Geranylgeranyltransferase I Inhibitors Target RalB To Inhibit Anchorage-Dependent Growth and Induce Apoptosis and RalA To Inhibit Anchorage-Independent Growth
Falsetti, Samuel C., Wang, De-an, Peng, Hairuo, Carrico, Dora, Cox, Adrienne D., Der, Channing J., Hamilton, Andrew D., Sebti, Saïd M.
Published in Molecular and Cellular Biology (01.11.2007)
Published in Molecular and Cellular Biology (01.11.2007)
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Journal Article
Novel Bicyclic Piperazine Derivatives of Triazolotriazine and Triazolopyrimidines as Highly Potent and Selective Adenosine A2A Receptor Antagonists
PENG, Hairuo, KUMARAVEL, Gnanasambandam, YAO, Gang, SHA, Li, WANG, Joy, VAN VLIJMEN, Herman, BOHNERT, Tonika, HUANG, Carol, VU, Chi B., ENSINGER, Carol L., CHANG, Hexi, ENGBER, Thomas M., WHALLEY, Eric T., PETTER, Russell C.
Published in Journal of medicinal chemistry (02.12.2004)
Published in Journal of medicinal chemistry (02.12.2004)
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Journal Article
Discovery of 4-aminomethylphenylacetic acids as γ-secretase modulators via a scaffold design approach
Xin, Zhili, Peng, Hairuo, Zhang, Andrew, Talreja, Tina, Kumaravel, Gnanasambandam, Xu, Lin, Rohde, Ellen, Jung, Mi-yong, Shackett, Melanie N., Kocisko, David, Chollate, Sowmya, Dunah, Anthone W., Snodgrass-Belt, Pamela A., Moore Arnold, H., Taveras, Arthur G., Rhodes, Kenneth J., Scannevin, Robert H.
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
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Journal Article
Synthesis and evaluation of potent, highly-selective, 3-aryl-piperazinone inhibitors of protein geranylgeranyltransferase-I
Peng, H, Carrico, D, Van, T, Blaskovich, M, Bucher, C, Pusateri, EE, Sebti, SM, Hamilton, AD
Published in Organic & biomolecular chemistry (01.01.2006)
Published in Organic & biomolecular chemistry (01.01.2006)
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Journal Article
Blockade of Protein Geranylgeranylation Inhibits Cdk2-Dependent p27Kip1 Phosphorylation on Thr187 and Accumulates p27Kip1 in the Nucleus: Implications for Breast Cancer Therapy
Kazi, Aslamuzzaman, Carie, Adam, Blaskovich, Michelle A., Bucher, Cynthia, Thai, Van, Moulder, Stacy, Peng, Hairuo, Carrico, Dora, Pusateri, Erin, Pledger, Warren J., Berndt, Norbert, Hamilton, Andrew, Sebti, Saïd M.
Published in Molecular and Cellular Biology (01.04.2009)
Published in Molecular and Cellular Biology (01.04.2009)
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Journal Article
Syntheses and Biological Activities of a Novel Group of Steroidal Derived Inhibitors for Human CDC25A Protein Phosphatase
Peng, Hairuo, Xie, Wenge, Otterness, Diane M, Cogswell, John P, McConnell, Randy T, Carter, H. Luke, Powis, Garth, Abraham, Robert T, Zalkow, Leon H
Published in Journal of medicinal chemistry (01.03.2001)
Published in Journal of medicinal chemistry (01.03.2001)
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Journal Article
Structure–activity relationship of Aza-steroids as PI-PLC inhibitors
Xie, Wenge, Peng, Hairuo, Kim, Deog-Il, Kunkel, Mark, Powis, Garth, Zalkow, Leon H.
Published in Bioorganic & medicinal chemistry (01.05.2001)
Published in Bioorganic & medicinal chemistry (01.05.2001)
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Journal Article
3β-Hydroxy-6-aza-cholestane and related analogues as phosphatidylinositol specific phospholipase C (PI-PLC) inhibitors with antitumor activity
WENGE XIE, HAIRUO PENG, ZALKOW, L. H, LI, Y.-H, CHENG ZHU, POWIS, G, KUNKEL, M
Published in Bioorganic & medicinal chemistry (01.04.2000)
Published in Bioorganic & medicinal chemistry (01.04.2000)
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Journal Article
Six New Eremophilane Derivatives from Two Ligularia Species
Zhao, Yu, Peng, Hairuo, Jia, Zhongjian
Published in Journal of natural products (Washington, D.C.) (01.12.1994)
Published in Journal of natural products (Washington, D.C.) (01.12.1994)
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Journal Article
Steroidal derived acids as inhibitors of human Cdc25A protein phosphatase
HAIRUO PENG, WENGE XIE, KIM, D.-I, ZALKOW, L. H, POWIS, G, OTTERNESS, D. M, ABRAHAM, R. T
Published in Bioorganic & medicinal chemistry (01.02.2000)
Published in Bioorganic & medicinal chemistry (01.02.2000)
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Journal Article
Investigating small molecules to inhibit germinal center kinase-like kinase (GLK/MAP4K3) upstream of PKCθ phosphorylation: Potential therapy to modulate T cell dependent immunity
May-Dracka, Tricia L., Arduini, Robert, Bertolotti-Ciarlet, Andrea, Bhisetti, Govinda, Brickelmaier, Margot, Cahir-McFarland, Ellen, Enyedy, Istvan, Fontenot, Jason D., Hesson, Thomas, Little, Kevin, Lyssikatos, Joe, Marcotte, Douglas, McKee, Timothy, Murugan, Paramasivam, Patterson, Thomas, Peng, Hairuo, Rushe, Mia, Silvian, Laura, Spilker, Kerri, Wu, Ping, Xin, Zhili, Burkly, Linda C.
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
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Journal Article
BIIB042, a novel γ-secretase modulator, reduces amyloidogenic Aβ isoforms in primates and rodents and plaque pathology in a mouse model of Alzheimer's disease
Scannevin, Robert H., Chollate, Sowmya, Brennan, Melanie S., Snodgrass-Belt, Pamela A., Peng, Hairuo, Xu, Lin, Jung, Mi-young, Bussiere, Thierry, Arastu, Mahin F., Talreja, Tina, Xin, Zhili, Dunstan, Robert W., Fahrer, Diana, Rohde, Ellen, Dunah, Anthone W., Wang, Joy, Kumaravel, Gnanasambandam, Taveras, Arthur G., Moore Arnold, H., Rhodes, Kenneth J.
Published in Neuropharmacology (01.04.2016)
Published in Neuropharmacology (01.04.2016)
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Journal Article
ATX MODULATING AGENTS
MI SHA, GNANASAMBANDAM KUMARAVEL, LEI ZHANG, MA BIN, WANG DEPING, XIN ZHILI, PENG HAIRUO, SUN LIHONG, SHAO ZHAOHUI, ARTHUR TAVERAS, KEVIN GUCKIAN
Year of Publication 30.08.2018
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Year of Publication 30.08.2018
Patent
Discovery of BIIB042, a Potent, Selective, and Orally Bioavailable γ-Secretase Modulator
Peng, Hairuo, Talreja, Tina, Xin, Zhili, Cuervo, J. Hernan, Kumaravel, Gnanasambandam, Humora, Michael J, Xu, Lin, Rohde, Ellen, Gan, Lawrence, Jung, Mi-young, Shackett, Melanie N, Chollate, Sowmya, Dunah, Anthone W, Snodgrass-belt, Pamela A, Arnold, H. Moore, Taveras, Arthur G, Rhodes, Kenneth J, Scannevin, Robert H
Published in ACS medicinal chemistry letters (13.10.2011)
Published in ACS medicinal chemistry letters (13.10.2011)
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Journal Article