Anti-TNF Thioester Glucocorticoid Antibody–Drug Conjugate Fully Inhibits Inflammation with Minimal Effect on Systemic Corticosterone Levels in a Mouse Arthritis Model
Marvin, Christopher C., Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Patel, Meena V., Schmidt, Diana L., Li, Tongmei, Randolph, John T., Bischoff, Agnieszka K., Fitzgibbons, Julia, Wang, Lu, Wang, Lu, Hernandez, Axel, Jia, Ying, Goess, Christian A., Bryant, Shaughn H., Mathieu, Suzanne L., Xu, Jianwen
Published in Journal of medicinal chemistry (23.05.2024)
Published in Journal of medicinal chemistry (23.05.2024)
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Journal Article
Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate
Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, Patel, Meena V., Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa
Published in Journal of medicinal chemistry (08.12.2022)
Published in Journal of medicinal chemistry (08.12.2022)
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Journal Article
Correction to “Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate”
Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, Patel, Meena V., Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa
Published in Journal of medicinal chemistry (27.04.2023)
Published in Journal of medicinal chemistry (27.04.2023)
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Journal Article
Synthesis of 4,5-Diaryl-1H-pyrazole-3-ol Derivatives as Potential COX-2 Inhibitors
Patel, Meena V, Bell, Randy, Majest, Sandra, Henry, Rodger, Kolasa, Teodozyj
Published in Journal of organic chemistry (15.10.2004)
Published in Journal of organic chemistry (15.10.2004)
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Journal Article
Synthesis and Structure−Activity Studies on N-[5-(1H-Imidazol-4-yl)-5,6,7,8-tetrahydro-1-naphthalenyl]methanesulfonamide, an Imidazole-Containing α1A-Adrenoceptor Agonist
Altenbach, Robert J, Khilevich, Albert, Kolasa, Teodozyj, Rohde, Jeffrey J, Bhatia, Pramila A, Patel, Meena V, Searle, Xenia B, Yang, Fan, Bunnelle, William H, Tietje, Karin, Bayburt, Erol K, Carroll, William A, Meyer, Michael D, Henry, Rodger, Buckner, Steven A, Kuk, Jane, Daza, Anthony V, Milicic, Ivan V, Cain, John C, Kang, Chae H, Ireland, Lynne M, Carr, Tracy L, Miller, Thomas R, Hancock, Arthur A, Nakane, Masaki, Esbenshade, Timothy A, Brune, Michael E, O'Neill, Alyssa B, Gauvin, Donna M, Katwala, Sweta P, Holladay, Mark W, Brioni, Jorge D, Sullivan, James P
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Journal Article
Discovery of 3-Methyl-N-(1-oxy-3‘,4‘,5‘,6‘-tetrahydro-2‘H-[2,4‘-bipyridine]-1‘-ylmethyl)benzamide (ABT-670), an Orally Bioavailable Dopamine D4 Agonist for the Treatment of Erectile Dysfunction
Patel, Meena V, Kolasa, Teodozyj, Mortell, Kathleen, Matulenko, Mark A, Hakeem, Ahmed A, Rohde, Jeffrey J, Nelson, Sherry L, Cowart, Marlon D, Nakane, Masaki, Miller, Loan N, Uchic, Marie E, Terranova, Marc A, El-Kouhen, Odile F, Donnelly-Roberts, Diana L, Namovic, Marian T, Hollingsworth, Peter R, Chang, Renjie, Martino, Brenda R, Wetter, Jill M, Marsh, Kennan C, Martin, Ruth, Darbyshire, John F, Gintant, Gary, Hsieh, Gin C, Moreland, Robert B, Sullivan, James P, Brioni, Jorge D, Stewart, Andrew O
Published in Journal of medicinal chemistry (14.12.2006)
Published in Journal of medicinal chemistry (14.12.2006)
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Journal Article
An efficient one-pot synthesis of substituted 2-arylbenzo[ b]thiophene derivatives
Patel, Meena V, Rohde, Jeffrey J, Gracias, Vijaya, Kolasa, Teodozyj
Published in Tetrahedron letters (25.08.2003)
Published in Tetrahedron letters (25.08.2003)
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Journal Article
1-Aryl-3-(4-pyridine-2-ylpiperazin-1-yl)propan-1-one Oximes as Potent Dopamine D4 Receptor Agonists for the Treatment of Erectile Dysfunction
Kolasa, Teodozyj, Matulenko, Mark A, Hakeem, Ahmed A, Patel, Meena V, Mortell, Kathleen, Bhatia, Pramila, Henry, Rodger, Nakane, Masaki, Hsieh, Gin C, Terranova, Marc A, Uchic, Marie E, Miller, Loan N, Chang, Renje, Donnelly-Roberts, Diana L, Namovic, Marian T, Hollingsworth, Peter R, Martino, Brenda, El Kouhen, Odile, Marsh, Kennan C, Wetter, Jill M, Moreland, Robert B, Brioni, Jorge D, Stewart, Andrew O
Published in Journal of medicinal chemistry (24.08.2006)
Published in Journal of medicinal chemistry (24.08.2006)
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Journal Article
Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator
Hobson, Adrian D., McPherson, Michael J., Hayes, Martin E., Goess, Christian, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Yang, Jindong, Sun, Liang, Zhang, Qiang, Qu, Pei, Yang, Shi, Hernandez, Axel, Bryant, Shaughn H., Mathieu, Suzanne L., Bischoff, Agnieszka K., Fitzgibbons, Julia, Santora, Ling C., Wang, Lu, Fettis, Margaret M., Li, Xiaofeng, Marvin, Christopher C., Wang, Zhi, V. Patel, Meena, Schmidt, Diana L., Li, Tongmei, Randolph, John T., Henry, Rodger F., Graff, Candace, Tian, Yu, Aguirre, Ana L., Shrestha, Anurupa
Published in Journal of medicinal chemistry (08.12.2022)
Published in Journal of medicinal chemistry (08.12.2022)
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Journal Article
6-- 6---2- 6-HETEROARYLOXY- AND 6-ARYLOXY-QUINOLINE-2-CARBOXAMIDES AND USES THEREOF
PATEL MEENA V, PELTIER HILLARY, KOENIG JOHN R, WAKEFIELD BRIAN D, JINKERSON TAMMIE K, KORT MICHAEL E, DEGOEY DAVID A, LIU BO, MATULENKO MARK A, COWART MARLON D, SCANIO MARC J, NELSON DEREK W, BOGDAN ANDREW
Year of Publication 11.10.2016
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Year of Publication 11.10.2016
Patent
Synthesis of N,N‘-Orthogonally Protected (S)-Piperazine-2-carboxylic Acid
Warshawsky, Alan M, Patel, Meena V, Chen, Teng-Man
Published in Journal of organic chemistry (05.09.1997)
Published in Journal of organic chemistry (05.09.1997)
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Journal Article
Discovery of (R)-(3-fluoropyrrolidin-1-yl)(6-((5-(trifluoromethyl)pyridin-2-yl)oxy)quinolin-2-yl)methanone (ABBV-318) and analogs as small molecule Na v 1.7/ Nav1.8 blockers for the treatment of pain
Patel, Meena V, Peltier, Hillary M, Matulenko, Mark A, Koenig, John R, C Scanio, Marc J, Gum, Rebecca J, El-Kouhen, Odile F, Fricano, Meagan M, Lundgaard, Greta L, Neelands, Torben, Zhang, Xu-Feng, Zhan, Cenchen, Pai, Madhavi, Ghoreishi-Haack, Nayereh, Hudzik, Thomas, Gintant, Gary, Martin, Ruth, McGaraughty, Steve, Xu, Jun, Bow, Daniel, Kalvass, John C, Kym, Philip R, DeGoey, David A, Kort, Michael E
Published in Bioorganic & medicinal chemistry (01.06.2022)
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Published in Bioorganic & medicinal chemistry (01.06.2022)
Journal Article
Discovery of 3-methyl-N-(1-oxy-3 ',4 ',5 ',6 '-tetrahydro-2 ' H-[2,4 '-bipyridine]-1 '-ylmethyl)benzamide (ABT-670), an orally bioavailable dopamine D-4 agonist for the treatment of erectile dysfunction
Patel, Meena V., Kolasa, Teodozyj, Mortell, Kathleen, Matulenko, Mark A., Hakeem, Ahmed A., Rohde, Jeffrey J., Nelson, Sherry L., Cowart, Marlon D., Nakane, Masaki, Miller, Loan N., Uchic, Marie E., Terranova, Marc A., El-Kouhen, Odile F., Donnelly-Roberts, Diana L., Namovic, Marian T., Hollingsworth, Peter R., Chang, Renjie, Martino, Brenda R., Wetter, Jill M., Marsh, Kennan C., Martin, Ruth, Darbyshire, John F., Gintant, Gary, Hsieh, Gin C., Moreland, Robert B., Sullivan, James P., Brioni, Jorge D., Stewart, Andrew O.
Published in Journal of medicinal chemistry (14.12.2006)
Published in Journal of medicinal chemistry (14.12.2006)
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Journal Article
1-Aryl-3-(4-pyridine-2-ylpiperazin-1-yl)propan-1-one oximes as potent dopamine D-4 receptor agonists for the treatment of erectile dysfunction
Kolasa, Teodozyj, Matulenko, Mark A., Hakeem, Ahmed A., Patel, Meena V., Mortell, Kathleen, Bhatia, Pramila, Henry, Rodger, Nakane, Masaki, Hsieh, Gin C., Terranova, Marc A., Uchic, Marie E., Miller, Loan N., Chang, Renje, Donnelly-Roberts, Diana L., Namovic, Marian T., Hollingsworth, Peter R., Martino, Brenda, El Kouhen, Odile, Marsh, Kennan C., Wetter, Jill M., Moreland, Robert B., Brioni, Jorge D., Stewart, Andrew O.
Published in Journal of medicinal chemistry (24.08.2006)
Published in Journal of medicinal chemistry (24.08.2006)
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Journal Article
Synthesis of 4,5-Diaryl-1 H -pyrazole-3-ol Derivatives as Potential COX-2 Inhibitors
Patel, Meena V., Bell, Randy, Majest, Sandra, Henry, Rodger, Kolasa, Teodozyj
Published in Journal of organic chemistry (01.10.2004)
Published in Journal of organic chemistry (01.10.2004)
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Journal Article
Discovery of Inhibitors of Cell Adhesion Molecule Expression in Human Endothelial Cells. 1. Selective Inhibition of ICAM-1 and E-Selectin Expression
Stewart, Andrew O, Bhatia, Pramila A, McCarty, Catherine M, Patel, Meena V, Staeger, Michael A, Arendsen, David L, Gunawardana, Indrani W, Melcher, Laura M, Zhu, Gui-Dong, Boyd, Steven A, Fry, Dennis G, Cool, Barbara L, Kifle, Lemma, Lartey, Kraig, Marsh, Kennan C, Kempf-Grote, Anita J, Kilgannon, Patrick, Wisdom, Wendy, Meyer, Joey, Gallatin, W. Michael, Okasinski, Gregory F
Published in Journal of medicinal chemistry (15.03.2001)
Published in Journal of medicinal chemistry (15.03.2001)
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Journal Article
Synthesis and structure-activity studies on N-[5-(1H-imidazol-4-yl)-5,6,7,8-tetrahydro-1-naphthalenyl]methanesulfonamide, an imidazole-containing alpha(1A)-adrenoceptor agonist
Altenbach, RJ, Khilevich, A, Kolasa, T, Rohde, JJ, Bhatia, PA, Patel, MV, Searle, XB, Yang, F, Bunnelle, WH, Tietje, K, Bayburt, EK, Carroll, WA, Meyer, MD, Henry, R, Buckner, SA, Kuk, J, Daza, AV, Milicic, Cain, JC, Kang, CH, Ireland, LM, Carr, TL, Miller, TR, Hancock, AA, Nakane, M, Esbenshade, TA, Brune, ME, O'Neill, AB, Gauvin, DM, Katwala, SP, Holladay, MW, Brioni, JD, Sullivan, JP
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Journal Article
Synthesis and Structure−Activity Studies on N -[5-(1 H -Imidazol-4-yl)-5,6,7,8-tetrahydro-1-naphthalenyl]methanesulfonamide, an Imidazole-Containing α 1A -Adrenoceptor Agonist
Altenbach, Robert J., Khilevich, Albert, Kolasa, Teodozyj, Rohde, Jeffrey J., Bhatia, Pramila A., Patel, Meena V., Searle, Xenia B., Yang, Fan, Bunnelle, William H., Tietje, Karin, Bayburt, Erol K., Carroll, William A., Meyer, Michael D., Henry, Rodger, Buckner, Steven A., Kuk, Jane, Daza, Anthony V., Milicic, Ivan V., Cain, John C., Kang, Chae H., Ireland, Lynne M., Carr, Tracy L., Miller, Thomas R., Hancock, Arthur A., Nakane, Masaki, Esbenshade, Timothy A., Brune, Michael E., O'Neill, Alyssa B., Gauvin, Donna M., Katwala, Sweta P., Holladay, Mark W., Brioni, Jorge D., Sullivan, James P.
Published in Journal of medicinal chemistry (01.06.2004)
Published in Journal of medicinal chemistry (01.06.2004)
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Journal Article
6-heteroaryloxy- and 6-aryloxy-quinoline-2-carboxamides and uses thereof
Bogdan, Andrew, Koenig, John R, Peltier, Hillary, Cowart, Marlon D, Jinkerson, Tammie K, Kort, Michael E, Wakefield, Brian D, Liu, Bo, Matulenko, Mark A, Scanio, Marc J, Degoey, David A, Nelson, Derek W, Patel, Meena V
Year of Publication 18.04.2019
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Year of Publication 18.04.2019
Patent
6-HETEROARYLOXY- OR 6-ARYLOXY-QUINOLINE-2-CARBOXAMIDES AND METHOD OF USE
Bogdan, Andrew, Koenig, John R, Peltier, Hillary, Cowart, Marlon D, Jinkerson, Tammie K, Kort, Michael E, Liu, Bo, Wakefield, Brian D, DeGoey, David A, Matulenko, Mark A, Scanio, Marc J, Nelson, Derek W, Patel, Meena V
Year of Publication 22.11.2018
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Year of Publication 22.11.2018
Patent