Greening the synthesis of peptide therapeutics: an industrial perspective
Martin, Vincent, Egelund, Peter H. G, Johansson, Henrik, Thordal Le Quement, Sebastian, Wojcik, Felix, Sejer Pedersen, Daniel
Published in RSC advances (24.11.2020)
Published in RSC advances (24.11.2020)
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Journal Article
Exploring endoperoxides as a new entry for the synthesis of branched azasugars
Domeyer, Svenja, Bjerregaard, Mark, Johansson, Henrik, Sejer Pedersen, Daniel
Published in Beilstein journal of organic chemistry (03.04.2017)
Published in Beilstein journal of organic chemistry (03.04.2017)
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Journal Article
Rational Design of Nanobody80 Loop Peptidomimetics: Towards Biased β2 Adrenergic Receptor Ligands
Martin, Charlotte, Moors, Samuel L. C., Danielsen, Mia, Betti, Cecilia, Fabris, Cecilia, Sejer Pedersen, Daniel, Pardon, Els, Peyressatre, Marion, Fehér, Krisztina, Martins, José C., Mosolff Mathiesen, Jesper, Morris, May C., Devoogdt, Nick, Caveliers, Vicky, De Proft, Frank, Steyaert, Jan, Ballet, Steven
Published in Chemistry : a European journal (18.07.2017)
Published in Chemistry : a European journal (18.07.2017)
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Journal Article
1,2,3-Triazoles in Peptidomimetic Chemistry
Pedersen, Daniel Sejer, Abell, Andrew
Published in European Journal of Organic Chemistry (01.05.2011)
Published in European Journal of Organic Chemistry (01.05.2011)
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Book Review
Journal Article
Azide- and Alkyne-Derivatised α-Amino Acids
Johansson, Henrik, Pedersen, Daniel Sejer
Published in European journal of organic chemistry (01.08.2012)
Published in European journal of organic chemistry (01.08.2012)
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Journal Article
Synthesis of the calcilytic ligand NPS 2143
Johansson, Henrik, Cailly, Thomas, Rojas Bie Thomsen, Alex, Bräuner-Osborne, Hans, Sejer Pedersen, Daniel
Published in Beilstein journal of organic chemistry (09.07.2013)
Published in Beilstein journal of organic chemistry (09.07.2013)
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Journal Article
Green Solid-Phase Peptide Synthesis: Oxyma-Triggered Spectrophotometric Monitoring of Residual Piperidine
Broman, So̷ren Lindbæk, Rosenberg, Martin, Wojcik, Felix, Holm Hansen, Anders, Egelund, Peter Hammer Guldager, Malmstro̷m, Joan, Sejer Pedersen, Daniel
Published in Organic process research & development (15.03.2024)
Published in Organic process research & development (15.03.2024)
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Journal Article
Bitopic Ligands Support the Presence of a Metastable Binding Site at the β2 Adrenergic Receptor
Gaiser, Birgit Isabel, Danielsen, Mia, Xu, Xinyu, Røpke Jørgensen, Kira, Fronik, Philipp, Märcher-Rørsted, Emil, Wróbel, Tomasz M., Liu, Xiangyu, Mosolff Mathiesen, Jesper, Sejer Pedersen, Daniel
Published in Journal of medicinal chemistry (11.07.2024)
Published in Journal of medicinal chemistry (11.07.2024)
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Journal Article
Fmoc-Removal with Pyrrolidine Expands the Available Solvent Space in Green Solid-Phase Peptide Synthesis
Egelund, Peter H. G, Jadhav, Sandip, Martin, Vincent, Johansson Castro, Henrik, Richner, Franziska, Le Quement, Sebastian Thordal, Dettner, Frank, Lechner, Carolin, Schoenleber, Ralph, Sejer Pedersen, Daniel
Published in ACS sustainable chemistry & engineering (25.10.2021)
Published in ACS sustainable chemistry & engineering (25.10.2021)
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Journal Article
Process Mass Intensity (PMI): A Holistic Analysis of Current Peptide Manufacturing Processes Informs Sustainability in Peptide Synthesis
Kekessie, Ivy, Wegner, Katarzyna, Martinez, Isamir, Kopach, Michael E., White, Timothy D., Tom, Janine K., Kenworthy, Martin N., Gallou, Fabrice, Lopez, John, Koenig, Stefan G., Payne, Philippa R., Eissler, Stefan, Arumugam, Balasubramanian, Li, Changfeng, Mukherjee, Subha, Isidro-Llobet, Albert, Ludemann-Hombourger, Olivier, Richardson, Paul, Kittelmann, Jörg, Sejer Pedersen, Daniel, van den Bos, Leendert J.
Published in Journal of organic chemistry (05.04.2024)
Published in Journal of organic chemistry (05.04.2024)
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Journal Article
Identification of a new psychoactive substance in seized material: the synthetic opioid N‐phenyl‐N‐[1‐(2‐phenethyl)piperidin‐4‐yl]prop‐2‐enamide (Acrylfentanyl)
Breindahl, Torben, Kimergård, Andreas, Andreasen, Mette Findal, Pedersen, Daniel Sejer
Published in Drug testing and analysis (01.03.2017)
Published in Drug testing and analysis (01.03.2017)
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Journal Article
Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2‑Phenylindole Privileged Structure Scaffold
Johansson, Henrik, Boesgaard, Michael Worch, Nørskov-Lauritsen, Lenea, Larsen, Inna, Kuhne, Sebastiaan, Gloriam, David E, Bräuner-Osborne, Hans, Sejer Pedersen, Daniel
Published in Journal of medicinal chemistry (25.11.2015)
Published in Journal of medicinal chemistry (25.11.2015)
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Journal Article
Amino Triazolo Diazepines (Ata) as Constrained Histidine Mimics
Buysse, Koen, Farard, Julien, Nikolaou, Alexandros, Vanderheyden, Patrick, Vauquelin, Georges, Sejer Pedersen, Daniel, Tourwé, Dirk, Ballet, Steven
Published in Organic letters (16.12.2011)
Published in Organic letters (16.12.2011)
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Journal Article
New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds
Heng, Sabrina, Tieu, William, Hautmann, Stephanie, Kuan, Kevin, Pedersen, Daniel Sejer, Pietsch, Markus, Gütschow, Michael, Abell, Andrew D.
Published in Bioorganic & medicinal chemistry (15.12.2011)
Published in Bioorganic & medicinal chemistry (15.12.2011)
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Journal Article