R428, a Selective Small Molecule Inhibitor of Axl Kinase, Blocks Tumor Spread and Prolongs Survival in Models of Metastatic Breast Cancer
HOLLAND, Sacha J, PAN, Alison, JING ZHANG, PINGYU DING, APATIRA, Ayodele, CHUA, Joanne, BRANDT, Ralf, PINE, Polly, GOFF, Dane, SINGH, Rajinder, PAYAN, Donald G, HITOSHI, Yasumichi, FRANCI, Christian, YUANMING HU, CHANG, Betty, WEIQUN LI, DUAN, Matt, TORNEROS, Allan, JIAXIN YU, HECKRODT, Thilo J
Published in Cancer research (Chicago, Ill.) (15.02.2010)
Published in Cancer research (Chicago, Ill.) (15.02.2010)
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Discovery and Development of Spleen Tyrosine Kinase (SYK) Inhibitors
Singh, Rajinder, Masuda, Esteban S, Payan, Donald G
Published in Journal of medicinal chemistry (26.04.2012)
Published in Journal of medicinal chemistry (26.04.2012)
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R406, an Orally Available Spleen Tyrosine Kinase Inhibitor Blocks Fc Receptor Signaling and Reduces Immune Complex-Mediated Inflammation
Braselmann, Sylvia, Taylor, Vanessa, Zhao, Haoran, Wang, Su, Sylvain, Catherine, Baluom, Muhammad, Qu, Kunbin, Herlaar, Ellen, Lau, Angela, Young, Chi, Wong, Brian R, Lovell, Scott, Sun, Thomas, Park, Gary, Argade, Ankush, Jurcevic, Stipo, Pine, Polly, Singh, Rajinder, Grossbard, Elliott B, Payan, Donald G, Masuda, Esteban S
Published in The Journal of pharmacology and experimental therapeutics (01.12.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2006)
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Developing structure–activity relationships from an HTS hit for inhibition of the Cks1–Skp2 protein–protein interaction
Singh, Rajinder, Sran, Arvinder, Carroll, David C., Huang, Jianing, Tsvetkov, Lyuben, Zhou, Xiulan, Sheung, Julie, McLaughlin, John, Issakani, Sarkiz D., Payan, Donald G., Shaw, Simon J.
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
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AMPK activation through mitochondrial regulation results in increased substrate oxidation and improved metabolic parameters in models of diabetes
Jenkins, Yonchu, Sun, Tian-Qiang, Markovtsov, Vadim, Foretz, Marc, Li, Wei, Nguyen, Henry, Li, Yingwu, Pan, Alison, Uy, Gerald, Gross, Lisa, Baltgalvis, Kristen, Yung, Stephanie L, Gururaja, Tarikere, Kinoshita, Taisei, Owyang, Alexander, Smith, Ira J, McCaughey, Kelly, White, Kathy, Godinez, Guillermo, Alcantara, Raniel, Choy, Carmen, Ren, Hong, Basile, Rachel, Sweeny, David J, Xu, Xiang, Issakani, Sarkiz D, Carroll, David C, Goff, Dane A, Shaw, Simon J, Singh, Rajinder, Boros, Laszlo G, Laplante, Marc-André, Marcotte, Bruno, Kohen, Rita, Viollet, Benoit, Marette, André, Payan, Donald G, Kinsella, Todd M, Hitoshi, Yasumichi
Published in PloS one (05.12.2013)
Published in PloS one (05.12.2013)
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JAK3 Inhibition Significantly Attenuates Psoriasiform Skin Inflammation in CD18 Mutant PL/J Mice
Chang, Betty Y, Zhao, Feifei, He, Xiaodong, Ren, Hong, Braselmann, Sylvia, Taylor, Vanessa, Wicks, Joan, Payan, Donald G, Grossbard, Elliott B, Pine, Polly R, Bullard, Daniel C
Published in The Journal of immunology (1950) (01.08.2009)
Published in The Journal of immunology (1950) (01.08.2009)
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Critical role of the ubiquitin ligase activity of UHRF1, a nuclear RING finger protein, in tumor cell growth
Jenkins, Yonchu, Markovtsov, Vadim, Lang, Wayne, Sharma, Poonam, Pearsall, Denise, Warner, Justin, Franci, Christian, Huang, Betty, Huang, Jianing, Yam, George C, Vistan, Joseph P, Pali, Erlina, Vialard, Jorge, Janicot, Michel, Lorens, James B, Payan, Donald G, Hitoshi, Yasumichi
Published in Molecular biology of the cell (01.12.2005)
Published in Molecular biology of the cell (01.12.2005)
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Multiple roles for the receptor tyrosine kinase axl in tumor formation
HOLLAND, Sacha J, POWELL, Mark J, WONG, Stephen, LASAGA, Joe, SHEN, Mary R, SIMON YU, WEIDUAN XU, HITOSHI, Yasumichi, BOGENBERGER, Jakob, NÖR, Jacques E, PAYAN, Donald G, LORENS, James B, FRANCI, Christian, CHAN, Emily W, FRIERA, Annabelle M, ATCHISON, Robert E, MCLAUGHLIN, John, SWIFT, Susan E, PALI, Erlina S, YAM, George
Published in Cancer research (Chicago, Ill.) (15.10.2005)
Published in Cancer research (Chicago, Ill.) (15.10.2005)
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Substrate Modification with Lysine 63-linked Ubiquitin Chains through the UBC13-UEV1A Ubiquitin-conjugating Enzyme
Petroski, Matthew D., Zhou, Xiulan, Dong, GuoQiang, Daniel-Issakani, Sarkiz, Payan, Donald G., Huang, Jianing
Published in The Journal of biological chemistry (12.10.2007)
Published in The Journal of biological chemistry (12.10.2007)
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Journal Article
R723, a selective JAK2 inhibitor, effectively treats JAK2V617F-induced murine myeloproliferative neoplasm
Shide, Kotaro, Kameda, Takuro, Markovtsov, Vadim, Shimoda, Haruko K., Tonkin, Elizabeth, Fang, Shuling, Liu, Chian, Gelman, Marina, Lang, Wayne, Romero, Jason, McLaughlin, John, Bhamidipati, Somasekhar, Clough, Jeffrey, Low, Caroline, Reitsma, Andrea, Siu, Stacey, Pine, Polly, Park, Gary, Torneros, Allan, Duan, Matt, Singh, Rajinder, Payan, Donald G., Matsunaga, Takuya, Hitoshi, Yasumichi, Shimoda, Kazuya
Published in Blood (23.06.2011)
Published in Blood (23.06.2011)
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Noninvasive imaging of in vivo MuRF1 expression during muscle atrophy
Li, Wei, Claypool, Mark D, Friera, Annabelle M, McLaughlin, John, Baltgalvis, Kristen A, Smith, Ira J, Kinoshita, Taisei, White, Kathy, Lang, Wayne, Godinez, Guillermo, Payan, Donald G, Kinsella, Todd M
Published in PloS one (01.04.2014)
Published in PloS one (01.04.2014)
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Journal Article
Activation of the PKB/AKT Pathway by ICAM-2
Perez, Omar D, Kinoshita, Shigemi, Hitoshi, Yasumichi, Payan, Donald G, Kitamura, Toshio, Nolan, Garry P, Lorens, James B
Published in Immunity (Cambridge, Mass.) (2002)
Published in Immunity (Cambridge, Mass.) (2002)
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Journal Article
Optimization of Pharmacokinetic and In Vitro Safety Profile of a Series of Pyridine Diamide Indirect AMPK Activators
Shaw, Simon J., Goff, Dane A., Boralsky, Luke A., Singh, Rajinder, Sweeny, David J., Park, Gary, Sun, Tian-Qiang, Jenkins, Yonchu, Markovtsov, Vadim, Issakani, Sarkiz D., Payan, Donald G., Hitoshi, Yasumichi
Published in Journal of medicinal chemistry (28.12.2023)
Published in Journal of medicinal chemistry (28.12.2023)
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Journal Article
The Poxvirus p28 Virulence Factor Is an E3 Ubiquitin Ligase
Huang, Jianing, Huang, Qi, Zhou, Xiulan, Shen, Mary M., Yen, Ann, Yu, Simon X., Dong, GuoQiang, Qu, Kunbin, Huang, Peiyong, Anderson, Emily M., Daniel-Issakani, Sarkiz, Buller, R. Mark L., Payan, Donald G., Lu, H. Henry
Published in The Journal of biological chemistry (24.12.2004)
Published in The Journal of biological chemistry (24.12.2004)
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Journal Article
Bicyclic pyrimidine compounds as potent IRAK4 inhibitors
Chen, Yan, Tso, Kin, Heckrodt, Thilo J., Li, Hui, Yen, Rose, Lin, Nan, Singh, Rajinder, Taylor, Vanessa, Masuda, Esteban S., Park, Gary, Payan, Donald G.
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
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Discovery of 5‑Aryl-2,4-diaminopyrimidine Compounds as Potent and Selective IRAK4 Inhibitors
Chen, Yan, Singh, Rajinder, Lin, Nan, Taylor, Vanessa, Masuda, Esteban S, Payan, Donald G
Published in ACS medicinal chemistry letters (14.04.2022)
Published in ACS medicinal chemistry letters (14.04.2022)
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Retrovirally Delivered Random Cyclic Peptide Libraries Yield Inhibitors of Interleukin-4 Signaling in Human B Cells
Kinsella, Todd M., Ohashi, Cara T., Harder, Amy Grace, Yam, George C., Li, Weiqun, Peelle, Beau, Pali, Erlina S., Bennett, Mark K., Molineaux, Susan M., Anderson, D.A., Masuda, Esteban S., Payan, Donald G.
Published in The Journal of biological chemistry (04.10.2002)
Published in The Journal of biological chemistry (04.10.2002)
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Structure activity relationships leading to the identification of the indirect activator of AMPK, R419
Shaw, Simon J., Goff, Dane A., Carroll, David C., Singh, Rajinder, Sweeny, David J., Park, Gary, Jenkins, Yonchu, Markovtsov, Vadim, Sun, Tian-Qiang, Issakani, Sarkiz D., Hitoshi, Yasumichi, Payan, Donald G.
Published in Bioorganic & medicinal chemistry (01.10.2022)
Published in Bioorganic & medicinal chemistry (01.10.2022)
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Journal Article
R-253 Disrupts Microtubule Networks in Multiple Tumor Cell Lines
GURURAJA, Tarikere L, GOFF, Dane, HITOSHI, Yasumichi, COOPER, R. D. G, PAYAN, Donald G, KINOSHITA, Taisei, GOLDSTEIN, Eileen, YUNG, Stephanie, MCLAUGHLIN, John, PALI, Erlina, JIANING HUANG, SINGH, Rajinder, DANIEL-ISSAKANI, Sarkiz
Published in Clinical cancer research (15.06.2006)
Published in Clinical cancer research (15.06.2006)
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