Paralog-selective Hsp90 inhibitors define tumor-specific regulation of HER2
Patel, Pallav D, Yan, Pengrong, Seidler, Paul M, Patel, Hardik J, Sun, Weilin, Yang, Chenghua, Que, Nanette S, Taldone, Tony, Finotti, Paola, Stephani, Ralph A, Gewirth, Daniel T, Chiosis, Gabriela
Published in Nature chemical biology (01.11.2013)
Published in Nature chemical biology (01.11.2013)
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Journal Article
Improved targeting of JAK2 leads to increased therapeutic efficacy in myeloproliferative neoplasms
Bhagwat, Neha, Koppikar, Priya, Keller, Matthew, Marubayashi, Sachie, Shank, Kaitlyn, Rampal, Raajit, Qi, Jun, Kleppe, Maria, Patel, Hardik J., Shah, Smit K., Taldone, Tony, Bradner, James E., Chiosis, Gabriela, Levine, Ross L.
Published in Blood (27.03.2014)
Published in Blood (27.03.2014)
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Journal Article
Experimental and Structural Testing Module to Analyze Paralogue-Specificity and Affinity in the Hsp90 Inhibitors Series
Taldone, Tony, Patel, Pallav D, Patel, Maulik, Patel, Hardik J, Evans, Christopher E, Rodina, Anna, Ochiana, Stefan, Shah, Smit K, Uddin, Mohammad, Gewirth, Daniel, Chiosis, Gabriela
Published in Journal of medicinal chemistry (12.09.2013)
Published in Journal of medicinal chemistry (12.09.2013)
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Journal Article
Molecular Stressors Engender Protein Connectivity Dysfunction through Aberrant N-Glycosylation of a Chaperone
Yan, Pengrong, Patel, Hardik J., Sharma, Sahil, Corben, Adriana, Wang, Tai, Panchal, Palak, Yang, Chenghua, Sun, Weilin, Araujo, Thais L., Rodina, Anna, Joshi, Suhasini, Robzyk, Kenneth, Gandu, Srinivasa, White, Julie R., de Stanchina, Elisa, Modi, Shanu, Janjigian, Yelena Y., Hill, Elizabeth G., Liu, Bei, Erdjument-Bromage, Hediye, Neubert, Thomas A., Que, Nanette L.S., Li, Zihai, Gewirth, Daniel T., Taldone, Tony, Chiosis, Gabriela
Published in Cell reports (Cambridge) (30.06.2020)
Published in Cell reports (Cambridge) (30.06.2020)
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Journal Article
Synthesis and evaluation of cell-permeable biotinylated PU-H71 derivatives as tumor Hsp90 probes
Taldone, Tony, Rodina, Anna, DaGama Gomes, Erica M, Riolo, Matthew, Patel, Hardik J, Alonso-Sabadell, Raul, Zatorska, Danuta, Patel, Maulik R, Kishinevsky, Sarah, Chiosis, Gabriela
Published in Beilstein journal of organic chemistry (15.03.2013)
Published in Beilstein journal of organic chemistry (15.03.2013)
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Journal Article
The epichaperome is an integrated chaperome network that facilitates tumour survival
Rodina, Anna, Wang, Tai, Yan, Pengrong, Gomes, Erica DaGama, Dunphy, Mark P. S., Pillarsetty, Nagavarakishore, Koren, John, Gerecitano, John F., Taldone, Tony, Zong, Hongliang, Caldas-Lopes, Eloisi, Alpaugh, Mary, Corben, Adriana, Riolo, Matthew, Beattie, Brad, Pressl, Christina, Peter, Radu I., Xu, Chao, Trondl, Robert, Patel, Hardik J., Shimizu, Fumiko, Bolaender, Alexander, Yang, Chenghua, Panchal, Palak, Farooq, Mohammad F., Kishinevsky, Sarah, Modi, Shanu, Lin, Oscar, Chu, Feixia, Patil, Sujata, Erdjument-Bromage, Hediye, Zanzonico, Pat, Hudis, Clifford, Studer, Lorenz, Roboz, Gail J., Cesarman, Ethel, Cerchietti, Leandro, Levine, Ross, Melnick, Ari, Larson, Steven M., Lewis, Jason S., Guzman, Monica L., Chiosis, Gabriela
Published in Nature (London) (20.10.2016)
Published in Nature (London) (20.10.2016)
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Journal Article
N‐Glycosylation‐Induced Pathologic Protein Conformations as a Tool to Guide the Selection of Biologically Active Small Molecules
Magni, Andrea, Sciva, Cristiano, Castelli, Matteo, Digwal, Chander S., Rodina, Anna, Sharma, Sahil, Ochiana, Stefan, Patel, Hardik J., Shah, Smit, Chiosis, Gabriela, Moroni, Elisabetta, Colombo, Giorgio
Published in Chemistry : a European journal (25.09.2024)
Published in Chemistry : a European journal (25.09.2024)
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Journal Article
Structure–Activity Relationship in a Purine-Scaffold Compound Series with Selectivity for the Endoplasmic Reticulum Hsp90 Paralog Grp94
Patel, Hardik J, Patel, Pallav D, Ochiana, Stefan O, Yan, Pengrong, Sun, Weilin, Patel, Maulik R, Shah, Smit K, Tramentozzi, Elisa, Brooks, James, Bolaender, Alexander, Shrestha, Liza, Stephani, Ralph, Finotti, Paola, Leifer, Cynthia, Li, Zihai, Gewirth, Daniel T, Taldone, Tony, Chiosis, Gabriela
Published in Journal of medicinal chemistry (14.05.2015)
Published in Journal of medicinal chemistry (14.05.2015)
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Journal Article
Chemical tools for epichaperome-mediated interactome dysfunctions of the central nervous system
Bolaender, Alexander, Zatorska, Danuta, He, Huazhong, Joshi, Suhasini, Sharma, Sahil, Digwal, Chander S., Patel, Hardik J., Sun, Weilin, Imber, Brandon S., Ochiana, Stefan O., Patel, Maulik R., Shrestha, Liza, Shah, Smit. K., Wang, Shuo, Karimov, Rashad, Tao, Hui, Patel, Pallav D., Martin, Ananda Rodilla, Yan, Pengrong, Panchal, Palak, Almodovar, Justina, Corben, Adriana, Rimner, Andreas, Ginsberg, Stephen D., Lyashchenko, Serge, Burnazi, Eva, Ku, Anson, Kalidindi, Teja, Lee, Sang Gyu, Grkovski, Milan, Beattie, Bradley J., Zanzonico, Pat, Lewis, Jason S., Larson, Steve, Rodina, Anna, Pillarsetty, Nagavarakishore, Tabar, Viviane, Dunphy, Mark P., Taldone, Tony, Shimizu, Fumiko, Chiosis, Gabriela
Published in Nature communications (03.08.2021)
Published in Nature communications (03.08.2021)
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Journal Article
Mutations in the Yeast Hsp70, Ssa1, at P417 Alter ATP Cycling, Interdomain Coupling, and Specific Chaperone Functions
Needham, Patrick G., Patel, Hardik J., Chiosis, Gabriela, Thibodeau, Patrick H., Brodsky, Jeffrey L.
Published in Journal of molecular biology (11.09.2015)
Published in Journal of molecular biology (11.09.2015)
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Journal Article
Heat Shock Protein 70 Inhibitors. 1. 2,5′-Thiodipyrimidine and 5‑(Phenylthio)pyrimidine Acrylamides as Irreversible Binders to an Allosteric Site on Heat Shock Protein 70
Kang, Yanlong, Taldone, Tony, Patel, Hardik J, Patel, Pallav D, Rodina, Anna, Gozman, Alexander, Maharaj, Ronnie, Clement, Cristina C, Patel, Maulik R, Brodsky, Jeffrey L, Young, Jason C, Chiosis, Gabriela
Published in Journal of medicinal chemistry (27.02.2014)
Published in Journal of medicinal chemistry (27.02.2014)
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Journal Article
Heat Shock Protein 70 Inhibitors. 2. 2,5′-Thiodipyrimidines, 5‑(Phenylthio)pyrimidines, 2‑(Pyridin-3-ylthio)pyrimidines, and 3‑(Phenylthio)pyridines as Reversible Binders to an Allosteric Site on Heat Shock Protein 70
Taldone, Tony, Kang, Yanlong, Patel, Hardik J, Patel, Maulik R, Patel, Pallav D, Rodina, Anna, Patel, Yogita, Gozman, Alexander, Maharaj, Ronnie, Clement, Cristina C, Lu, Alvin, Young, Jason C, Chiosis, Gabriela
Published in Journal of medicinal chemistry (27.02.2014)
Published in Journal of medicinal chemistry (27.02.2014)
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Journal Article
Protein chaperones: a composition of matter review (2008 - 2013)
Taldone, Tony, Patel, Hardik J, Bolaender, Alexander, Patel, Maulik R, Chiosis, Gabriela
Published in Expert opinion on therapeutic patents (01.05.2014)
Published in Expert opinion on therapeutic patents (01.05.2014)
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Journal Article
About the reaction of aryl fluorides with sodium sulfide: investigation into the selectivity of substitution of fluorobenzonitriles to yield mercaptobenzonitriles via SNAr displacement of fluorine
Taldone, Tony, Patel, Pallav D., Patel, Hardik J., Chiosis, Gabriela
Published in Tetrahedron letters (16.05.2012)
Published in Tetrahedron letters (16.05.2012)
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