Aurora Isoform Selectivity: Design and Synthesis of Imidazo[4,5‑b]pyridine Derivatives as Highly Selective Inhibitors of Aurora‑A Kinase in Cells
Bavetsias, Vassilios, Faisal, Amir, Crumpler, Simon, Brown, Nathan, Kosmopoulou, Magda, Joshi, Amar, Atrash, Butrus, Pérez-Fuertes, Yolanda, Schmitt, Jessica A, Boxall, Katherine J, Burke, Rosemary, Sun, Chongbo, Avery, Sian, Bush, Katherine, Henley, Alan, Raynaud, Florence I, Workman, Paul, Bayliss, Richard, Linardopoulos, Spiros, Blagg, Julian
Published in Journal of medicinal chemistry (27.11.2013)
Published in Journal of medicinal chemistry (27.11.2013)
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Asymmetric Strecker Synthesis of α-Arylglycines
Pérez-Fuertes, Yolanda, Taylor, James E, Tickell, David A, Mahon, Mary F, Bull, Steven D, James, Tony D
Published in Journal of organic chemistry (05.08.2011)
Published in Journal of organic chemistry (05.08.2011)
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Simple protocols for NMR analysis of the enantiomeric purity of chiral diols
Bull, Steven D, James, Tony D, Kelly, Andrew M, Pérez-Fuertes, Yolanda, Fossey, John S, Yeste, Sonia Lozano
Published in Nature protocols (01.02.2008)
Published in Nature protocols (01.02.2008)
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Journal Article
Simple protocols for NMR analysis of the enantiomeric purity of chiral primary amines
Bull, Steven D, James, Tony D, Pérez-Fuertes, Yolanda, Kelly, Andrew M, Fossey, John S, Powell, Magdalena E
Published in Nature protocols (01.02.2008)
Published in Nature protocols (01.02.2008)
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Bromonium Ion Induced Transannular Oxonium Ion Formation−Fragmentation in Model Obtusallene Systems and Structural Reassignment of Obtusallenes V−VII
Braddock, D. Christopher, Millan, David S, Pérez-Fuertes, Yolanda, Pouwer, Rebecca H, Sheppard, Richard N, Solanki, Savade, White, Andrew J. P
Published in Journal of organic chemistry (06.03.2009)
Published in Journal of organic chemistry (06.03.2009)
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The stereochemical course of bromoetherification of enynes
Braddock, D. Christopher, Bhuva, Roshni, Perez-Fuertes, Yolanda, Pouwer, Rebecca, Roberts, Craig A., Ruggiero, Andrea, Stokes, Elaine S. E., White, Andrew J. P.
Published in Chemical communications (Cambridge, England) (01.01.2008)
Published in Chemical communications (Cambridge, England) (01.01.2008)
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A Biosynthetically-Inspired Synthesis of the Tetrahydrofuran Core of Obtusallenes II and IV
Braddock, D. Christopher, Bhuva, Roshni, Millan, David S, Pérez-Fuertes, Yolanda, Roberts, Craig A, Sheppard, Richard N, Solanki, Savade, Stokes, Elaine S. E, White, Andrew J. P
Published in Organic letters (01.02.2007)
Published in Organic letters (01.02.2007)
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7-(Pyrazol-4-yl)-3H-imidazo[4,5-b]pyridine-based derivatives for kinase inhibition: Co-crystallisation studies with Aurora-A reveal distinct differences in the orientation of the pyrazole N1-substituent
Bavetsias, Vassilios, Pérez-Fuertes, Yolanda, McIntyre, Patrick J., Atrash, Butrus, Kosmopoulou, Magda, O’Fee, Lisa, Burke, Rosemary, Sun, Chongbo, Faisal, Amir, Bush, Katherine, Avery, Sian, Henley, Alan, Raynaud, Florence I., Linardopoulos, Spiros, Bayliss, Richard, Blagg, Julian
Published in Bioorganic & medicinal chemistry letters (01.10.2015)
Published in Bioorganic & medicinal chemistry letters (01.10.2015)
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Journal Article
Simple Protocol for NMR Analysis of the Enantiomeric Purity of Primary Amines
Pérez-Fuertes, Yolanda, Kelly, Andrew M, Johnson, Andrew L, Arimori, Susumu, Bull, Steven D, James, Tony D
Published in Organic letters (16.02.2006)
Published in Organic letters (16.02.2006)
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Journal Article
Simple Protocol for NMR Analysis of the Enantiomeric Purity of Diols
Kelly, Andrew M, Pérez-Fuertes, Yolanda, Arimori, Susumu, Bull, Steven D, James, Tony D
Published in Organic letters (11.05.2006)
Published in Organic letters (11.05.2006)
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Design, synthesis and structure-activity relationships of a novel class of sulfonylpyridine inhibitors of Interleukin-2 inducible T-cell kinase (ITK)
Trani, Giancarlo, Barker, John J., Bromidge, Steven M., Brookfield, Frederick A., Burch, Jason D., Chen, Yuan, Eigenbrot, Charles, Heifetz, Alexander, Ismaili, M. Hicham A., Johnson, Adam, Krulle, Thomas M., MacKinnon, Colin H., Maghames, Rosemary, McEwan, Paul A., Montalbetti, Christian A. G. N., Ortwine, Daniel F., Perez-Fuertes, Yolanda, Vaidya, Darshan G., Wang, Xiaolu, Zarrin, Ali A., Pei, Zhonghua
Published in Bioorganic & medicinal chemistry letters (15.12.2014)
Published in Bioorganic & medicinal chemistry letters (15.12.2014)
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Structure-based design and synthesis of potent benzothiazole inhibitors of interleukin-2 inducible T cell kinase (ITK)
MacKinnon, Colin H., Lau, Kevin, Burch, Jason D., Chen, Yuan, Dines, Jonathon, Ding, Xiao, Eigenbrot, Charles, Heifetz, Alexander, Jaochico, Allan, Johnson, Adam, Kraemer, Joachim, Kruger, Susanne, Krülle, Thomas M., Liimatta, Marya, Ly, Justin, Maghames, Rosemary, Montalbetti, Christian A.G.N., Ortwine, Daniel F., Pérez-Fuertes, Yolanda, Shia, Steven, Stein, Daniel B., Trani, Giancarlo, Vaidya, Darshan G., Wang, Xiaolu, Bromidge, Steven M., Wu, Lawren C., Pei, Zhonghua
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
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ChemInform Abstract: Asymmetric Strecker Synthesis of α-Arylglycines
Perez-Fuertes, Yolanda, Taylor, James E., Tickell, David A., Mahon, Mary F., Bull, Steven D., James, Tony D.
Published in ChemInform (06.12.2011)
Published in ChemInform (06.12.2011)
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ChemInform Abstract: Bromonium Ion Induced Transannular Oxonium Ion Formation-Fragmentation in Model Obtusallene Systems and Structural Reassignment of Obtusallenes V-VII
Braddock, D. Christopher, Millan, David S., Perez-Fuertes, Yolanda, Pouwer, Rebecca H., Sheppard, Richard N., Solanki, Savade, White, Andrew J. P.
Published in ChemInform (28.07.2009)
Published in ChemInform (28.07.2009)
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Journal Article
ChemInform Abstract: The Stereochemical Course of Bromoetherification of Enynes
Braddock, D. Christopher, Bhuva, Roshni, Perez-Fuertes, Yolanda, Pouwer, Rebecca, Roberts, Craig A., Ruggiero, Andrea, Stokes, Elaine S. E., White, Andrew J. P.
Published in ChemInform (15.07.2008)
Published in ChemInform (15.07.2008)
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BENZOXAZINONE DERIVATIVES AND ANALOGUES THEREOF AS MODULATORS OF TNF ACTIVITY
CHOVATIA, PRAFULKUMAR TULSHIBHAI, MANDAL, AJAY, JONES, SEVERINE DANIELLE, LECOMTE, FABIEN CLAUDE, PORTER, JOHN ROBERT, JOHNSON, JAMES ANDREW, FOULKES, GREGORY, SMYTH, DONALD, LOWE, MARTIN ALEXANDER, ZHU, ZHAONING, PALMER, CHRISTOPHER FRANCIS, PEREZ-FUERTES, YOLANDA, TRANI, GIANCARLO, NORMAN, TIMOTHY JOHN, KROEPLIEN, BORIS, LOKE, PUI LENG, BRACE, GARETH NEIL, UDDIN, MUHAMMED
Year of Publication 15.12.2016
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Year of Publication 15.12.2016
Patent
Simple Protocol for NMR Analysis of the Enantiomeric Purity of Primary Amines
Pérez-Fuertes, Yolanda, Kelly, Andrew M, Johnson, Andrew L, Arimori, Susumu, Bull, Steven D, James, Tony D
Published in Organic letters (11.05.2006)
Published in Organic letters (11.05.2006)
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BENZOXAZINONE DERIVATIVES AND ANALOGUES THEREOF AS MODULATORS OF TNF ACTIVITY
ZHU, Zhaoning, PEREZ-FUERTES, Yolanda, PALMER, Christopher Francis, PORTER, John Robert, KROEPLIEN, Boris, BRACE, Gareth Neil, LOKE, Pui Leng, JOHNSON, James Andrew, CHOVATIA, Prafulkumar Tulshibhai, NORMAN, Timothy John, LOWE, Martin Alexander, UDDIN, Muhammed, MANDAL, Ajay, SMYTH, Donald, TRANI, Giancarlo, FOULKES, Gregory, JONES, Severine Danielle, LECOMTE, Fabien Claude
Year of Publication 14.04.2020
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Year of Publication 14.04.2020
Patent
Non-linear effects operate and dynamic ligand exchange occurs when chiral BINOL–boron Lewis acids are used for asymmetric catalysis
Cros, Jean Philippe, Pérez-Fuertes, Yolanda, Thatcher, Michael J, Arimori, Susumu, Bull, Steven D, James, Tony D
Published in Tetrahedron: asymmetry (18.07.2003)
Published in Tetrahedron: asymmetry (18.07.2003)
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