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Published in Journal of medicinal chemistry (01.03.1992)
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Synthesis and Structure−Affinity Relationship Investigations of 5-Heteroaryl-Substituted Analogues of the Antipsychotic Sertindole. A New Class of Highly Selective α1 Adrenoceptor Antagonists
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Published in Journal of medicinal chemistry (16.01.2003)
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First Demonstration of a Functional Role for Central Nervous System Betaine/γ-Aminobutyric Acid Transporter (mGAT2) Based on Synergistic Anticonvulsant Action among Inhibitors of mGAT1 and mGAT2
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Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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Selective inhibitors of GABA uptake: synthesis and molecular pharmacology of 4- N-methylamino-4,5,6,7-tetrahydrobenzo[ d]isoxazol-3-ol analogues
Clausen, Rasmus P., Moltzen, Ejner K., Perregaard, Jens, Lenz, Sibylle M., Sanchez, Connie, Falch, Erik, Frølund, Bente, Bolvig, Tina, Sarup, Alan, Larsson, Orla M., Schousboe, Arne, Krogsgaard-Larsen, Povl
Published in Bioorganic & medicinal chemistry (01.02.2005)
Published in Bioorganic & medicinal chemistry (01.02.2005)
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Synthesis and structure-affinity relationship investigations of 5-heteroaryl-substituted analogues of the antipsychotic sertindole. A new class of highly selective alpha(1) adrenoceptor antagonists
Balle, T, Perregaard, J, Ramirez, MT, Larsen, AK, Soby, KK, Liljefors, T, Andersen, K
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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Serotonin 5-HT2 Receptor, Dopamine D2 Receptor, and α1 Adrenoceptor Antagonists. Conformationally Flexible Analogues of the Atypical Antipsychotic Sertindole
Andersen, Kim, Liljefors, Tommy, Hyttel, John, Perregaard, Jens
Published in Journal of medicinal chemistry (13.09.1996)
Published in Journal of medicinal chemistry (13.09.1996)
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Synthesis and structure-affinity relationship investigations of 5-aminomethyl and 5-carbamoyl analogues of the antipsychotic sertindole. A new class of selective α1 adrenoceptor antagonists
BALLE, Thomas, PERREGAARD, Jens, LARSEN, Anna K, RAMIREZ, Martha Teresa, SØBY, Karina Krøjer, LILJEFORS, Tommy, ANDERSEN, Kim
Published in Bioorganic & medicinal chemistry (01.03.2003)
Published in Bioorganic & medicinal chemistry (01.03.2003)
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New α1-adrenoceptor antagonists derived from the antipsychotic sertindole - carbon-11 labelling and pet examination of brain uptake in the cynomolgus monkey
Balle, Thomas, Halldin, Christer, Andersen, Linus, Hjorth Alifrangis, Lene, Badolo, Lassina, Gjervig Jensen, Klaus, Chou, Yuan-Wha, Andersen, Kim, Perregaard, Jens, Farde, Lars
Published in Nuclear medicine and biology (01.04.2004)
Published in Nuclear medicine and biology (01.04.2004)
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First Demonstration of a Functional Role for Central Nervous System Betaine/γ-Aminobutyric Acid Transporter (mGAT2) Based on Synergistic Anticonvulsant Action among Inhibitors of mGAT1 and mGAT2
H. Steve White, William P. Watson, Suzanne L. Hansen, Scott Slough, Jens Perregaard, Alan Sarup, Tina Bolvig, Gitte Petersen, Orla M. Larsson, Rasmus P. Clausen, Bente Frølund, Erik Falch, Povl Krogsgaard-Larsen, Arne Schousboe
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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First demonstration of a functional role for central nervous system betaine/{gamma}-aminobutyric acid transporter (mGAT2) based on synergistic anticonvulsant action among inhibitors of mGAT1 and mGAT2
White, H Steve, Watson, William P, Hansen, Suzanne L, Slough, Scott, Perregaard, Jens, Sarup, Alan, Bolvig, Tina, Petersen, Gitte, Larsson, Orla M, Clausen, Rasmus P, Frølund, Bente, Falch, Erik, Krogsgaard-Larsen, Povl, Schousboe, Arne
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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Synthesis and Structure−Affinity Relationship Investigations of 5-Heteroaryl-Substituted Analogues of the Antipsychotic Sertindole. A New Class of Highly Selective α 1 Adrenoceptor Antagonists
Balle, Thomas, Perregaard, Jens, Ramirez, Martha Teresa, Larsen, Anna Kirstine, Søby, Karina Krøjer, Liljefors, Tommy, Andersen, Kim
Published in Journal of medicinal chemistry (01.01.2003)
Published in Journal of medicinal chemistry (01.01.2003)
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Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues
Falch, Erik, Perregaard, Jens, Frølund, Bente, Søkilde, Birgitte, Buur, Anders, Hansen, Lene M, Frydenvang, Karla, Brehm, Lotte, Bolvig, Tina, Larsson, Orla M, Sanchez, Connie, White, Harold S, Schousboe, Arne, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (30.12.1999)
Published in Journal of medicinal chemistry (30.12.1999)
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