Search Results - "PIEPOLI, Tiziana" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Pharmacological characterisation of CR6086, a potent prostaglandin E2 receptor 4 antagonist, as a new potential disease-modifying anti-rheumatic drug

Pharmacological characterisation of CR6086, a potent prostaglandin E2 receptor 4 antagonist, as a new potential disease-modifying anti-rheumatic drug

by Caselli, Gianfranco, Bonazzi, Albino, Lanza, Marco, Ferrari, Flora, Maggioni, Daniele, Ferioli, Cristian, Giambelli, Roberto, Comi, Eleonora, Zerbi, Silvia, Perrella, Marco, Letari, Ornella, Di Luccio, Elena, Colovic, Milena, Persiani, Stefano, Zanelli, Tiziano, Mennuni, Laura, Piepoli, Tiziana, Rovati, Lucio Claudio
Published in Arthritis research & therapy (01.03.2018)

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Journal Article

The neural progenitor-restricted isoform of the MARK4 gene in 19q13.2 is upregulated in human gliomas and overexpressed in a subset of glioblastoma cell lines

The neural progenitor-restricted isoform of the MARK4 gene in 19q13.2 is upregulated in human gliomas and overexpressed in a subset of glioblastoma cell lines

by BEGHINI, Alessandro, MAGNANI, Ivana, LARIZZA, Lidia, ROVERSI, Gaia, PIEPOLI, Tiziana, DI TERLIZZI, Simona, MORONI, Ramona F, POLLO, Bianca, FUHRMAN CONTI, Anna M, COWELL, John K, FINOCCHIARO, Gaetano
Published in Oncogene (01.05.2003)

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Journal Article

Experimental Pharmacology of Glucosamine Sulfate

Experimental Pharmacology of Glucosamine Sulfate

by Piepoli, Tiziana, Chiusaroli, Riccardo, Zanelli, Tiziano, Ballanti, Paola, Lanza, Marco, Rovati, Lucio C., Caselli, Gianfranco
Published in International Journal of Rheumatology (01.01.2011)

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Journal Article

CR10049, THE FIRST OA-TARGETED KINASE INHIBITOR, IMPROVES PAIN BEHAVIOUR, RESOLVES INFLAMMATION AND PRESERVES JOINT STRUCTURE IN SMALL AND LARGE ANIMAL MODELS

CR10049, THE FIRST OA-TARGETED KINASE INHIBITOR, IMPROVES PAIN BEHAVIOUR, RESOLVES INFLAMMATION AND PRESERVES JOINT STRUCTURE IN SMALL AND LARGE ANIMAL MODELS

by Piepoli, Tiziana, Giancotti, Luigino A., Artusi, Roberto, Ghirri, Matteo, Visintin, Michela, Caselli, Gianfranco, Rovati, Lucio
Published in Osteoarthritis and cartilage (01.06.2024)

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Journal Article

LB-005 - CR10049, THE FIRST OA-TARGETED KINASE INHIBITOR, IMPROVES PAIN BEHAVIOUR, RESOLVES INFLAMMATION AND PRESERVES JOINT STRUCTURE IN SMALL AND LARGE ANIMAL MODELS

LB-005 - CR10049, THE FIRST OA-TARGETED KINASE INHIBITOR, IMPROVES PAIN BEHAVIOUR, RESOLVES INFLAMMATION AND PRESERVES JOINT STRUCTURE IN SMALL AND LARGE ANIMAL MODELS

by Piepoli, Tiziana, Giancotti, Luigino A., Artusi, Roberto, Ghirri, Matteo, Visintin, Michela, Caselli, Gianfranco, Rovati, Lucio
Published in Osteoarthritis and cartilage (01.06.2024)

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Journal Article

Abstract 2208: Combination of the EP4 antagonist CR6086 and anti-PD-1 monoclonal antibody inhibits tumor growth in a microsatellite stable colorectal cancer in mice

Abstract 2208: Combination of the EP4 antagonist CR6086 and anti-PD-1 monoclonal antibody inhibits tumor growth in a microsatellite stable colorectal cancer in mice

by Caselli, Gianfranco, Ferrari, Flora, Piepoli, Tiziana, Grotti, Adriana, Cavagnoli, Rosanna, Montagna, Giuseppe M., Romanelli, Pierpaolo, Bonazzi, Albino, Lanza, Marco, Recordati, Camilla, Rovati, Lucio C.
Published in Cancer research (Chicago, Ill.) (15.08.2020)

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Journal Article

Abstract 4219: Efficacy of CR13626, a novel oral brain penetrant multi-kinase inhibitor, in a mouse model of glioblastoma

Abstract 4219: Efficacy of CR13626, a novel oral brain penetrant multi-kinase inhibitor, in a mouse model of glioblastoma

by Galimberti, Chiara, Piepoli, Tiziana, Montagna, Giuseppe M., Zerbi, Silvia, Letari, Ornella, Artusi, Roberto, Colovic, Milena, Persiani, Stefano, Caselli, Gianfranco, Rovati, Lucio C.
Published in Cancer research (Chicago, Ill.) (15.08.2020)

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Journal Article

Pharmacological characterisation of CR6086, a potent prostaglandin E 2 receptor 4 antagonist, as a new potential disease-modifying anti-rheumatic drug

Pharmacological characterisation of CR6086, a potent prostaglandin E 2 receptor 4 antagonist, as a new potential disease-modifying anti-rheumatic drug

by Caselli, Gianfranco, Bonazzi, Albino, Lanza, Marco, Ferrari, Flora, Maggioni, Daniele, Ferioli, Cristian, Giambelli, Roberto, Comi, Eleonora, Zerbi, Silvia, Perrella, Marco, Letari, Ornella, Di Luccio, Elena, Colovic, Milena, Persiani, Stefano, Zanelli, Tiziano, Mennuni, Laura, Piepoli, Tiziana, Rovati, Lucio Claudio
Published in Arthritis research & therapy (01.03.2018)

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Journal Article

CR13626: a novel oral brain penetrant tyrosine kinase inhibitor that reduces tumor growth and prolongs survival in a mouse model of glioblastoma

CR13626: a novel oral brain penetrant tyrosine kinase inhibitor that reduces tumor growth and prolongs survival in a mouse model of glioblastoma

by Galimberti, Chiara, Piepoli, Tiziana, Letari, Ornella, Artusi, Roberto, Persiani, Stefano, Caselli, Gianfranco, Rovati, Lucio C
Published in American journal of cancer research (01.01.2021)

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Journal Article

단백질 키나제 억제제로서의 벤조- 및 피리도-피라졸

단백질 키나제 억제제로서의 벤조- 및 피리도-피라졸

by ARTUSI ROBERTO, MANDELLI STEFANO, ROVATI LUCIO CLAUDIO, PIEPOLI TIZIANA, BOVINO CLARA, COLACE FABRIZIO, BUZZI BENEDETTA
Year of Publication 07.01.2022

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Patent

종양 치료를 위한 EP4 길항제 및 면역 체크포인트 억제제의 약제학적 조합물

종양 치료를 위한 EP4 길항제 및 면역 체크포인트 억제제의 약제학적 조합물

by BONAZZI ALBINO, CASELLI GIANFRANCO, MAGGIONI DANIELE, GIORDANI ANTONIO, ROVATI LUCIO CLAUDIO, MAGARACI FILIPPO, PIEPOLI TIZIANA
Year of Publication 13.12.2021

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Patent

Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[b,f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP₄ receptor

Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[b,f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP₄ receptor

by Stasi, Luigi Piero, Bhimani, Kanji, Borriello, Manuela, Canciani, Luca, Caselli, Gianfranco, Colace, Fabrizio, Ferioli, Cristian, Kaswala, Mehul, Mennuni, Laura, Piepoli, Tiziana, Pucci, Sabrina, Salvi, Matteo, Shirsath, Vikas, Zanelli, Tiziano, Zerbi, Silvia
Published in Bioorganic & medicinal chemistry letters (01.11.2011)

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Journal Article

Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[b,f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP sub(4 receptor)

Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[b,f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP sub(4 receptor)

by Stasi, Luigi Piero, Bhimani, Kanji, Borriello, Manuela, Canciani, Luca, Caselli, Gianfranco, Colace, Fabrizio, Ferioli, Cristian, Kaswala, Mehul, Mennuni, Laura, Piepoli, Tiziana, Pucci, Sabrina, Salvi, Matteo, Shirsath, Vikas, Zanelli, Tiziano, Zerbi, Silvia
Published in Bioorganic & medicinal chemistry letters (01.11.2011)

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Journal Article

CCK1 Receptor and CCK Gene Polymorphisms in Constipation-Predominant Irritable Bowel Syndrome

CCK1 Receptor and CCK Gene Polymorphisms in Constipation-Predominant Irritable Bowel Syndrome

by Jobbagy-Ovari, Gabriella, Piepoli, Tiziana, Foldes, Anna, Beglinger, Christoph, Whorwell, Peter J, Thompson, David G, Dzieniszewski, Jan, Rovati, Lucio C, D'Amato, Massimo, Varga, Gabor
Published in Gastroenterology (New York, N.Y. 1943) (2011)

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Journal Article

Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[ b, f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP 4 receptor

Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[ b, f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP 4 receptor

by Stasi, Luigi Piero, Bhimani, Kanji, Borriello, Manuela, Canciani, Luca, Caselli, Gianfranco, Colace, Fabrizio, Ferioli, Cristian, Kaswala, Mehul, Mennuni, Laura, Piepoli, Tiziana, Pucci, Sabrina, Salvi, Matteo, Shirsath, Vikas, Zanelli, Tiziano, Zerbi, Silvia
Published in Bioorganic & medicinal chemistry letters (2011)

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Journal Article

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

by ROVATI, Lucio Claudio, PIEPOLI, Tiziana, CASELLI, Gianfranco
Year of Publication 10.01.2024

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Patent

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5] OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5] OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

by ROVATI, Lucio Claudio, PIEPOLI, Tiziana, CASELLI, Gianfranco
Year of Publication 26.01.2023

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Patent

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

by ROVATI, Lucio Claudio, PIEPOLI, Tiziana, CASELLI, Gianfranco
Year of Publication 05.10.2022

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Patent

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

by ROVATI, Lucio Claudio, PIEPOLI, Tiziana, CASELLI, Gianfranco
Year of Publication 03.06.2021

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Patent

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

(R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR ITS SALT ALSO IN POLYMORPHIC FORM A FOR USE IN THE PREVENTION OF HETEROTOPIC OSSIFICATION

by ROVATI, Lucio Claudio, PIEPOLI, Tiziana, CASELLI, Gianfranco
Year of Publication 02.06.2021

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Patent