Orphan G-protein-coupled receptors and natural ligand discovery
Howard, Andrew D, McAllister, George, Feighner, Scott D, Liu, Qingyun, Nargund, Ravi P, Van der Ploeg, Lex H.T, Patchett, Arthur A
Published in Trends in Pharmacological Sciences (01.03.2001)
Published in Trends in Pharmacological Sciences (01.03.2001)
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Book Review
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Receptor for Motilin Identified in the Human Gastrointestinal System
Feighner, Scott D., Tan, Carina P., McKee, Karen Kulju, Palyha, Oksana C., Hreniuk, Donna L., Pong, Sheng-Shung, Austin, Christopher P., Figueroa, David, MacNeil, Douglas, Cascieri, Margaret A., Nargund, Ravi, Bakshi, Raman, Abramovitz, Mark, Stocco, Rino, Kargman, Stacia, O'Neill, Gary, Lex H. T. Van Der Ploeg, Evans, Jilly, Patchett, Arthur A., Smith, Roy G., Howard, Andrew D.
Published in Science (American Association for the Advancement of Science) (25.06.1999)
Published in Science (American Association for the Advancement of Science) (25.06.1999)
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A Role for the Melanocortin 4 Receptor in Sexual Function
Lex H. T. Van der Ploeg, Martin, William J., Howard, Andrew D., Nargund, Ravi P., Austin, Christopher P., Guan, Xiaoming, Drisko, Jennifer, Cashen, Doreen, Sebhat, Iyassu, Patchett, Arthur A., Figueroa, David J., DiLella, Anthony G., Connolly, Brett M., Weinberg, David H., Tan, Carina P., Palyha, Oksana C., Pong, Sheng-Shung, MacNeil, Tanya, Rosenblum, Charles, Vongs, Aurawan, Tang, Rui, Yu, Hong, Sailer, Andreas W., Fong, Tung Ming, Huang, Cathy, Tota, Michael R., Chang, Ray S., Stearns, Ralph, Tamvakopoulos, Constantin, Christ, George, Drazen, Deborah L., Spar, Brian D., Nelson, Randy J., MacIntyre, D. Euan
Published in Proceedings of the National Academy of Sciences - PNAS (20.08.2002)
Published in Proceedings of the National Academy of Sciences - PNAS (20.08.2002)
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Antibacterial Agents That Inhibit Lipid a Biosynthesis
Onishi, H. Russell, Pelak, Barbara A., Gerckens, Lynn S., Silver, Lynn L., Kahan, Frederick M., Chen, Meng-Hsin, Patchett, Arthur A., Galloway, Susan M., Hyland, Sheryl A., Anderson, Matt S., Christian R. H. Raetz
Published in Science (American Association for the Advancement of Science) (08.11.1996)
Published in Science (American Association for the Advancement of Science) (08.11.1996)
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Rapid Identification of Subtype-Selective Agonists of the Somatostatin Receptor Through Combinatorial Chemistry
Rohrer, Susan P., Birzin, Elizabeth T., Mosley, Ralph T., Berk, Scott C., Hutchins, Steven M., Shen, Dong-Ming, Xiong, Yusheng, Hayes, Edward C., Parmar, Rupa M., Foor, Forrest, Mitra, Sudha W., Degrado, Sylvia J., Shu, Min, Klopp, John M., Cai, Sheng-Jian, Blake, Allan, Wanda W. S. Chan, Pasternak, Alex, Yang, Lihu, Patchett, Arthur A., Smith, Roy G., Chapman, Kevin T., Schaeffer, James M.
Published in Science (American Association for the Advancement of Science) (23.10.1998)
Published in Science (American Association for the Advancement of Science) (23.10.1998)
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Peptidomimetic Regulation of Growth Hormone Secretion
Smith, Roy G, Van der Ploeg, Lex H. T, Howard, Andrew D, Feighner, Scott D, Cheng, Kang, Hickey, Gerard J, Wyvratt, Matthew J, Fisher, Mike H, Nargund, Ravi P, Patchett, Arthur A
Published in Endocrine reviews (01.10.1997)
Published in Endocrine reviews (01.10.1997)
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Design and Pharmacology of N-[(3R)-1,2,3,4-Tetrahydroisoquinolinium- 3-ylcarbonyl]-(1R)-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1H-1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine (1), a Potent, Selective, Melanocortin Subtype-4 Receptor Agonist
Sebhat, Iyassu K, Martin, William J, Ye, Zhixiong, Barakat, Khaled, Mosley, Ralph T, Johnston, David B. R, Bakshi, Raman, Palucki, Brenda, Weinberg, David H, MacNeil, Tanya, Kalyani, Rubana N, Tang, Rui, Stearns, Ralph A, Miller, Randy R, Tamvakopoulos, Constantin, Strack, Alison M, McGowan, Erin, Cashen, Doreen E, Drisko, Jennifer E, Hom, Gary J, Howard, Andrew D, MacIntyre, D. Euan, van der Ploeg, Lex H. T, Patchett, Arthur A, Nargund, Ravi P
Published in Journal of medicinal chemistry (10.10.2002)
Published in Journal of medicinal chemistry (10.10.2002)
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Design and Biological Activities of L-163,191 (MK-0677): A Potent, Orally Active Growth Hormone Secretagogue
Patchett, A. A., Nargund, R. P., Tata, J. R., M.-H. Chen, Barakat, K. J., Johnston, D. B. R., Cheng, K., W. W.-S. CHan, Butler, B., Hickey, G., Jacks, T., Schleim, K., S.-S. Pong, L.-Y. P. Chaung, Chen, H. Y., Frazier, E., Leung, K. H., S.-H. L. Chiu, Smith, Roy G.
Published in Proceedings of the National Academy of Sciences - PNAS (18.07.1995)
Published in Proceedings of the National Academy of Sciences - PNAS (18.07.1995)
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Structural Requirements for the Activation of the Human Growth Hormone Secretagogue Receptor by Peptide and Nonpeptide Secretagogues
Feighner, Scott D, Howard, Andrew D, Prendergast, Kristine, Palyha, Oksana C, Hreniuk, Donna L, Nargund, Ravi, Underwood, Dennis, Tata, James R, Dean, Dennis C, Tan, Carina P, McKee, Karen Kulju, Woods, John W, Patchett, Arthur A, Smith, Roy G, Van der Ploeg, Lex H. T
Published in Molecular endocrinology (Baltimore, Md.) (01.01.1998)
Published in Molecular endocrinology (Baltimore, Md.) (01.01.1998)
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Peptidomimetic Growth Hormone Secretagogues. Design Considerations and Therapeutic Potential
Nargund, Ravi P, Patchett, Arthur A, Bach, Mark A, Murphy, M. Gail, Smith, Roy G
Published in Journal of medicinal chemistry (13.08.1998)
Published in Journal of medicinal chemistry (13.08.1998)
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Allele-specific activation of genetically engineered receptors
Strader, C D, Gaffney, T, Sugg, E E, Candelore, M R, Keys, R, Patchett, A A, Dixon, R A
Published in The Journal of biological chemistry (05.01.1991)
Published in The Journal of biological chemistry (05.01.1991)
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Identification of a new G-protein-linked receptor for growth hormone secretagogues
Pong, S S, Chaung, L Y, Dean, D C, Nargund, R P, Patchett, A A, Smith, R G
Published in Molecular endocrinology (Baltimore, Md.) (01.01.1996)
Published in Molecular endocrinology (Baltimore, Md.) (01.01.1996)
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Spiro[1H-indene-1,4‘-piperidine] Derivatives As Potent and Selective Non-Peptide Human Somatostatin Receptor Subtype 2 (sst2) Agonists
Yang, Lihu, Guo, Liangqin, Pasternak, Alexander, Mosley, Ralph, Rohrer, Susan, Birzin, Elizabeth, Foor, Forrest, Cheng, Kang, Schaeffer, James, Patchett, Arthur A
Published in Journal of medicinal chemistry (18.06.1998)
Published in Journal of medicinal chemistry (18.06.1998)
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Ligand Activation Domain of Human Orphan Growth Hormone (GH) Secretagogue Receptor (GHS-R) Conserved from Pufferfish to Humans
Palyha, Oksana C, Feighner, Scott D, Tan, Carina P, McKee, Karen Kulju, Hreniuk, Donna L, Gao, Ying-Duo, Schleim, Klaus D, Yang, Lihu, Morriello, Gregori J, Nargund, Ravi, Patchett, Arthur A, Howard, Andrew D, Smith, Roy G
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2000)
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2000)
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Optimization of a privileged structure leading to potent and selective human melanocortin subtype-4 receptor ligands
Bakshi, Raman K., Hong, Qingmei, Tang, Rui, Kalyani, Rubana N., MacNeil, Tanya, Weinberg, David H., Van der Ploeg, Lex H.T., Patchett, Arthur A., Nargund, Ravi P.
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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Synthesis and Biological Activities of Potent Peptidomimetics Selective for Somatostatin Receptor Subtype 2
Yang, Lihu, Berk, Scott C., Rohrer, Susan P., Mosley, Ralph T., Guo, Liangqin, Underwood, Dennis J., Arison, Byron H., Birzin, Elizabeth T., Hayes, Edward C., Mitra, Sudha W., Parmar, Rupa M., Cheng, Kang, Wu, Tsuei-Ju, Butler, Bridgette S., Foor, Forrest, Pasternak, Alexander, Pan, Yanping, Silva, Maria, Freidinger, Roger M., Smith, Roy G., Chapman, Kevin, Schaeffer, James M., Patchett, Arthur A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1998)
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Discovery and activity of (1 R,4 S,6 R)- N-[(1 R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-2-methyl-2-azabicyclo[2.2.2]octane-6-carboxamide (3, RY764), a potent and selective melanocortin subtype-4 receptor agonist
Ye, Zhixiong, Guo, Liangqin, Barakat, Khaled J., Pollard, Patrick G., Palucki, Brenda L., Sebhat, Iyassu K., Bakshi, Raman K., Tang, Rui, Kalyani, Rubana N., Vongs, Aurawan, Chen, Airu S., Chen, Howard Y., Rosenblum, Charles I., MacNeil, Tanya, Weinberg, David H., Peng, Qianping, Tamvakopoulos, Constantin, Miller, Randy R., Stearns, Ralph A., Cashen, Doreen E., Martin, William J., Metzger, Joseph M., Strack, Alison M., MacIntyre, D. Euan, Van der Ploeg, Lex H.T., Patchett, Arthur A., Wyvratt, Matthew J., Nargund, Ravi P.
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
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A high proportion of fat relative to muscle mass is associated with poor bone strength and balance in pre-pubertal boys and girls: Implications for fracture risk
Ducher, G, Daly, R, Eser, P, Naughton, G, English, R, Patchett, A, Gravenmaker, K, Seibel, M, Javaid, A, McGrath, M, Haynes, W, Telford, R, Bass, S
Published in Bone (New York, N.Y.) (01.07.2009)
Published in Bone (New York, N.Y.) (01.07.2009)
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In vitro pharmacology of L-158,809, a new highly potent and selective angiotensin II receptor antagonist
CHANG, R. S. L, SIEGL, P. K. S, CLINESCHMIDT, B. V, MANTLO, N. B, CHAKRAVARTY, P. K, GREENLEE, W. J, PATCHETT, A. A, LOTTI, V. J
Published in The Journal of pharmacology and experimental therapeutics (01.07.1992)
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Published in The Journal of pharmacology and experimental therapeutics (01.07.1992)
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