gaps
Isberg, Vignir, de Graaf, Chris, Bortolato, Andrea, Cherezov, Vadim, Katritch, Vsevolod, Marshall, Fiona H, Mordalski, Stefan, Pin, Jean-Philippe, Stevens, Raymond C, Vriend, Gerrit, Gloriam, David E
Published in Trends in pharmacological sciences (Regular ed.) (01.01.2015)
Published in Trends in pharmacological sciences (Regular ed.) (01.01.2015)
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Structures of human mGlu2 and mGlu7 homo- and heterodimers
Du, Juan, Wang, Dejian, Fan, Hongcheng, Xu, Chanjuan, Tai, Linhua, Lin, Shuling, Han, Shuo, Tan, Qiuxiang, Wang, Xinwei, Xu, Tuo, Zhang, Hui, Chu, Xiaojing, Yi, Cuiying, Liu, Peng, Wang, Xiaomei, Zhou, Yu, Pin, Jean-Philippe, Rondard, Philippe, Liu, Hong, Liu, Jianfeng, Sun, Fei, Wu, Beili, Zhao, Qiang
Published in Nature (London) (24.06.2021)
Published in Nature (London) (24.06.2021)
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Dimers and beyond: The functional puzzles of class C GPCRs
Kniazeff, Julie, Prézeau, Laurent, Rondard, Philippe, Pin, Jean-Philippe, Goudet, Cyril
Published in Pharmacology & therapeutics (Oxford) (01.04.2011)
Published in Pharmacology & therapeutics (Oxford) (01.04.2011)
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Biased signaling due to oligomerization of the G protein-coupled platelet-activating factor receptor
Liu, Junke, Tang, Hengmin, Xu, Chanjuan, Zhou, Shengnan, Zhu, Xunying, Li, Yuanyuan, Prézeau, Laurent, Xu, Tao, Pin, Jean-Philippe, Rondard, Philippe, Ji, Wei, Liu, Jianfeng
Published in Nature communications (26.10.2022)
Published in Nature communications (26.10.2022)
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Journal Article
Distinct roles of metabotropic glutamate receptor dimerization in agonist activation and G-protein coupling
El Moustaine, Driss, Granier, Sébastien, Doumazane, Etienne, Scholler, Pauline, Rahmeh, Rita, Bron, Patrick, Mouillac, Bernard, Banères, Jean-Louis, Rondard, Philippe, Pin, Jean-Philippe
Published in Proceedings of the National Academy of Sciences - PNAS (02.10.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (02.10.2012)
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Rearrangement of the transmembrane domain interfaces associated with the activation of a GPCR hetero-oligomer
Xue, Li, Sun, Qian, Zhao, Han, Rovira, Xavier, Gai, Siyu, He, Qianwen, Pin, Jean-Philippe, Liu, Jianfeng, Rondard, Philippe
Published in Nature communications (24.06.2019)
Published in Nature communications (24.06.2019)
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International Union of Basic and Clinical Pharmacology. XC. multisite pharmacology: recommendations for the nomenclature of receptor allosterism and allosteric ligands
Christopoulos, Arthur, Changeux, Jean-Pierre, Catterall, William A, Fabbro, Doriano, Burris, Thomas P, Cidlowski, John A, Olsen, Richard W, Peters, John A, Neubig, Richard R, Pin, Jean-Philippe, Sexton, Patrick M, Kenakin, Terry P, Ehlert, Frederick J, Spedding, Michael, Langmead, Christopher J
Published in Pharmacological reviews (01.10.2014)
Published in Pharmacological reviews (01.10.2014)
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Specific pharmacological and Gi/o protein responses of some native GPCRs in neurons
Xu, Chanjuan, Zhou, Yiwei, Liu, Yuxuan, Lin, Li, Liu, Peng, Wang, Xiaomei, Xu, Zhengyuan, Pin, Jean-Philippe, Rondard, Philippe, Liu, Jianfeng
Published in Nature communications (05.03.2024)
Published in Nature communications (05.03.2024)
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Journal Article
Illuminating the activation mechanisms and allosteric properties of metabotropic glutamate receptors
Doumazane, Etienne, Scholler, Pauline, Fabre, Ludovic, Zwier, Jurriaan M., Trinquet, Eric, Pin, Jean-Philippe, Rondard, Philippe
Published in Proceedings of the National Academy of Sciences - PNAS (09.04.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (09.04.2013)
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The chemokine CXC4 and CC2 receptors form homo- and heterooligomers that can engage their signaling G-protein effectors and βarrestin
Armando, Sylvain, Quoyer, Julie, Lukashova, Viktorya, Maiga, Arhamatoulaye, Percherancier, Yann, Heveker, Nikolaus, Pin, Jean-Philippe, Prézeau, Laurent, Bouvier, Michel
Published in The FASEB journal (01.10.2014)
Published in The FASEB journal (01.10.2014)
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