Development of Prodrug 4-Chloro-3-(5-methyl-3-{[4-(2-pyrrolidin-1-ylethoxy)phenyl]amino}-1,2,4-benzotriazin-7-yl)phenyl Benzoate (TG100801): A Topically Administered Therapeutic Candidate in Clinical Trials for the Treatment of Age-Related Macular Degeneration
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Published in Journal of medicinal chemistry (27.03.2008)
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Round Cell Vaginal Malignant Melanoma: A rare entity
Chauhan, Neena, Gaur, Dushyant S, Pathak, Ved P
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Discovery and preliminary structure–activity relationship studies of novel benzotriazine based compounds as Src inhibitors
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Biological Characterization of a Novel, Orally Active Small Molecule Gonadotropin-Releasing Hormone (GnRH) Antagonist Using Castrated and Intact Rats
Anderes, Kenna L, Luthin, David R, Castillo, Rosemary, Kraynov, Eugenia A, Castro, Mary, Nared-Hood, Karen, Gregory, Margaret L, Pathak, Ved P, Christie, Lance C, Paderes, Genevieve, Vazir, Haresh, Ye, Qiang, Anderson, Mark B, May, John M
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Design and Synthesis of Benzoic Acid Derivatives as Influenza Neuraminidase Inhibitors Using Structure-Based Drug Design
Chand, Pooran, Babu, Yarlagadda S, Bantia, Shanta, Chu, Naiming, Cole, L. Brent, Kotian, Pravin L, Laver, W. Graeme, Montgomery, John A, Pathak, Ved P, Petty, Sandra L, Shrout, David P, Walsh, David A, Walsh, Gerald M
Published in Journal of medicinal chemistry (05.12.1997)
Published in Journal of medicinal chemistry (05.12.1997)
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Inhibitors of ABL and the ABL-T315I mutation
Noronha, Glenn, Cao, Jianguo, Chow, Chun P, Dneprovskaia, Elena, Fine, Richard M, Hood, John, Kang, Xinshan, Klebansky, Boris, Lohse, Dan, Mak, Chi Ching, McPherson, Andre, Palanki, Moorthy S S, Pathak, Ved P, Renick, Joel, Soll, Richard, Zeng, Binqi
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Published in Current topics in medicinal chemistry (01.07.2008)
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Discovery of [7-(2,6-dichlorophenyl)-5-methylbenzo [1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]amine—a potent, orally active Src kinase inhibitor with anti-tumor activity in preclinical assays
Noronha, Glenn, Barrett, Kathy, Boccia, Antonio, Brodhag, Tessa, Cao, Jianguo, Chow, Chun P., Dneprovskaia, Elena, Doukas, John, Fine, Richard, Gong, Xianchang, Gritzen, Colleen, Gu, Hong, Hanna, Ehab, Hood, John D., Hu, Steven, Kang, Xinshan, Key, Jann, Klebansky, Boris, Kousba, Ahmed, Li, Ge, Lohse, Dan, Mak, Chi Ching, McPherson, Andrew, Palanki, Moorthy S.S., Pathak, Ved P., Renick, Joel, Shi, Feng, Soll, Richard, Splittgerber, Ute, Stoughton, Silva, Tang, Suhan, Yee, Shiyin, Zeng, Binqi, Zhao, Ningning, Zhu, Hong
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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The design and preliminary structure–activity relationship studies of benzotriazines as potent inhibitors of Abl and Abl-T315I enzymes
Cao, Jianguo, Fine, Richard, Gritzen, Colleen, Hood, John, Kang, Xinshan, Klebansky, Boris, Lohse, Dan, Mak, Chi Ching, McPherson, Andrew, Noronha, Glenn, Palanki, Moorthy S.S., Pathak, Ved P., Renick, Joel, Soll, Richard, Zeng, Binqi, Zhu, Hong
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Electrophilic Tetraalkylammonium Nitrate Nitration. II. Improved Anhydrous Aromatic and Heteroaromatic Mononitration with Tetramethylammonium Nitrate and Triflic Anhydride, Including Selected Microwave Examples
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Structure-Based Design of Inhibitors of Purine Nucleoside Phosphorylase. 5. 9-Deazahypoxanthines
Niwas, Shri, Chand, Pooran, Pathak, Ved P, Montgomery, John A
Published in Journal of medicinal chemistry (01.07.1994)
Published in Journal of medicinal chemistry (01.07.1994)
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Discovery of a Novel, Orally Active, Small Molecule Gonadotropin-Releasing Hormone (GnRH) Receptor Antagonist
Li, Haitao, Anderes, Kenna L, Kraynov, Eugenia A, Luthin, David R, Do, Quyen-Quyen, Hong, Yufeng, Tompkins, Eileen, Sun, Eric T, Rajapakse, Ranjan, Pathak, Ved P, Christie, Lance C, Vazir, Haresh, Castillo, Rosemary, Gregory, Margaret L, Castro, Mary, Nared-Hood, Karen, Paderes, Genevieve, Anderson, Mark B
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Development of novel benzotriazines for drug discovery
Palanki, Moorthy Ss, Cao, Jianguo, Chow, Chun P, Dneprovskaia, Elena, Mak, Chi Ching, McPherson, Andrew, Pathak, Ved P, Renick, Joel, Soll, Richard, Zeng, Binqi, Noronha, Glenn
Published in Expert opinion on drug discovery (01.01.2009)
Published in Expert opinion on drug discovery (01.01.2009)
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Journal Article
Discovery of a Novel, Orally Active, Small Molecule Gonadotropin-Releasing Hormone (GnRH) Receptor Antagonist
Li, Haitao, Anderes, Kenna L, Kraynov, Eugenia A, Luthin, David R, Do, Quyen-Quyen, Hong, Yufeng, Tompkins, Eileen, Sun, Eric T, Rajapakse, Ranjan, Pathak, Ved P, Christie, Lance C, Feng, Jun, Vazir, Haresh, Castillo, Rosemary, Gregory, Margaret L, Castro, Mary, Nared-Hood, Karen, Paderes, Genevieve, Anderson, Mark B
Published in Journal of medicinal chemistry (21.09.2006)
Published in Journal of medicinal chemistry (21.09.2006)
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The discovery of novel small molecule non-peptide gonadotropin releasing hormone (GnRH) receptor antagonists
Luthin, David R., Hong, Yufeng, Pathak, Ved P., Paderes, Genevieve, Nared-Hood, Karen D., Castro, Mary A., Vazir, Haresh, Li, Haitao, Tompkins, Eileen, Christie, Lance, May, John M., Anderson, Mark B.
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
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Electrophilic Tetraalkylammonium Nitrate Nitration. II. Improved Anhydrous Aromatic and Heteroaromatic Mononitration with Tetramethylammonium Nitrate and Triflic Anhydride, Including Selected Microwave Examples
Shackelford, Scott A, Anderson, Mark B, Christie, Lance C, Goetzen, Thomas, Guzman, Mark C, Hananel, Martha A, Kornreich, Wayne D, Li, Haitao, Pathak, Ved P, Rabinovich, Alex K, Rajapakse, Ranjan J, Truesdale, Larry K, Tsank, Stella M, Vazir, Haresh N
Published in Journal of organic chemistry (04.04.2003)
Published in Journal of organic chemistry (04.04.2003)
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In Vitro and In Vivo Inhibition of the T315I Mutant BCR/ABL Kinase
Zhu, Hong, Hanna, Ehab, Lohse, Dan, Stoughton, Silva, Tam, Betty, Barrett, Kathy, Noronha, Glenn, Dneprovskaia, Elena, Cao, Jon, Chow, Chun, Hwang, Linda, Mak, Chiching, McPherson, Andy, Palanki, Moorthy, Pathak, Ved P., Renick, Joe, Soll, Richard, Zeng, Binqi, Hood, John
Published in Blood (16.11.2006)
Published in Blood (16.11.2006)
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