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Leucine-rich Repeat Kinase 2 (LRRK2) Pharmacological Inhibition Abates α-Synuclein Gene-induced Neurodegeneration
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Enantioselective Construction of Cyclic Ethers by An Aldol-Cyclization Sequence
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Published in Journal of organic chemistry (25.07.1997)
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Kinase domain inhibition of leucine rich repeat kinase 2 (LRRK2) using a [1,2,4]triazolo[4,3-b]pyridazine scaffold
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Published in Bioorganic & medicinal chemistry letters (01.09.2014)
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Ligand–Protein Interactions of Selective Casein Kinase 1δ Inhibitors
Mente, Scot, Arnold, Eric, Butler, Todd, Chakrapani, Subramanyam, Chandrasekaran, Ramalakshmi, Cherry, Kevin, DiRico, Ken, Doran, Angela, Fisher, Katherine, Galatsis, Paul, Green, Michael, Hayward, Matthew, Humphrey, John, Knafels, John, Li, Jianke, Liu, Shenping, Marconi, Michael, McDonald, Scott, Ohren, Jeff, Paradis, Vanessa, Sneed, Blossom, Walton, Kevin, Wager, Travis
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Discovery of selective 2,4-diaminopyrimidine-based photoaffinity probes for glyoxalase IElectronic supplementary information (ESI) available: Detailed synthetic procedures, 1H and 13C NMR spectra, HPLC chromatograms for compounds L1, L2, L3, L1-Biotin and L1-Bpyne; detailed procedures for biological assays; mass spectroscopy data for GLO-1. See DOI: 10.1039/c3md00286a
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Year of Publication 26.02.2014
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NOVEL 3,4-DISUBSTITUTED-1H-PYRROLO[2,3-b]PYRIDINE AND 4,5-DISUBSTITUTED-7H-PYRROLO[2,3-C]PYRIDAZINE AS LRRK2 INHIBITOR
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Year of Publication 11.07.2019
Patent
NOVEL 4-(SUBSTITUTED AMINO)-7H-PYRROLO[2,3-D]PYRIMIDINES AS LRRK2 INHIBITORS
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Year of Publication 16.05.2019
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Year of Publication 16.05.2019
Patent