A Selective and Brain Penetrant p38αMAPK Inhibitor Candidate for Neurologic and Neuropsychiatric Disorders That Attenuates Neuroinflammation and Cognitive Dysfunction
Roy, Saktimayee M, Minasov, George, Arancio, Ottavio, Chico, Laura W, Van Eldik, Linda J, Anderson, Wayne F, Pelletier, Jeffrey C, Watterson, D. Martin
Published in Journal of medicinal chemistry (13.06.2019)
Published in Journal of medicinal chemistry (13.06.2019)
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Development of Novel In Vivo Chemical Probes to Address CNS Protein Kinase Involvement in Synaptic Dysfunction
Watterson, D Martin, Grum-Tokars, Valerie L, Roy, Saktimayee M, Schavocky, James P, Bradaric, Brinda Desai, Bachstetter, Adam D, Xing, Bin, Dimayuga, Edgardo, Saeed, Faisal, Zhang, Hong, Staniszewski, Agnieszka, Pelletier, Jeffrey C, Minasov, George, Anderson, Wayne F, Arancio, Ottavio, Van Eldik, Linda J
Published in PloS one (26.06.2013)
Published in PloS one (26.06.2013)
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A Spontaneous Melanoma Mouse Model Applicable for a Longitudinal Chemotherapy and Immunotherapy Study
Eddy, Kevinn, Gupta, Kajal, Pelletier, Jeffrey C., Isola, Allison L., Marinaro, Christina, Rasheed, Maryam Abdur, Campagnolo, Joseph, Eddin, Mohamad Naser, Rossi, Marco, Fateeva, Anna, Reuhl, Kenneth, Shah, Raj, Robinson, Ann K., Chaly, Anna, Freeman, Katie B., Chen, Wenjin, Diaz, Jesus, Furmanski, Philip, Silk, Ann W., Reitz, Allen B., Zloza, Andrew, Chen, Suzie
Published in Journal of investigative dermatology (01.10.2023)
Published in Journal of investigative dermatology (01.10.2023)
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Highly potent, broadly active antifungal agents for the treatment of invasive fungal infections
Baugh, Simon D.P., Chaly, Anna, Weaver, Damian G., Pelletier, Jeffrey C., Thanna, Sandeep, Freeman, Katie B., Reitz, Allen B., Scott, Richard W.
Published in Bioorganic & medicinal chemistry letters (01.02.2021)
Published in Bioorganic & medicinal chemistry letters (01.02.2021)
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Correction to “A Selective and Brain Penetrant p38αMAPK Inhibitor Candidate for Neurologic and Neuropsychiatric Disorders That Attenuates Neuroinflammation and Cognitive Dysfunction”
Roy, Saktimayee M, Minasov, George, Arancio, Ottavio, Chico, Laura W, Van Eldik, Linda J, Anderson, Wayne F, Pelletier, Jeffrey C, Watterson, D. Martin
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Identification of Clinically Viable Quinolinol Inhibitors of Botulinum Neurotoxin A Light Chain
Caglič, Dejan, Krutein, Michelle C, Bompiani, Kristin M, Barlow, Deborah J, Benoni, Galit, Pelletier, Jeffrey C, Reitz, Allen B, Lairson, Luke L, Houseknecht, Karen L, Smith, Garry R, Dickerson, Tobin J
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Amide- and bis-amide-linked highly potent and broadly active antifungal agents for the treatment of invasive fungal infections- towards the discovery of pre-clinical development candidate FC12406
Baugh, Simon D. P., Chaly, Anna, Weaver, Damian G., Whitman, David B., Pelletier, Jeffrey C., Bian, Haiyan, Freeman, Katie B., Reitz, Allen B., Scott, Richard W.
Published in Medicinal chemistry research (01.07.2023)
Published in Medicinal chemistry research (01.07.2023)
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Targeting Human Central Nervous System Protein Kinases: An Isoform Selective p38αMAPK Inhibitor That Attenuates Disease Progression in Alzheimer’s Disease Mouse Models
Roy, Saktimayee M, Grum-Tokars, Valerie L, Schavocky, James P, Saeed, Faisal, Staniszewski, Agnieszka, Teich, Andrew F, Arancio, Ottavio, Bachstetter, Adam D, Webster, Scott J, Van Eldik, Linda J, Minasov, George, Anderson, Wayne F, Pelletier, Jeffrey C, Watterson, D. Martin
Published in ACS chemical neuroscience (15.04.2015)
Published in ACS chemical neuroscience (15.04.2015)
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Assessing Longitudinal Treatment Efficacies and Alterations in Molecular Markers Associated with Glutamatergic Signaling and Immune Checkpoint Inhibitors in a Spontaneous Melanoma Mouse Model
Eddy, Kevinn, Gupta, Kajal, Eddin, Mohamad Naser, Marinaro, Christina, Putta, Sanjana, Sauer, John Michael, Chaly, Anna, Freeman, Katie B., Pelletier, Jeffrey C., Fateeva, Anna, Furmanski, Philip, Silk, Ann W., Reitz, Allen B., Zloza, Andrew, Chen, Suzie
Published in JID innovations (01.03.2024)
Published in JID innovations (01.03.2024)
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Dipeptide Prodrugs of the Glutamate Modulator Riluzole
Pelletier, Jeffrey C., Chen, Suzie, Bian, Haiyan, Shah, Raj, Smith, Garry R., Wrobel, Jay E., Reitz, Allen B.
Published in ACS medicinal chemistry letters (12.07.2018)
Published in ACS medicinal chemistry letters (12.07.2018)
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Intramolecular rearrangement of α-amino acid amide derivatives of 2-aminobenzothiazoles
Pelletier, Jeffrey C., Velvadapu, Venkata, McDonnell, Mark E., Wrobel, Jay E., Reitz, Allen B.
Published in Tetrahedron letters (23.07.2014)
Published in Tetrahedron letters (23.07.2014)
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Riluzole prodrugs for melanoma and ALS: Design, synthesis, and in vitro metabolic profiling
McDonnell, Mark E., Vera, Matthew D., Blass, Benjamin E., Pelletier, Jeffrey C., King, Richard C., Fernandez-Metzler, Carmen, Smith, Garry R., Wrobel, Jay, Chen, Suzie, Wall, Brian A., Reitz, Allen B.
Published in Bioorganic & medicinal chemistry (15.09.2012)
Published in Bioorganic & medicinal chemistry (15.09.2012)
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(1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-yl)methanamine: A Wingless β-Catenin Agonist That Increases Bone Formation Rate
Pelletier, Jeffrey C, Lundquist, Joseph T, Gilbert, Adam M, Alon, Nipa, Bex, Frederick J, Bhat, Bheem M, Bursavich, Mattew G, Coleburn, Valerie E, Felix, Luciana A, Green, Daniel M, Green, Paula, Hauze, Diane B, Kharode, Yogendra P, Lam, Ho-Sun, Lockhead, Susan R, Magolda, Ronald L, Matteo, Jeanne J, Mehlmann, John F, Milligan, Colleen, Murrills, Richard J, Pirrello, Jennifer, Selim, Sally, Sharp, Michael C, Unwalla, Ray J, Vera, Matthew D, Wrobel, Jay E, Yaworsky, Paul, Bodine, Peter V. N
Published in Journal of medicinal chemistry (26.11.2009)
Published in Journal of medicinal chemistry (26.11.2009)
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2-Phenyl-4-piperazinylbenzimidazoles: Orally active inhibitors of the gonadotropin releasing hormone (GnRH) receptor
Pelletier, Jeffrey C., Chengalvala, Murty, Cottom, Josh, Feingold, Irene, Garrick, Lloyd, Green, Daniel, Hauze, Diane, Huselton, Christine, Jetter, James, Kao, Wenling, Kopf, Gregory S., Lundquist, Joseph T., Mann, Charles, Mehlmann, John, Rogers, John, Shanno, Linda, Wrobel, Jay
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
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Discovery of 6-({4-[2-(4-tert-Butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): An Orally Active Antagonist of the Gonadotropin Releasing Hormone Receptor (GnRH-R)
Pelletier, Jeffrey C, Chengalvala, Murty V, Cottom, Joshua E, Feingold, Irene B, Green, Daniel M, Hauze, Diane B, Huselton, Christine A, Jetter, James W, Kopf, Gregory S, Lundquist, Joseph T, Magolda, Ronald L, Mann, Charles W, Mehlmann, John F, Rogers, John F, Shanno, Linda K, Adams, William R, Tio, Cesario O, Wrobel, Jay E
Published in Journal of medicinal chemistry (09.04.2009)
Published in Journal of medicinal chemistry (09.04.2009)
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