Discovery of Potent, Orally Bioavailable, Small-Molecule Inhibitors of WNT Signaling from a Cell-Based Pathway Screen
Mallinger, Aurélie, Crumpler, Simon, Pichowicz, Mark, Waalboer, Dennis, Stubbs, Mark, Adeniji-Popoola, Olajumoke, Wood, Bozena, Smith, Elizabeth, Thai, Ching, Henley, Alan T, Georgi, Katrin, Court, William, Hobbs, Steve, Box, Gary, Ortiz-Ruiz, Maria-Jesus, Valenti, Melanie, De Haven Brandon, Alexis, TePoele, Robert, Leuthner, Birgitta, Workman, Paul, Aherne, Wynne, Poeschke, Oliver, Dale, Trevor, Wienke, Dirk, Esdar, Christina, Rohdich, Felix, Raynaud, Florence, Clarke, Paul A, Eccles, Suzanne A, Stieber, Frank, Schiemann, Kai, Blagg, Julian
Published in Journal of medicinal chemistry (26.02.2015)
Published in Journal of medicinal chemistry (26.02.2015)
Get full text
Journal Article
Thiyl Radicals in Organic Synthesis
Dénès, Fabrice, Pichowicz, Mark, Povie, Guillaume, Renaud, Philippe
Published in Chemical reviews (12.03.2014)
Published in Chemical reviews (12.03.2014)
Get full text
Journal Article
Structural and mechanistic analysis of ATPase inhibitors targeting mycobacterial DNA gyrase
Henderson, Sara R, Stevenson, Clare E M, Malone, Brandon, Zholnerovych, Yelyzaveta, Mitchenall, Lesley A, Pichowicz, Mark, McGarry, David H, Cooper, Ian R, Charrier, Cedric, Salisbury, Anne-Marie, Lawson, David M, Maxwell, Anthony
Published in Journal of antimicrobial chemotherapy (01.10.2020)
Published in Journal of antimicrobial chemotherapy (01.10.2020)
Get full text
Journal Article
Novel Bacterial Topoisomerase Inhibitors with Potent Broad-Spectrum Activity against Drug-Resistant Bacteria
Charrier, Cédric, Salisbury, Anne-Marie, Savage, Victoria J, Duffy, Thomas, Moyo, Emmanuel, Chaffer-Malam, Nathan, Ooi, Nicola, Newman, Rebecca, Cheung, Jonathan, Metzger, Richard, McGarry, David, Pichowicz, Mark, Sigerson, Ralph, Cooper, Ian R, Nelson, Gary, Butler, Hayley S, Craighead, Mark, Ratcliffe, Andrew J, Best, Stuart A, Stokes, Neil R
Published in Antimicrobial agents and chemotherapy (01.05.2017)
Published in Antimicrobial agents and chemotherapy (01.05.2017)
Get full text
Journal Article
Design, synthesis and antibacterial properties of pyrimido[4,5-b]indol-8-amine inhibitors of DNA gyrase
McGarry, David H., Cooper, Ian R., Walker, Rolf, Warrilow, Catherine E., Pichowicz, Mark, Ratcliffe, Andrew J., Salisbury, Anne-Marie, Savage, Victoria J., Moyo, Emmanuel, Maclean, John, Smith, Andrew, Charrier, Cédric, Stokes, Neil R., Lindsay, David M., Kerr, William J.
Published in Bioorganic & medicinal chemistry letters (15.09.2018)
Published in Bioorganic & medicinal chemistry letters (15.09.2018)
Get full text
Journal Article
Microwave-assisted synthesis of 4-amino-3,5-dihalopyridines
Pichowicz, Mark, Crumpler, Simon, McDonald, Edward, Blagg, Julian
Published in Tetrahedron (27.03.2010)
Published in Tetrahedron (27.03.2010)
Get full text
Journal Article
Discovery and structure–activity relationships of a novel isothiazolone class of bacterial type II topoisomerase inhibitors
Cooper, Ian R., McCarroll, Andrew J., McGarry, David, Kirkham, James, Pichowicz, Mark, Walker, Rolf, Warrilow, Catherine, Salisbury, Anne-Marie, Savage, Victoria J., Moyo, Emmanuel, Forward, Henry, Cheung, Jonathan, Metzger, Richard, Gault, Zoe, Nelson, Gary, Hughes, Diarmaid, Cao, Sha, Maclean, John, Charrier, Cédric, Craighead, Mark, Best, Stuart, Stokes, Neil R., Ratcliffe, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.09.2016)
Published in Bioorganic & medicinal chemistry letters (01.09.2016)
Get full text
Journal Article
효소 저해제
BIRCH LOUISE MICHELLE, CHILDS MITCHELL LEWIS, HODGSON SIMON TEANBY, GREVES WILLIAM JACK, OBARA ALICJA STELA, PITTAWAY RACHAEL, EVANS DAVID MICHAEL, WRIGGLESWORTH JOSEPH WILLIAM, CLARK DAVID EDWARD, EDWARDS HANNAH JOY, MAZZACANI ALESSANDRO, DAVIE REBECCA LOUISE, PICHOWICZ MARK, YANG XUEZHENG, ROOKER DAVID PHILIP, ROE MICHAEL BRYAN, NORTH CARL LESLIE, THROUP ADAM ERIC, STOCKS MICHAEL JOHN, SMITH ALUN JOHN
Year of Publication 04.09.2023
Get full text
Year of Publication 04.09.2023
Patent
Synthesis towards complex bridged alkaloids derived from diketopiperazines: a cationic cascade approach to stephacidins, paraherquamides and related systems
Pichowicz, Mark, Simpkins, Nigel S., Blake, Alexander J., Wilson, Claire
Published in Tetrahedron letters (20.11.2006)
Published in Tetrahedron letters (20.11.2006)
Get full text
Journal Article
MODULATORS OF G PROTEIN-COUPLED RECEPTOR 88
Pichowicz, Mark, Quibell, Martin, Murray, Fraser, Schulz-Utermoehl, Tim
Year of Publication 25.04.2024
Get full text
Year of Publication 25.04.2024
Patent
MODULATORS OF G PROTEIN-COUPLED RECEPTOR 88
PICHOWICZ, Mark, MURRAY, Fraser, SCHULZ-UTERMOEHL, Tim, QUIBELL, Martin
Year of Publication 25.10.2023
Get full text
Year of Publication 25.10.2023
Patent
MODULATORS OF G PROTEIN-COUPLED RECEPTOR 88
PICHOWICZ, Mark, MURRAY, Fraser, SCHULZ-UTERMOEHL, Tim, QUIBELL, Martin
Year of Publication 23.06.2022
Get full text
Year of Publication 23.06.2022
Patent
ENZYME INHIBITORS
NORTH, Carl Leslie, HODGSON, Simon Teanby, ROOKER, David Philip, BIRCH, Louise Michelle, PITTAWAY, Rachael, OBARA, Alicja Stela, ROE, Michael Bryan, EDWARDS, Hannah Joy, YANG, Xuezheng, PICHOWICZ, Mark, SMITH, Alun John, CHILDS, Mitchell Lewis, GREVES, William Jack, CLARK, David Edward, WRIGGLESWORTH, Joseph William, STOCKS, Michael John, THROUP, Adam Eric, EVANS, David Michael, MAZZACANI, Alessandro, DAVIE, Rebecca Louise
Year of Publication 02.05.2024
Get full text
Year of Publication 02.05.2024
Patent
ENZYME INHIBITORS
NORTH, Carl Leslie, HODGSON, Simon Teanby, ROOKER, David Philip, BIRCH, Louise Michelle, PITTAWAY, Rachael, OBARA, Alicja Stela, ROE, Michael Bryan, EDWARDS, Hannah Joy, YANG, Xuezheng, PICHOWICZ, Mark, SMITH, Alun John, CHILDS, Mitchell Lewis, GREVES, William Jack, CLARK, David Edward, WRIGGLESWORTH, Joseph William, STOCKS, Michael John, THROUP, Adam Eric, EVANS, David Michael, MAZZACANI, Alessandro, DAVIE, Rebecca Louise
Year of Publication 22.02.2024
Get full text
Year of Publication 22.02.2024
Patent
ChemInform Abstract: Thiyl Radicals in Organic Synthesis
Denes, Fabrice, Pichowicz, Mark, Povie, Guillaume, Renaud, Philippe
Published in ChemInform (06.05.2014)
Published in ChemInform (06.05.2014)
Get full text
Journal Article