Quantitation of isocitrate dehydrogenase (IDH)-induced D and L enantiomers of 2-hydroxyglutaric acid in biological fluids by a fully validated liquid tandem mass spectrometry method, suitable for clinical applications
Poinsignon, Vianney, Mercier, Lionel, Nakabayashi, Koïchi, David, Muriel D., Lalli, Alexandre, Penard- Lacronique, Virginie, Quivoron, Cyril, Saada, Véronique, De Botton, Stéphane, Broutin, Sophie, Paci, Angelo
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2016)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2016)
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Enasidenib induces acute myeloid leukemia cell differentiation to promote clinical response
Amatangelo, Michael D., Quek, Lynn, Shih, Alan, Stein, Eytan M., Roshal, Mikhail, David, Muriel D., Marteyn, Benoit, Farnoud, Noushin Rahnamay, de Botton, Stephane, Bernard, Olivier A., Wu, Bin, Yen, Katharine E., Tallman, Martin S., Papaemmanuil, Elli, Penard-Lacronique, Virginie, Thakurta, Anjan, Vyas, Paresh, Levine, Ross L.
Published in Blood (10.08.2017)
Published in Blood (10.08.2017)
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Targeted Inhibition of Mutant IDH2 in Leukemia Cells Induces Cellular Differentiation
Wang, Fang, Travins, Jeremy, DeLaBarre, Byron, Penard-Lacronique, Virginie, Schalm, Stefanie, Hansen, Erica, Straley, Kimberly, Kernytsky, Andrew, Liu, Wei, Gliser, Camelia, Yang, Hua, Gross, Stefan, Artin, Erin, Saada, Veronique, Mylonas, Elena, Quivoron, Cyril, Popovici-Muller, Janeta, Saunders, Jeffrey O., Salituro, Francesco G., Yan, Shunqi, Murray, Stuart, Wei, Wentao, Gao, Yi, Dang, Lenny, Dorsch, Marion, Agresta, Sam, Schenkein, David P., Biller, Scott A., Su, Shinsan M., de Botton, Stephane, Yen, Katharine E.
Published in Science (American Association for the Advancement of Science) (03.05.2013)
Published in Science (American Association for the Advancement of Science) (03.05.2013)
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Senescence is a Spi1-induced anti-proliferative mechanism in primary hematopoietic cells
Delestré, Laure, Cui, Hengxiang, Esposito, Michela, Quiveron, Cyril, Mylonas, Elena, Penard-Lacronique, Virginie, Bischof, Oliver, Guillouf, Christel
Published in Haematologica (Roma) (01.11.2017)
Published in Haematologica (Roma) (01.11.2017)
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Activating mutations in human acute megakaryoblastic leukemia
Malinge, Sébastien, Ragu, Christine, Della-Valle, Veronique, Pisani, Didier, Constantinescu, Stefan N., Perez, Christelle, Villeval, Jean-Luc, Reinhardt, Dirk, Landman-Parker, Judith, Michaux, Lucienne, Dastugue, Nicole, Baruchel, André, Vainchenker, William, Bourquin, Jean-Pierre, Penard-Lacronique, Virginie, Bernard, Olivier A.
Published in Blood (15.11.2008)
Published in Blood (15.11.2008)
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Gene-Environment Interaction Modulated by Allelic Heterogeneity in Inflammatory Diseases
Chamaillard, Mathias, Philpott, Dana, Girardin, Stephen E., Zouali, Habib, Lesage, Suzanne, Chareyre, Fabrice, Bui, The Hung, Giovannini, Marco, Zaehringer, Ulrich, Penard-Lacronique, Virginie, Sansonetti, Philippe J., Hugot, Jean-Pierre, Thomas, Gilles
Published in Proceedings of the National Academy of Sciences - PNAS (18.03.2003)
Published in Proceedings of the National Academy of Sciences - PNAS (18.03.2003)
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The TEL-Jak2 oncoprotein induces Socs1 expression and altered cytokine response in Ba/F3 cells
Monni, R, Santos, S C, Mauchauffe, M, Berger, R, Ghysdael, J, Gouilleux, F, Gisselbrecht, S, Bernard, O, Penard-Lacronique, V
Published in Oncogene (15.02.2001)
Published in Oncogene (15.02.2001)
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A small molecule inhibitor of mutant IDH2 rescues cardiomyopathy in a D-2-hydroxyglutaric aciduria type II mouse model
Wang, Fang, Travins, Jeremy, Lin, Zhizhong, Si, Yaguang, Chen, Yue, Powe, Josh, Murray, Stuart, Zhu, Dongwei, Artin, Erin, Gross, Stefan, Santiago, Stephanie, Steadman, Mya, Kernytsky, Andrew, Straley, Kimberly, Lu, Chenming, Pop, Ana, Struys, Eduard A., Jansen, Erwin E. W., Salomons, Gajja S., David, Muriel D., Quivoron, Cyril, Penard-Lacronique, Virginie, Regan, Karen S., Liu, Wei, Dang, Lenny, Yang, Hua, Silverman, Lee, Agresta, Samuel, Dorsch, Marion, Biller, Scott, Yen, Katharine, Cang, Yong, Su, Shin-San Michael, Jin, Shengfang
Published in Journal of inherited metabolic disease (01.11.2016)
Published in Journal of inherited metabolic disease (01.11.2016)
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NUP98-MLL fusion in human acute myeloblastic leukemia
Kaltenbach, Sophie, Soler, Gwendoline, Barin, Carole, Gervais, Carine, Bernard, Olivier A., Penard-Lacronique, Virginie, Romana, Serge P.
Published in Blood (30.09.2010)
Published in Blood (30.09.2010)
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Functional analysis of the NUP98-CCDC28A fusion protein
PETIT, Arnaud, RAGU, Christine, BERNARD, Olivier A, ROMANA, Serge, PENARD-LACRONIQUE, Virginie, SOLER, Gwendoline, OTTOLENGHI, Chris, SCHLUTH, Caroline, RADFORD-WEISS, Isabelle, SCHNEIDER-MAUNOURY, Sylvie, CALLEBAUT, Isabelle, DASTUGUE, Nicole, DRABKIN, Harry A
Published in Haematologica (Roma) (01.03.2012)
Published in Haematologica (Roma) (01.03.2012)
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Clonal heterogeneity of acute myeloid leukemia treated with the IDH2 inhibitor enasidenib
Quek, Lynn, David, Muriel D., Kennedy, Alison, Metzner, Marlen, Amatangelo, Michael, Shih, Alan, Stoilova, Bilyana, Quivoron, Cyril, Heiblig, Maël, Willekens, Christophe, Saada, Véronique, Alsafadi, Samar, Vijayabaskar, M. S., Peniket, Andy, Bernard, Oliver A., Agresta, Sam, Yen, Katharine, MacBeth, Kyle, Stein, Eytan, Vassiliou, George S., Levine, Ross, De Botton, Stephane, Thakurta, Anjan, Penard-Lacronique, Virginie, Vyas, Paresh
Published in Nature medicine (01.08.2018)
Published in Nature medicine (01.08.2018)
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AG-221, a First-in-Class Therapy Targeting Acute Myeloid Leukemia Harboring Oncogenic IDH2 Mutations
Yen, Katharine, Travins, Jeremy, Wang, Fang, David, Muriel D, Artin, Erin, Straley, Kimberly, Padyana, Anil, Gross, Stefan, DeLaBarre, Byron, Tobin, Erica, Chen, Yue, Nagaraja, Raj, Choe, Sung, Jin, Lei, Konteatis, Zenon, Cianchetta, Giovanni, Saunders, Jeffrey O, Salituro, Francesco G, Quivoron, Cyril, Opolon, Paule, Bawa, Olivia, Saada, Véronique, Paci, Angelo, Broutin, Sophie, Bernard, Olivier A, de Botton, Stéphane, Marteyn, Benoît S, Pilichowska, Monika, Xu, YingXia, Fang, Cheng, Jiang, Fan, Wei, Wentao, Jin, Shengfang, Silverman, Lee, Liu, Wei, Yang, Hua, Dang, Lenny, Dorsch, Marion, Penard-Lacronique, Virginie, Biller, Scott A, Su, Shin-San Michael
Published in Cancer discovery (01.05.2017)
Published in Cancer discovery (01.05.2017)
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Coordinated alterations in RNA splicing and epigenetic regulation drive leukaemogenesis
Yoshimi, Akihide, Lin, Kuan-Ting, Wiseman, Daniel H., Rahman, Mohammad Alinoor, Pastore, Alessandro, Wang, Bo, Lee, Stanley Chun-Wei, Micol, Jean-Baptiste, Zhang, Xiao Jing, de Botton, Stephane, Penard-Lacronique, Virginie, Stein, Eytan M., Cho, Hana, Miles, Rachel E., Inoue, Daichi, Albrecht, Todd R., Somervaille, Tim C. P., Batta, Kiran, Amaral, Fabio, Simeoni, Fabrizio, Wilks, Deepti P., Cargo, Catherine, Intlekofer, Andrew M., Levine, Ross L., Dvinge, Heidi, Bradley, Robert K., Wagner, Eric J., Krainer, Adrian R., Abdel-Wahab, Omar
Published in Nature (London) (01.10.2019)
Published in Nature (London) (01.10.2019)
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Discovery of AG-120 (Ivosidenib): A First-in-Class Mutant IDH1 Inhibitor for the Treatment of IDH1 Mutant Cancers
Popovici-Muller, Janeta, Lemieux, René M, Artin, Erin, Saunders, Jeffrey O, Salituro, Francesco G, Travins, Jeremy, Cianchetta, Giovanni, Cai, Zhenwei, Zhou, Ding, Cui, Dawei, Chen, Ping, Straley, Kimberly, Tobin, Erica, Wang, Fang, David, Muriel D, Penard-Lacronique, Virginie, Quivoron, Cyril, Saada, Véronique, de Botton, Stéphane, Gross, Stefan, Dang, Lenny, Yang, Hua, Utley, Luke, Chen, Yue, Kim, Hyeryun, Jin, Shengfang, Gu, Zhiwei, Yao, Gui, Luo, Zhiyong, Lv, Xiaobing, Fang, Cheng, Yan, Liping, Olaharski, Andrew, Silverman, Lee, Biller, Scott, Su, Shin-San M, Yen, Katharine
Published in ACS medicinal chemistry letters (12.04.2018)
Published in ACS medicinal chemistry letters (12.04.2018)
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Enasidenib treatment in two individuals with D-2-hydroxyglutaric aciduria carrying a germline IDH2 mutation
Geoerger, Birgit, Schiff, Manuel, Penard-Lacronique, Virginie, Darin, Niklas, Saad, Selim-Maria, Duchon, Clarisse, Lamazière, Antonin, Desmons, Aurore, Pontoizeau, Clément, Berlanga, Pablo, Ducassou, Stéphane, Yen, Katharine, Su, Michael, Schenkein, David, Ottolenghi, Chris, De Botton, Stéphane
Published in Nature Medicine (01.06.2023)
Published in Nature Medicine (01.06.2023)
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Dysregulation of Stem-Progenitor and Differentiation Programmes through Modulation of Bivalent Chromatin Drives Leukemogenesis in Mutant IDH2 Acute Myeloid Leukaemia
Silveira, Douglas RA RA, Chatzikyriakou, Prodromos, Casares Alaez, Maria del Pilar, Mackie, Sarah, Hulks, Roan, Yavorska, Olena, Siejka-Zielinska, Paulina, Metzner, Marlen, Smith, Alastair, Usukhbayar, Batchimeg, Penard-Lacronique, Virginie, Song, Chunxiao, Gandhi, Anita K., Hasan, Maroof, Vyas, Paresh, Milne, Thomas A., Kriaucionis, Skirmantas, Quek, Lynn
Published in Blood (15.11.2022)
Published in Blood (15.11.2022)
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Abstract 280: Aberrant β-catenin signaling from the bone marrow niche leads to transformation of IDH1/2 -mutant hematopoietic stem cells and compromises response to IDH1/2 inhibitors
Vgenopoulou, Paraskevi, Flores, Luis, Mosialou, Ioanna, Zhao, Junfei, Liu, X. Shawn, Sung, Pamela, Penard-Lacronique, Virginie, Carroll, Martin, Kousteni, Stavroula
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Repressed Chromatin Drives Leukaemogenesis in Mutant IDH2 Acute Myeloid Leukaemia Via Inhibition of Granulocyte Differentiation and Cell Cycle Progression
Silveira, Douglas RA, Chatzikyriakou, Prodromos, Yavorska, Olena, Mackie, Sarah, Hulks, Roan, Siejka-Zielinska, Paulina, Corby, Anna, Smith, Alastair, Brown, Benjamin, Metzner, Marlen, Milne, Thomas A., Penard-Lacronique, Virginie, Song, Chunxiao, Hasan, Maroof, Thakurta, Anjan, Vyas, Paresh, Kriaucionis, Skirmantas, Quek, Lynn
Published in Blood (23.11.2021)
Published in Blood (23.11.2021)
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