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CoMFA, Synthesis, and Pharmacological Evaluation of ( E )-3-(2-Carboxy-2-arylvinyl)-4,6-dichloro-1 H -indole-2-carboxylic Acids: 3-[2-(3-Aminophenyl)-2-carboxyvinyl]-4,6-dichloro-1 H -indole-2-carboxylic Acid, a Potent Selective Glycine-Site NMDA Receptor Antagonist
Baron, Bruce M., Cregge, Robert J., Farr, Robert A., Friedrich, Dirk, Gross, Raymond S., Harrison, Boyd L., Janowick, David A., Matthews, Donald, McCloskey, Timothy C., Meikrantz, Scott, Nyce, Philip L., Vaz, Roy, Metz, William A.
Published in Journal of medicinal chemistry (01.02.2005)
Published in Journal of medicinal chemistry (01.02.2005)
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Journal Article
CoMFA, synthesis, and pharmacological evaluation of (E)-3-(2-carboxy-2-arylvinyl)-4,6-dichloro-1H-indole-2-carboxylic acids: 3-[2-(3-Aminophenyl)-2-carboxyvinyl]-4,6-dichloro-1H-indole-2-carboxylic acid, a potent selective glycine-site NMDA receptor antagonis
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Published in Journal of medicinal chemistry (2005)
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Published in Journal of medicinal chemistry (2005)
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3-(2-Carboxyindol-3-yl)propionic acid-based antagonists of the N-methyl-D-aspartic acid receptor associated glycine binding site
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