In silico identification of a novel Cdc2‐like kinase 2 (CLK2) inhibitor in triple negative breast cancer
Huang, Cheng‐Chiao, Hsu, Chia‐Ming, Chao, Min‐Wu, Hsu, Kai‐Cheng, Lin, Tony Eight, Yen, Shih‐Chung, Tu, Huang‐Ju, Pan, Shiow‐Lin
Published in Protein science (01.06.2024)
Published in Protein science (01.06.2024)
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An ensemble machine learning model generates a focused screening library for the identification of CDK8 inhibitors
Lin, Tony Eight, Yen, Dyan, HuangFu, Wei‐Chun, Wu, Yi‐Wen, Hsu, Jui‐Yi, Yen, Shih‐Chung, Sung, Tzu‐Ying, Hsieh, Jui‐Hua, Pan, Shiow‐Lin, Yang, Chia‐Ron, Huang, Wei‐Jan, Hsu, Kai‐Cheng
Published in Protein science (01.06.2024)
Published in Protein science (01.06.2024)
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Anti-metastatic activity of MPT0G211, a novel HDAC6 inhibitor, in human breast cancer cells in vitro and in vivo
Hsieh, Yi-Ling, Tu, Huang-Ju, Pan, Shiow-Lin, Liou, Jing-Ping, Yang, Chia-Ron
Published in Biochimica et biophysica acta. Molecular cell research (01.06.2019)
Published in Biochimica et biophysica acta. Molecular cell research (01.06.2019)
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The study of a novel CDK8 inhibitor E966-0530–45418 that inhibits prostate cancer metastasis in vitro and in vivo
Ho, Tai-Yuan, Sung, Ting-Yi, Pan, Shiow-Lin, Huang, Wei-Jan, Hsu, Kai-Cheng, Hsu, Jui-Yi, Lin, Tony Eight, Hsu, Chia-Ming, Yang, Chia-Ron
Published in Biomedicine & pharmacotherapy (01.06.2023)
Published in Biomedicine & pharmacotherapy (01.06.2023)
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Synthesis and evaluation of potent (iso)ellipticine-based inhibitors of MYLK4 accessed via expeditious synthesis from isoquinolin-5-ol
Lee, Szu, Chao, Min-Wu, Wu, Yi-Wen, Hsu, Chia-Min, Lin, Tony Eight, Hsu, Kai-Cheng, Pan, Shiow-Lin, Lee, Hsueh-Yun
Published in RSC advances (26.10.2023)
Published in RSC advances (26.10.2023)
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Isoindoline scaffold-based dual inhibitors of HDAC6 and HSP90 suppressing the growth of lung cancer in vitro and in vivo
Ojha, Ritu, Nepali, Kunal, Chen, Chun-Han, Chuang, Kuo-Hsiang, Wu, Tung-Yun, Lin, Tony Eight, Hsu, Kai-Cheng, Chao, Min-Wu, Lai, Mei-Jung, Lin, Mei-Hsiang, Huang, Han-Li, Chang, Chao-Di, Pan, Shiow-Lin, Chen, Mei-Chuan, Liou, Jing-Ping
Published in European journal of medicinal chemistry (15.03.2020)
Published in European journal of medicinal chemistry (15.03.2020)
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In silico identification and biological evaluation of a selective MAP4K4 inhibitor against pancreatic cancer
Chang, Chao-Di, Chao, Min-Wu, Lee, Hsueh-Yun, Liu, Yi-Ting, Tu, Huang-Ju, Lien, Ssu-Ting, Lin, Tony Eight, Sung, Tzu-Ying, Yen, Shih-Chung, Huang, Sing-Han, Hsu, Kai-Cheng, Pan, Shiow-Lin
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
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Physalin F induces cell apoptosis in human renal carcinoma cells by targeting NF-kappaB and generating reactive oxygen species
Wu, Szu-Ying, Leu, Yann-Lii, Chang, Ya-Ling, Wu, Tian-Shung, Kuo, Ping-Chung, Liao, Yu-Ren, Teng, Che-Ming, Pan, Shiow-Lin
Published in PloS one (16.07.2012)
Published in PloS one (16.07.2012)
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A novel dual HDAC and HSP90 inhibitor, MPT0G449, downregulates oncogenic pathways in human acute leukemia in vitro and in vivo
Wu, Yi-Wen, Chao, Min-Wu, Tu, Huang-Ju, Chen, Liang-Chieh, Hsu, Kai-Cheng, Liou, Jing-Ping, Yang, Chia-Ron, Yen, Shih-Chung, HuangFu, Wei-Chun, Pan, Shiow-Lin
Published in Oncogenesis (New York, NY) (13.05.2021)
Published in Oncogenesis (New York, NY) (13.05.2021)
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TIMP3 expression associates with prognosis in colorectal cancer and its novel arylsulfonamide inducer, MPT0B390, inhibits tumor growth, metastasis and angiogenesis
Huang, Han-Li, Liu, Yi-Min, Sung, Ting-Yi, Huang, Tsui-Chin, Cheng, Ya-Wen, Liou, Jing-Ping, Pan, Shiow-Lin
Published in Theranostics (01.01.2019)
Published in Theranostics (01.01.2019)
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Dehydrocostuslactone suppresses angiogenesis in vitro and in vivo through inhibition of Akt/GSK-3β and mTOR signaling pathways
Wang, Chih-Ya, Tsai, An-Chi, Peng, Chieh-Yu, Chang, Ya-Ling, Lee, Kuo-Hsiung, Teng, Che-Ming, Pan, Shiow-Lin
Published in PloS one (16.02.2012)
Published in PloS one (16.02.2012)
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Design, Synthesis, Mechanisms of Action, and Toxicity of Novel 20(S)‑Sulfonylamidine Derivatives of Camptothecin as Potent Antitumor Agents
Wang, Mei-Juan, Liu, Ying-Qian, Chang, Ling-Chu, Wang, Chih-Ya, Zhao, Yong-Long, Zhao, Xiao-Bo, Qian, Keduo, Nan, Xiang, Yang, Liu, Yang, Xiao-Ming, Hung, Hsin-Yi, Yang, Jai-Sing, Kuo, Daih-Huang, Goto, Masuo, Morris-Natschke, Susan L, Pan, Shiow-Lin, Teng, Che-Ming, Kuo, Sheng-Chu, Wu, Tian-Shung, Wu, Yang-Chang, Lee, Kuo-Hsiung
Published in Journal of medicinal chemistry (24.07.2014)
Published in Journal of medicinal chemistry (24.07.2014)
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Dual Phosphoinositide 3-kinase/mammalian target of rapamycin inhibitor is an effective radiosensitizer for colorectal cancer
Chen, Yu-Hsuan, Wei, Ming-Feng, Wang, Chun-Wei, Lee, Hsiao-Wei, Pan, Shiow-Lin, Gao, Ming, Kuo, Sung-Hsin, Cheng, Ann-Lii, Teng, Che-Ming
Published in Cancer letters (28.02.2015)
Published in Cancer letters (28.02.2015)
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Combination treatment strategy for pancreatic cancer involving the novel HDAC inhibitor MPT0E028 with a MEK inhibitor beyond K-Ras status
Chao, Min-Wu, Chang, Li-Hsun, Tu, Huang-Ju, Chang, Chao-Di, Lai, Mei-Jung, Chen, Yi-Ying, Liou, Jing-Ping, Teng, Che-Ming, Pan, Shiow-Lin
Published in Clinical epigenetics (29.05.2019)
Published in Clinical epigenetics (29.05.2019)
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α-Tomatine-mediated anti-cancer activity in vitro and in vivo through cell cycle- and caspase-independent pathways
Chao, Min-Wu, Chen, Chun-Han, Chang, Ya-Ling, Teng, Che-Ming, Pan, Shiow-Lin
Published in PloS one (06.09.2012)
Published in PloS one (06.09.2012)
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Journal Article
Identification and analysis of a selective DYRK1A inhibitor
Lin, Tony Eight, Chao, Min-Wu, HuangFu, Wei-Chun, Tu, Huang-Ju, Peng, Zhao-Xiang, Su, Chih-Jou, Sung, Tzu-Ying, Hsieh, Jui-Hua, Lee, Cheng-Chung, Yang, Chia-Ron, Pan, Shiow-Lin, Hsu, Kai-Cheng
Published in Biomedicine & pharmacotherapy (01.02.2022)
Published in Biomedicine & pharmacotherapy (01.02.2022)
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