Search Results - "PIERARD Francoise" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

The discovery of the potent aurora inhibitor MK-0457 (VX-680)

The discovery of the potent aurora inhibitor MK-0457 (VX-680)

by Bebbington, David, Binch, Hayley, Charrier, Jean-Damien, Everitt, Simon, Fraysse, Damien, Golec, Julian, Kay, David, Knegtel, Ronald, Mak, Chau, Mazzei, Francesca, Miller, Andrew, Mortimore, Michael, O’Donnell, Michael, Patel, Sanjay, Pierard, Francoise, Pinder, Joanne, Pollard, John, Ramaya, Sharn, Robinson, Daniel, Rutherford, Alistair, Studley, John, Westcott, James
Published in Bioorganic & medicinal chemistry letters (01.07.2009)

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Journal Article

Discovery of Selective, Orally Bioavailable Pyrazolopyridine Inhibitors of Protein Kinase Cθ (PKCθ) That Ameliorate Symptoms of Experimental Autoimmune Encephalomyelitis

Discovery of Selective, Orally Bioavailable Pyrazolopyridine Inhibitors of Protein Kinase Cθ (PKCθ) That Ameliorate Symptoms of Experimental Autoimmune Encephalomyelitis

by Collier, Philip N, Twin, Heather C, Knegtel, Ronald M. A, Boyall, Dean, Brenchley, Guy, Davis, Christopher J, Keily, Shazia, Mak, Chau, Miller, Andrew, Pierard, Françoise, Settimo, Luca, Bolton, Clare M, Chiu, Peter, Curnock, Adam, Doyle, Elisabeth, Tanner, Adam J, Jimenez, Juan-Miguel
Published in ACS medicinal chemistry letters (08.08.2019)

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The Scope of Catalytic Enantioselective Tandem Carbonyl Ylide Formation−Intramolecular [3 + 2] Cycloadditions

The Scope of Catalytic Enantioselective Tandem Carbonyl Ylide Formation−Intramolecular [3 + 2] Cycloadditions

by Hodgson, David M, Labande, Agnès H, Pierard, Françoise Y. T. M, Expósito Castro, María Á
Published in Journal of organic chemistry (08.08.2003)

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Catalytic enantioselective rearrangements and cycloadditions involving ylides from diazo compounds

Catalytic enantioselective rearrangements and cycloadditions involving ylides from diazo compounds

by Hodgson, David M., Pierard, Françoise Y. T. M., Stupple, Paul A.
Published in Chemical Society reviews (2001)

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Synthesis of a stable pyridyl boronate and its reaction with aryl and heteroaryl halides

Synthesis of a stable pyridyl boronate and its reaction with aryl and heteroaryl halides

by Durrant, Steven J., Pinder, Joanne L., Charrier, Jean-Damien, Jimenez, Juan-Miguel, Brenchley, Guy, Collier, Philip N., Kay, David, Miller, Andrew, Pierard, Francoise, Ramaya, Sharn, Sadiq, Shazia, Twin, Heather C.
Published in Heterocycles (31.12.2006)

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Development of Dirhodium(II)-Catalyzed Generation and Enantioselective 1,3-Dipolar Cycloaddition of Carbonyl Ylides

Development of Dirhodium(II)-Catalyzed Generation and Enantioselective 1,3-Dipolar Cycloaddition of Carbonyl Ylides

by Hodgson, David M., Stupple, Paul A., Pierard, Françoise Y. T. M., Labande, Agnès H., Johnstone, Craig
Published in Chemistry : a European journal (15.10.2001)

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Journal Article

Design and Optimization of Selective Protein Kinase C θ (PKCθ) Inhibitors for the Treatment of Autoimmune Diseases

Design and Optimization of Selective Protein Kinase C θ (PKCθ) Inhibitors for the Treatment of Autoimmune Diseases

by Jimenez, Juan-Miguel, Boyall, Dean, Brenchley, Guy, Collier, Philip N, Davis, Christopher J, Fraysse, Damien, Keily, Shazia B, Henderson, Jaclyn, Miller, Andrew, Pierard, Francoise, Settimo, Luca, Twin, Heather C, Bolton, Claire M, Curnock, Adam P, Chiu, Peter, Tanner, Adam J, Young, Stephen
Published in Journal of medicinal chemistry (14.03.2013)

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Journal Article

Strategies for the modulation of phase II metabolism in a series of PKC epsilon inhibitors

Strategies for the modulation of phase II metabolism in a series of PKC epsilon inhibitors

by Clemens, Jeremy J., Coon, Timothy, Busch, Brett B., Asgian, Juliana L., Hudson, Sarah, Termin, Andreas, Flores, Tina B., Tran, Dao, Chiang, Peggy, Sperry, Sam, Gross, Ray, Abt, Jeffrey, Heim, Roger, Lechner, Sandra, Twin, Heather, Studley, John, Brenchley, Guy, Collier, Philip N., Pierard, Francoise, Miller, Andrew, Mak, Chau, Dvornikovs, Vadims, Jimenez, Juan-Miguel, Stamos, Dean
Published in Bioorganic & medicinal chemistry letters (01.08.2014)

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Journal Article

PROCESSES FOR MAKING COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

PROCESSES FOR MAKING COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

by LITTLER BENJAMIN JOSEPH, PIERARD FRANCOISE YVONNE THEODORA MARIE, ANGELL PAUL, CHARRIER JEAN DAMIEN, STUDLEY JOHN, SHI YI, DURRANT STEVEN JOHN, HUGHES ROBERT MICHAEL, SIESEL DAVID ANDREW, URBINA ARMANDO
Year of Publication 26.08.2019

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Patent

ATR 2--6--N-[5---3-]-[15-A]-3- RADIOLABELLED DERIVATIVES OF A 2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]- PYRAZOLO[15-A]PYRIMIDIN-3-CARBOXAMIDE COMPOUND USEFUL AS ATR KINASE INHIBITOR THE PREPARATION OF SAID COMPOUND AND DIFFERENT SOLID FORMS THEREOF

ATR 2--6--N-[5---3-]-[15-A]-3- RADIOLABELLED DERIVATIVES OF A 2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]- PYRAZOLO[15-A]PYRIMIDIN-3-CARBOXAMIDE COMPOUND USEFUL AS ATR KINASE INHIBITOR THE PREPARATION OF SAID COMPOUND AND DIFFERENT SOLID FORMS THEREOF

by PIERARD FRANCOISE, DAVIS CHRIS, CHARRIER JEAN DAMIEN, STUDLEY JOHN, ETXEBARRIA I JARDI GORKA, PINDER JOANNE, STORCK PIERRE HENRI, KNEGTEL RONALD, FRAYSSE DAMIEN, PANESAR MANINDER, AHMAD NADIA
Year of Publication 20.01.2017

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Patent

2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]PYRAZOLO[1,5-A]PYRIMIDIN-3-CARBOXAMIDE COMPOUND USEFUL AS ATR KINASE INHIBITOR, ITS PREPARATION, DIFFERENT SOLID FORMS AND RADIOLABELLED DERIVATIVES THEREOF

2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]PYRAZOLO[1,5-A]PYRIMIDIN-3-CARBOXAMIDE COMPOUND USEFUL AS ATR KINASE INHIBITOR, ITS PREPARATION, DIFFERENT SOLID FORMS AND RADIOLABELLED DERIVATIVES THEREOF

by SANGHVI TAPAN, DAVIS CHRISTOPHER JOHN, ETXEBARRIA I JARDI GORKA, MEDEK ALES, PANESAR MANINDER, SHAW DAVID MATTHEW, ZWICKER CARL, PIERARD FRANCOISE, CHARRIER JEAN DAMIEN, ZHANG YUEGANG, PEGG SIMON, STUDLEY JOHN, PINDER JOANNE, FRAYSSE DAMIEN, WALDO MICHAEL, ALEM NAZIHA
Year of Publication 08.08.2016

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Patent

PROCESSES FOR MAKING COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

PROCESSES FOR MAKING COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

by LITTLER BENJAMIN JOSEPH, PIERARD FRANCOISE YVONNE THEODORA MARIE, ANGELL PAUL, CHARRIER JEAN DAMIEN, STUDLEY JOHN, SHI YI, DURRANT STEVEN JOHN, HUGHES ROBERT MICHAEL, SIESEL DAVID ANDREW, URBINA ARMANDO
Year of Publication 16.07.2014

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Patent

COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

by STORCK PIERRE HENRI, DURRANT STEVEN JOHN, ZWICKER CARL, LITTLER BENJAMIN JOSEPH, PIERARD FRANCOISE YVONNE THEODORA MARIE, ANGELL PAUL, LOCONTE NICHOLAS, CHARRIER JEAN DAMIEN, STUDLEY JOHN, BARDER TIMOTHY, HUGHES ROBERT MICHAEL, SIESEL DAVID ANDREW, URBINA ARMANDO
Year of Publication 04.07.2014

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Patent

COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

by SHAW DAVID, BOYALL DEAN, ETXEBARRIA I JARDI GORKA, MIDDLETON DONALD, STORCK PIERRE HENRI, TWIN HEATHER, PANESAR MANINDER, DURRANT STEVEN, ODONNELL MICHAEL, PIERARD FRANCOISE, KAY DAVID, DAVIS CHRIS, CHARRIER JEAN DAMIEN, JIMENEZ JUAN MIGUEL, STUDLEY JOHN, PINDER JOANNE, KNEGTEL RONALD, DAVIS REBECCA, FRAYSSE DAMIEN, AHMAD NADIA
Year of Publication 07.08.2015

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Patent

AZAINDOLE USEFUL AS JAK AND OTHER PROTEIN KINASE INHIBITOR

AZAINDOLE USEFUL AS JAK AND OTHER PROTEIN KINASE INHIBITOR

by EVERITT SIMON, BOYALL DEAN, BETHIEL RANDY, COME JON, LAUFFER DAVID, SALITURO FRANCESCO, ROBINSON DANIEL, HARRINGTON EDMUND, BINCH HAYLEY, FARMER LUC, MORTIMORE MICHAEL, WANG JIAN, ARONOV ALEX, PIERARD FRANCOISE, PIERCE ALBERT, GREEN JEREMY, CHARRIER JEAN-DAMIEN, COURT JOHN, PINDER JOANNE, WANG TIANSHENG, FRAYSSE DAMIEN
Year of Publication 22.06.2015

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Patent

Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof

Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof

by Panesar, Maninder, Davis, Chris, Studley, John, Charrier, Jean-Damien, Storck, Pierre-Henri, Etxebarria I Jardi, Gorka, Knegtel, Ronald, Fraysse, Damien, Pierard, Francoise, Ahmad, Nadia, Pinder, Joanne
Year of Publication 22.12.2023

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Patent

Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof

Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof

by Panesar, Maninder, Davis, Chris, Studley, John, Charrier, Jean-Damien, Storck, Pierre-Henri, Etxebarria I Jardi, Gorka, Knegtel, Ronald, Fraysse, Damien, Pierard, Francoise, Ahmad, Nadia, Pinder, Joanne
Year of Publication 22.12.2023

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Patent

2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]PYRAZOLO[1,5-A]PYRIMIDIN-3-CARBOXAMIDE COMPOUND USEFUL AS ATR KINASE INHIBITOR, ITS PREPARATION, DIFFERENT SOLID FORMS AND RADIOLABELLED DERIVATIVES THEREOF

2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]PYRAZOLO[1,5-A]PYRIMIDIN-3-CARBOXAMIDE COMPOUND USEFUL AS ATR KINASE INHIBITOR, ITS PREPARATION, DIFFERENT SOLID FORMS AND RADIOLABELLED DERIVATIVES THEREOF

by SHAW, DAVID MATTHEW, STUDLEY, JOHN, CHARRIER, JEAN-DAMIEN, ETXEBARRIA I JARDI, GORKA, PINDER, JOANNE, PANESAR, MANINDER, ALEM, NAZIHA, PIERARD, FRANCOISE, SANGHVI, TAPAN, PEGG, SIMON, FRAYSSE, DAMIEN, WALDO, MICHAEL, MEDEK, ALES, ZHANG, YUEGANG, DAVIS, CHRISTOPHER JOHN, ZWICKER, CARL
Year of Publication 31.10.2023

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Patent

HYDROXY AND (HALO)ALKOXY SUBSTITUTED TETRAHYDROFURANS AS MODULATORS OF SODIUM CHANNELS

HYDROXY AND (HALO)ALKOXY SUBSTITUTED TETRAHYDROFURANS AS MODULATORS OF SODIUM CHANNELS

by SKERRATT, Sarah, CARVALHO MEIRELES, Lidio Marx, PIERARD, Francoise, SHAW, David Matthew, PONTILLO, Joseph, NORTH, Kiri, ETXEBARRIA JARDI, Gorka, HURLEY, Dennis James, HADIDA RUAH, Sara S, NEUBERT, Timothy Donald, GALAN, Bhairavi, BECK, Elizabeth Mary, STAMOS, Dean, THOMSON, Stephen Andrew, VIRANI, Anisa Nizarali, AHMAD, Nadia M, CHUDYK, Ewa Iwona, PULLIN, Robert, DURRANT, Steven John, KNEGTEL, Ronald Marcellus, SCHMIDT, Yvonne, PINDER, Joanne Louise, WRAY, Christopher, SOUSA, Bruno Artur
Year of Publication 05.09.2024

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Patent

AZAINDOLES USEFUL AS INHIBITORS OF JAK AND OTHER PROTEIN KINASES

AZAINDOLES USEFUL AS INHIBITORS OF JAK AND OTHER PROTEIN KINASES

by EVERITT SIMON, BOYALL DEAN, BETHIEL RANDY, COME JON, LAUFFER DAVID, SALITURO FRANCESCO, ROBINSON DANIEL, HARRINGTON EDMUND, BINCH HAYLEY, FARMER LUC, MORTIMORE MICHAEL, WANG JIAN, ARONOV ALEX, PIERARD FRANCOISE, PIERCE ALBERT, GREEN JEREMY, CHARRIER JEAN DAMIEN, COURT JOHN, PINDER JOANNE, WANG TIANSHENG, FRAYSSE DAMIEN
Year of Publication 16.04.2010

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Patent

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