PI3K inhibitors are finally coming of age
Vanhaesebroeck, Bart, Perry, Matthew W D, Brown, Jennifer R, André, Fabrice, Okkenhaug, Klaus
Published in Nature reviews. Drug discovery (01.10.2021)
Published in Nature reviews. Drug discovery (01.10.2021)
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Design, Synthesis, and Biological Evaluation of MEK PROTACs
Vollmer, Stefan, Cunoosamy, Danen, Lv, Huafei, Feng, Huanxi, Li, Xia, Nan, Ziyang, Yang, Wenzhen, Perry, Matthew W. D
Published in Journal of medicinal chemistry (09.01.2020)
Published in Journal of medicinal chemistry (09.01.2020)
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Author Correction: PI3K inhibitors are finally coming of age
Vanhaesebroeck, Bart, Perry, Matthew W D, Brown, Jennifer R, André, Fabrice, Okkenhaug, Klaus
Published in Nature reviews. Drug discovery (01.10.2021)
Published in Nature reviews. Drug discovery (01.10.2021)
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Impact of Stereospecific Intramolecular Hydrogen Bonding on Cell Permeability and Physicochemical Properties
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Published in Journal of medicinal chemistry (27.03.2014)
Published in Journal of medicinal chemistry (27.03.2014)
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Structural and conformational determinants of macrocycle cell permeability
Over, Björn, Matsson, Pär, Tyrchan, Christian, Artursson, Per, Doak, Bradley C, Foley, Michael A, Hilgendorf, Constanze, Johnston, Stephen E, Lee, 4th, Maurice D, Lewis, Richard J, McCarren, Patrick, Muncipinto, Giovanni, Norinder, Ulf, Perry, Matthew W D, Duvall, Jeremy R, Kihlberg, Jan
Published in Nature chemical biology (01.12.2016)
Published in Nature chemical biology (01.12.2016)
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Stabilization of protein-protein interactions in drug discovery
Andrei, Sebastian A., Sijbesma, Eline, Hann, Michael, Davis, Jeremy, O'Mahony, Gavin, Perry, Matthew W. D., Karawajczyk, Anna, Eickhoff, Jan, Brunsveld, Luc, Doveston, Richard G., Milroy, Lech-Gustav, Ottmann, Christian
Published in Expert opinion on drug discovery (02.09.2017)
Published in Expert opinion on drug discovery (02.09.2017)
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A class of highly selective inhibitors bind to an active state of PI3Kγ
Gangadhara, Gangadhara, Dahl, Göran, Bohnacker, Thomas, Rae, Rebecca, Gunnarsson, Jenny, Blaho, Stefan, Öster, Linda, Lindmark, Helena, Karabelas, Kostas, Pemberton, Nils, Tyrchan, Christian, Mogemark, Mickael, Wymann, Matthias P, Williams, Roger L, Perry, Matthew W D, Papavoine, Tineke, Petersen, Jens
Published in Nature chemical biology (01.04.2019)
Published in Nature chemical biology (01.04.2019)
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Scaffold-hopping with zwitterionic CCR3 antagonists: Identification and optimisation of a series with good potency and pharmacokinetics leading to the discovery of AZ12436092
Bahl, Ash, Barton, Patrick, Bowers, Keith, Caffrey, Moya V., Denton, Rebecca, Gilmour, Peter, Hawley, Shaun, Linannen, Tero, Luckhurst, Christopher A., Mochel, Tobias, Perry, Matthew W.D., Riley, Robert J., Roe, Emma, Springthorpe, Brian, Stein, Linda, Webborn, Peter
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
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Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3‑Kinase (PI3K)‑γ Inhibitors
Pemberton, Nils, Mogemark, Mickael, Arlbrandt, Susanne, Bold, Peter, Cox, Rhona J, Gardelli, Cristina, Holden, Neil S, Karabelas, Kostas, Karlsson, Johan, Lever, Sarah, Li, Xueshan, Lindmark, Helena, Norberg, Monica, Perry, Matthew W. D, Petersen, Jens, Rodrigo Blomqvist, Sandra, Thomas, Matthew, Tyrchan, Christian, Westin Eriksson, Annika, Zlatoidsky, Pavol, Öster, Linda
Published in Journal of medicinal chemistry (28.06.2018)
Published in Journal of medicinal chemistry (28.06.2018)
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Discovery of AZD8154, a Dual PI3Kγδ Inhibitor for the Treatment of Asthma
Perry, Matthew W. D, Björhall, Karin, Bold, Peter, Brűlls, Mikael, Börjesson, Ulf, Carlsson, Johan, Chang, Hui-Fang Amy, Chen, Yunhua, Eriksson, Anders, Fihn, Britt-Marie, Fransson, Rebecca, Fredlund, Linda, Ge, Hongbin, Huang, Haijuan, Karabelas, Kostas, Lamm Bergström, Eva, Lever, Sarah, Lindmark, Helena, Mogemark, Mickael, Nikitidis, Antonios, Palmgren, Anna-Pia, Pemberton, Nils, Petersen, Jens, Rodrigo Blomqvist, Mio, Smith, Reed W, Thomas, Matthew J, Ullah, Victoria, Tyrchan, Christian, Wennberg, Tiiu, Westin Eriksson, Annika, Yang, Wenzhen, Zhao, Shuchun, Öster, Linda
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
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Design and Synthesis of Soluble and Cell-Permeable PI3Kδ Inhibitors for Long-Acting Inhaled Administration
Perry, Matthew W. D, Björhall, Karin, Bonn, Britta, Carlsson, Johan, Chen, Yunhua, Eriksson, Anders, Fredlund, Linda, Hao, Hai’e, Holden, Neil S, Karabelas, Kostas, Lindmark, Helena, Liu, Feifei, Pemberton, Nils, Petersen, Jens, Rodrigo Blomqvist, Sandra, Smith, Reed W, Svensson, Tor, Terstiege, Ina, Tyrchan, Christian, Yang, Wenzhen, Zhao, Shuchun, Öster, Linda
Published in Journal of medicinal chemistry (22.06.2017)
Published in Journal of medicinal chemistry (22.06.2017)
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Identification of Phosphate-Containing Compounds as New Inhibitors of 14-3-3/c-Abl Protein–Protein Interaction
Iralde-Lorente, Leire, Tassone, Giusy, Clementi, Letizia, Franci, Lorenzo, Munier, Claire C, Cau, Ylenia, Mori, Mattia, Chiariello, Mario, Angelucci, Adriano, Perry, Matthew W. D, Pozzi, Cecilia, Mangani, Stefano, Botta, Maurizio
Published in ACS chemical biology (17.04.2020)
Published in ACS chemical biology (17.04.2020)
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Spiro-fused Pyrrolidine, Piperidine, and Oxindole Scaffolds from Lactams
Hirschhäuser, Christoph, Parker, Jeremy S, Perry, Matthew W. D, Haddow, Mairi F, Gallagher, Timothy
Published in Organic letters (21.09.2012)
Published in Organic letters (21.09.2012)
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14-3-3 modulation of the inflammatory response
Munier, Claire C., Ottmann, Christian, Perry, Matthew W.D.
Published in Pharmacological research (01.01.2021)
Published in Pharmacological research (01.01.2021)
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Glucocorticoid receptor Thr524 phosphorylation by MINK1 induces interactions with 14-3-3 protein regulators
Munier, Claire C., De Maria, Leonardo, Edman, Karl, Gunnarsson, Anders, Longo, Marianna, MacKintosh, Carol, Patel, Saleha, Snijder, Arjan, Wissler, Lisa, Brunsveld, Luc, Ottmann, Christian, Perry, Matthew W.D.
Published in The Journal of biological chemistry (01.01.2021)
Published in The Journal of biological chemistry (01.01.2021)
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Designing Selective Drug-like Molecular Glues for the Glucocorticoid Receptor/14-3‑3 Protein–Protein Interaction
Pallesen, Jakob S., Munier, Claire C., Bosica, Francesco, Andrei, Sebastian A., Edman, Karl, Gunnarsson, Anders, La Sala, Giuseppina, Putra, Okky Dwichandra, Srdanović, Sonja, Wilson, Andrew J., Wissler, Lisa, Ottmann, Christian, Perry, Matthew W. D., O’Mahony, Gavin
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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Correction to “Designing Selective Drug-like Molecular Glues for the Glucocorticoid Receptor/14-3‑3 Protein–Protein Interaction”
Pallesen, Jakob S., Munier, Claire C., Bosica, Francesco, Andrei, Sebastian A., Edman, Karl, Gunnarsson, Anders, La Sala, Giuseppina, Putra, Okky Dwichandra, Srdanović, Sonja, Wilson, Andrew J., Wissler, Lisa, Ottmann, Christian, Perry, Matthew W. D., O’Mahony, Gavin
Published in Journal of medicinal chemistry (09.02.2023)
Published in Journal of medicinal chemistry (09.02.2023)
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