Synthesis, Structure−Activity Relationships, and Characterization of Novel Nonsteroidal and Selective Androgen Receptor Modulators
Schlienger, Nathalie, Lund, Birgitte W, Pawlas, Jan, Badalassi, Fabrizio, Bertozzi, Fabio, Lewinsky, Rasmus, Fejzic, Alma, Thygesen, Mikkel B, Tabatabaei, Ali, Bradley, Stefania Risso, Gardell, Luis R, Piu, Fabrice, Olsson, Roger
Published in Journal of medicinal chemistry (26.11.2009)
Published in Journal of medicinal chemistry (26.11.2009)
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Journal Article
Brønsted Acid–Lewis Acid (BA–LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/ t- Bu Solid-Phase Peptide Synthesis: HCl/FeCl 3 and AcOH/FeCl 3 as Viable PFAS-Free Alternatives for TFA
Pawlas, Jan, André, Christophe, Rasmussen, Jon H., Ludemann-Hombourger, Olivier
Published in Organic letters (09.08.2024)
Published in Organic letters (09.08.2024)
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Journal Article
2D green SPPS: green solvents for on-resin removal of acid sensitive protecting groups and lactamization
Pawlas, Jan, Antonic, Biljana, Lundqvist, Marika, Svensson, Thomas, Finnman, Jens, Rasmussen, Jon H
Published in Green chemistry : an international journal and green chemistry resource : GC (20.05.2019)
Published in Green chemistry : an international journal and green chemistry resource : GC (20.05.2019)
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Journal Article
Brønsted Acid–Lewis Acid (BA–LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/t-Bu Solid-Phase Peptide Synthesis: HCl/FeCl3 and AcOH/FeCl3 as Viable PFAS-Free Alternatives for TFA
Pawlas, Jan, André, Christophe, Rasmussen, Jon H., Ludemann-Hombourger, Olivier
Published in Organic letters (09.08.2024)
Published in Organic letters (09.08.2024)
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Journal Article
Sustainable, cost-efficient manufacturing of therapeutic peptides using chemo-enzymatic peptide synthesis (CEPS)
Pawlas, Jan, Nuijens, Timo, Persson, Jonas, Svensson, Thomas, Schmidt, Marcel, Toplak, Ana, Nilsson, Mikael, Rasmussen, Jon H
Published in Green chemistry : an international journal and green chemistry resource : GC (2019)
Published in Green chemistry : an international journal and green chemistry resource : GC (2019)
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Journal Article
Novel Anionic Annelation Tactics for Construction of Fused Heteroaromatic Frameworks. 1. Synthesis of 4-Substituted Pyrazolo[4,3-c]quinolines, 9-Substituted Pyrazolo[3,4-c]quinolines, and 1,4-Dihydrochromeno[4,3-c]pyrazoles
Pawlas, Jan, Vedsø, Per, Jakobsen, Palle, Huusfeldt, Per Olaf, Begtrup, Mikael
Published in Journal of organic chemistry (15.06.2001)
Published in Journal of organic chemistry (15.06.2001)
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Journal Article
Elevating 1-tert-Butyl-3-ethylcarbodiimide (TBEC) as a Reagent for Sustainable Peptide Synthesis: Quality Assessment and Minimizing Racemization, Precipitation, and Radical-Induced Side Reactions by TBEC/Oxyma Couplings in an Environmentally Sensible Solvent
Pawlas, Jan, Choi, Ji-Hyung, von Bargen, Christoph, Maibom-Thomsen, Sheila, Rasmussen, Jon H., Ludemann-Hombourger, Olivier
Published in Organic process research & development (21.07.2023)
Published in Organic process research & development (21.07.2023)
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Journal Article
Advancing Sustainable Peptide Synthesis by Solvent Quality Control: Understanding and Mitigating Hydroperoxide in 1-Butyl-2-pyrrolidinone (NBP)
Pawlas, Jan, El-Dine, Tharwat Mohy, Bargen, Katharina von, Bargen, Christoph von, Nilsson, Johan, Ludemann-Hombourger, Olivier, Rasmussen, Jon H.
Published in Organic process research & development (16.08.2024)
Published in Organic process research & development (16.08.2024)
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Journal Article
Green Chemistry Articles of Interest to the Pharmaceutical Industry
Ashley, Melissa A., Aukland, Miles H., Bryan, Marian C., Cismesia, Megan A., Dutschei, Theresa, Engl, Oliver D., Engl, Pascal S., Enriquez Garcia, Álvaro, Harawa, Vanessa, Karageorgis, George, Kelly, Christopher B., Leclair, Alexandre, Lee, Johnny W., Lei, Zhen, Li, Wei, Pawlas, Jan, Richardson, Paul F., Scott, Samuel C., Steven, Alan, Takale, Balaram S., Yerkozhanov, Dauzhan, Zeng, Mingshuo
Published in Organic process research & development (10.09.2024)
Published in Organic process research & development (10.09.2024)
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