A Novel Allosteric Activator of Free Fatty Acid 2 Receptor Displays Unique Gi-functional Bias
Bolognini, Daniele, Moss, Catherine E., Nilsson, Karolina, Petersson, Annika U., Donnelly, Iona, Sergeev, Eugenia, König, Gabriele M., Kostenis, Evi, Kurowska-Stolarska, Mariola, Miller, Ashley, Dekker, Niek, Tobin, Andrew B., Milligan, Graeme
Published in The Journal of biological chemistry (02.09.2016)
Published in The Journal of biological chemistry (02.09.2016)
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GPR103 Antagonists Demonstrating Anorexigenic Activity in Vivo: Design and Development of Pyrrolo[2,3‑c]pyridines That Mimic the C‑Terminal Arg-Phe Motif of QRFP26
Georgsson, Jennie, Bergström, Fredrik, Nordqvist, Anneli, Watson, Martin J, Blundell, Charles D, Johansson, Magnus J, Petersson, Annika U, Yuan, Zhong-Qing, Zhou, Yiqun, Kristensson, Lisbeth, Kakol-Palm, Dorota, Tyrchan, Christian, Wellner, Eric, Bauer, Udo, Brodin, Peter, Svensson Henriksson, Anette
Published in Journal of medicinal chemistry (24.07.2014)
Published in Journal of medicinal chemistry (24.07.2014)
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Identification and design of a novel series of MGAT2 inhibitors
Barlind, Jonas G., Buckett, Linda K., Crosby, Sharon G., Davidsson, Öjvind, Emtenäs, Hans, Ertan, Anne, Jurva, Ulrik, Lemurell, Malin, Gutierrez, Pablo Morentin, Nilsson, Karolina, O’Mahony, Gavin, Petersson, Annika U., Redzic, Alma, Wågberg, Fredrik, Yuan, Zhong-Qing
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
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Design and Optimization of Pyrazinecarboxamide-Based Inhibitors of Diacylglycerol Acyltransferase 1 (DGAT1) Leading to a Clinical Candidate Dimethylpyrazinecarboxamide Phenylcyclohexylacetic Acid (AZD7687)
Barlind, Jonas G., Bauer, Udo A., Birch, Alan M., Birtles, Susan, Buckett, Linda K., Butlin, Roger J., Davies, Robert D. M., Eriksson, Jan W., Hammond, Clare D., Hovland, Ragnar, Johannesson, Petra, Johansson, Magnus J., Kemmitt, Paul D., Lindmark, Bo T., Morentin Gutierrez, Pablo, Noeske, Tobias A., Nordin, Andreas, O’Donnell, Charles J., Petersson, Annika U., Redzic, Alma, Turnbull, Andrew V., Vinblad, Johanna
Published in Journal of medicinal chemistry (13.12.2012)
Published in Journal of medicinal chemistry (13.12.2012)
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Correction to GPR103 Antagonists Demonstrating Anorexigenic Activity in Vivo: Design and Development of Pyrrolo[2,3‑c]pyridines That Mimic the C‑Terminal Arg-Phe Motif of QRFP26
Georgsson, Jennie, Bergström, Fredrik, Nordqvist, Anneli, Watson, Martin J, Blundell, Charles D, Johansson, Magnus J, Petersson, Annika U, Yuan, Zhong-Qing, Zhou, Yiqun, Kristensson, Lisbeth, Kakol-Palm, Dorota, Tyrchan, Christian, Wellner, Eric, Bauer, Udo, Brodin, Peter, Svensson Henriksson, Anette
Published in Journal of medicinal chemistry (14.05.2015)
Published in Journal of medicinal chemistry (14.05.2015)
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A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y12 receptor
BACH, Peter, BOSTROM, Jonas, BRICKMANN, Kay, VAN GIEZEN, J. J. J, HOVLAND, Ragnar, PETERSSON, Annika U, RAY, Asim, ZETTERBERG, Fredrik
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y sub(12 receptor)
Bach, Peter, Bostroem, Jonas, Brickmann, Kay, Van Giezen, JJJ, Hovland, Ragnar, Petersson, Annika U, Ray, Asim, Zetterberg, Fredrik
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Journal Article
A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y 12 receptor
Bach, Peter, Boström, Jonas, Brickmann, Kay, van Giezen, J.J.J., Hovland, Ragnar, Petersson, Annika U., Ray, Asim, Zetterberg, Fredrik
Published in Bioorganic & medicinal chemistry letters (2011)
Published in Bioorganic & medicinal chemistry letters (2011)
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Compuestos derivados de 6-fenilpirazin-2-carboxamida y 6-fenilpirazin-2-carbotioamida, inhibidores de dgat-1; composicion farmaceutica; y su uso en el tratamiento de la diabetes mellitus y obesidad
JOHANNESSON PETRA, PETERSSON ANNIKA U, BAUER UDO ANDREAS, HANSSON JONAS GUNNAR, JOHANSSON JAN MAGNUS, NOESKE ALEXANDER TOBIAS
Year of Publication 27.11.2009
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Year of Publication 27.11.2009
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