Donated chemical probes for open science
Müller, Susanne, Ackloo, Suzanne, Arrowsmith, Cheryl H, Bauser, Marcus, Baryza, Jeremy L, Blagg, Julian, Böttcher, Jark, Bountra, Chas, Brown, Peter J, Bunnage, Mark E, Carter, Adrian J, Damerell, David, Dötsch, Volker, Drewry, David H, Edwards, Aled M, Edwards, James, Elkins, Jon M, Fischer, Christian, Frye, Stephen V, Gollner, Andreas, Grimshaw, Charles E, IJzerman, Adriaan, Hanke, Thomas, Hartung, Ingo V, Hitchcock, Steve, Howe, Trevor, Hughes, Terry V, Laufer, Stefan, Li, Volkhart Mj, Liras, Spiros, Marsden, Brian D, Matsui, Hisanori, Mathias, John, O'Hagan, Ronan C, Owen, Dafydd R, Pande, Vineet, Rauh, Daniel, Rosenberg, Saul H, Roth, Bryan L, Schneider, Natalie S, Scholten, Cora, Singh Saikatendu, Kumar, Simeonov, Anton, Takizawa, Masayuki, Tse, Chris, Thompson, Paul R, Treiber, Daniel K, Viana, Amélia Yi, Wells, Carrow I, Willson, Timothy M, Zuercher, William J, Knapp, Stefan, Mueller-Fahrnow, Anke
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Published in eLife (20.04.2018)
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Published in Journal of molecular biology (28.03.2008)
Published in Journal of molecular biology (28.03.2008)
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Sharma, Rakesh K., Otsuka, Masami, Pande, Vineet, Inoue, Jun-ichiro, João Ramos, Maria
Published in Bioorganic & medicinal chemistry letters (20.12.2004)
Published in Bioorganic & medicinal chemistry letters (20.12.2004)
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Koldenhof, Patrick, Bemelmans, Martijn P., Ghosh, Brahma, Damm‐Ganamet, Kelly L., van Vlijmen, Herman W. T., Pande, Vineet
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Published in Proteins, structure, function, and bioinformatics (09.02.2024)
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Verhoeven, Jonas, Deraet, Xavier, Pande, Vineet, Sun, Weimei, Alonso, Mercedes, De Proft, Frank, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido
Published in Journal of organic chemistry (04.12.2020)
Published in Journal of organic chemistry (04.12.2020)
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Alchemical Free Energy Calculations on Membrane-Associated Proteins
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Published in Journal of chemical theory and computation (14.11.2023)
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Brehmer, Dirk, Beke, Lijs, Wu, Tongfei, Millar, Hillary J, Moy, Christopher, Sun, Weimei, Mannens, Geert, Pande, Vineet, Boeckx, An, van Heerde, Erika, Nys, Thomas, Gustin, Emmanuel M, Verbist, Bie, Zhou, Longen, Fan, Yue, Bhargava, Vipul, Safabakhsh, Pegah, Vinken, Petra, Verhulst, Tinne, Gilbert, Angelique, Rai, Sumit, Graubert, Timothy A, Pastore, Friederike, Fiore, Danilo, Gu, Junchen, Johnson, Amy, Philippar, Ulrike, Morschhäuser, Barbara, Walker, David, De Lange, Desiree, Keersmaekers, Vikki, Viellevoye, Marcel, Diels, Gaston, Schepens, Wim, Thuring, Jan Willem, Meerpoel, Lieven, Packman, Kathryn, Lorenzi, Matthew V, Laquerre, Sylvie
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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Verhoeven, Jonas, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Pande, Vineet, Brambilla, Marta, Van Hecke, Kristof, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido
Published in Synlett (02.06.2021)
Published in Synlett (02.06.2021)
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Zhang, Zhuming, Connolly, Peter J, Lim, Heng Keang, Pande, Vineet, Meerpoel, Lieven, Teleha, Christopher, Branch, Jonathan R, Ondrus, Janine, Hickson, Ian, Bush, Tammy, Luistro, Leopoldo, Packman, Kathryn, Bischoff, James R, Ibrahim, Salam, Parrett, Christopher, Chong, Yolanda, Gottardis, Marco M, Bignan, Gilles
Published in Journal of medicinal chemistry (28.01.2021)
Published in Journal of medicinal chemistry (28.01.2021)
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Verhoeven, Jonas, De Vleeschouwer, Freija, Kong, Hanchu, Van Hecke, Kristof, Pande, Vineet, Sun, Weimei, Vos, Ann, Wu, Tongfei, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido
Published in Chemistry : a European journal (02.12.2019)
Published in Chemistry : a European journal (02.12.2019)
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Zhang, Zhuming, Ghosh, Avijit, Connolly, Peter J, King, Peter, Wilde, Thomas, Wang, Jianyao, Dong, Yawei, Li, Xueliang, Liao, Daohong, Chen, Hao, Tian, Gaochao, Suarez, Javier, Bonnette, William G, Pande, Vineet, Diloreto, Karen A, Shi, Yifan, Patel, Shefali, Pietrak, Beth, Szewczuk, Lawrence, Sensenhauser, Carlo, Dallas, Shannon, Edwards, James P, Bachman, Kurtis E, Evans, David C
Published in Journal of medicinal chemistry (12.08.2021)
Published in Journal of medicinal chemistry (12.08.2021)
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Cabaye, Alexandre, Nguyen, Kong T, Liu, Lihua, Pande, Vineet, Schapira, Matthieu
Published in Proteins, structure, function, and bioinformatics (01.07.2015)
Published in Proteins, structure, function, and bioinformatics (01.07.2015)
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Preclinical efficacy of the potent, selective menin-KMT2A inhibitor JNJ-75276617 (bleximenib) in KMT2A- and NPM1-altered leukemias
Kwon, Min Chul, Thuring, Jan Willem, Querolle, Olivier, Dai, Xuedong, Verhulst, Tinne, Pande, Vineet, Marien, Ann, Goffin, Dries, Wenge, Daniela V., Yue, Hong, Cutler, Jevon A., Jin, Cyrus, Perner, Florian, Hogeling, Shanna M., Shaffer, Paul L., Jacobs, Frank, Vinken, Petra, Cai, Wei, Keersmaekers, Vikki, Eyassu, Filmon, Bhogal, Balpreet, Verstraeten, Karin, El Ashkar, Sara, Perry, Jennifer A., Jayaguru, Prathiba, Barreyro, Laura, Kuchnio, Anna, Darville, Nicolas, Krosky, Daniel, Urbanietz, Gregor, Verbist, Bie, Edwards, James P., Cowley, Glenn S., Kirkpatrick, Robert, Steele, Ruth, Ferrante, Lucille, Guttke, Christina, Daskalakis, Nikki, Pietsch, E. Christine, Wilson, David M., Attar, Ricardo, Elsayed, Yusri, Fischer, Eric S., Schuringa, Jan Jacob, Armstrong, Scott A., Packman, Kathryn, Philippar, Ulrike
Published in Blood (12.09.2024)
Published in Blood (12.09.2024)
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Pharmacological Characterization of JNJ-75276617, a Menin-KMT2A Inhibitor, As Targeted Treatment for KMT2A-Altered and NPM1-Mutant Acute Leukemia
Kwon, Min Chul, Querolle, Olivier, Dai, Xuedong, Thuring, Jan Willem, Verhulst, Tinne, Marien, Ann, Goffin, Dries, Cai, Wei, Keersmaekers, Vikki, Eyassu, Filmon, Verstraeten, Karin, El Ashkar, Sara, Hogeling, Shanna M, Jacob, Frank, Vinken, Petra, Darville, Nicolas, Pande, Vineet, Krosky, Daniel, Urbanietz, Gregor, Verbist, Bie, Ferrante, Lucille A., Drenberg, Christina Diane, Wilson, David, Attar, Ricardo M., Schuringa, Jan Jacob, Daskalakis, Nikki, Packman, Kathryn, Pietsch, Christine, Elsayed, Yusri, Philippar, Ulrike
Published in Blood (15.11.2022)
Published in Blood (15.11.2022)
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