Synthesis and structure-activity relationships for a new class of tetrahydronaphthalene amide inhibitors of Mycobacterium tuberculosis
Sutherland, Hamish S., Lu, Guo-Liang, Tong, Amy S.T., Conole, Daniel, Franzblau, Scott G., Upton, Anna M., Lotlikar, Manisha U., Cooper, Christopher B., Palmer, Brian D., Choi, Peter J., Denny, William A.
Published in European journal of medicinal chemistry (05.02.2022)
Published in European journal of medicinal chemistry (05.02.2022)
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Journal Article
Discovery and evaluation of inhibitors to the immunosuppressive enzyme indoleamine 2,3-dioxygenase 1 (IDO1): Probing the active site-inhibitor interactions
Tomek, Petr, Palmer, Brian D., Flanagan, Jack U., Sun, Chuanwen, Raven, Emma L., Ching, Lai-Ming
Published in European journal of medicinal chemistry (27.01.2017)
Published in European journal of medicinal chemistry (27.01.2017)
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Journal Article
Synthetic Studies to Help Elucidate the Metabolism of the Preclinical Candidate TBAJ-876-A Less Toxic and More Potent Analogue of Bedaquiline
Choi, Peter J, Conole, Daniel, Sutherland, Hamish S, Blaser, Adrian, Tong, Amy S T, Cooper, Christopher B, Upton, Anna M, Palmer, Brian D, Denny, William A
Published in Molecules (Basel, Switzerland) (20.03.2020)
Published in Molecules (Basel, Switzerland) (20.03.2020)
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Journal Article
Evaluation of Novel Inhibitors of Tryptophan Dioxygenases for Enzyme and Species Selectivity Using Engineered Tumour Cell Lines Expressing Either Murine or Human IDO1 or TDO2
Tijono, Sofian M, Palmer, Brian D, Tomek, Petr, Flanagan, Jack U, Henare, Kimiora, Gamage, Swarna, Braun, Lukas, Ching, Lai-Ming
Published in Pharmaceuticals (Basel, Switzerland) (31.08.2022)
Published in Pharmaceuticals (Basel, Switzerland) (31.08.2022)
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Journal Article
Mechanisms and biomaterials in pH-responsive tumour targeted drug delivery: A review
Kanamala, Manju, Wilson, William R, Yang, Mimi, Palmer, Brian D, Wu, Zimei
Published in Biomaterials (01.04.2016)
Published in Biomaterials (01.04.2016)
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Journal Article
Synthesis and Structure–Activity Relationships for the Anti-Mycobacterial Activity of 3-Phenyl-N-(Pyridin-2-ylmethyl)Pyrazolo[1,5-a]Pyrimidin-7-Amines
Sutherland, Hamish S., Choi, Peter J., Lu, Guo-Liang, Giddens, Anna C., Tong, Amy S. T., Franzblau, Scott G., Cooper, Christopher B., Palmer, Brian D., Denny, William A.
Published in Pharmaceuticals (Basel, Switzerland) (08.09.2022)
Published in Pharmaceuticals (Basel, Switzerland) (08.09.2022)
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Journal Article
4-Phenylpyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione Inhibitors of the Checkpoint Kinase Wee1. Structure−Activity Relationships for Chromophore Modification and Phenyl Ring Substitution
Palmer, Brian D, Thompson, Andrew M, Booth, R. John, Dobrusin, Ellen M, Kraker, Alan J, Lee, Ho H, Lunney, Elizabeth A, Mitchell, Lorna H, Ortwine, Daniel F, Smaill, Jeff B, Swan, Leesa M, Denny, William A
Published in Journal of medicinal chemistry (10.08.2006)
Published in Journal of medicinal chemistry (10.08.2006)
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Journal Article
3,5-Dialkoxypyridine analogues of bedaquiline are potent antituberculosis agents with minimal inhibition of the hERG channel
Sutherland, Hamish S., Tong, Amy S.T., Choi, Peter J., Blaser, Adrian, Conole, Daniel, Franzblau, Scott G., Lotlikar, Manisha U., Cooper, Christopher B., Upton, Anna M., Denny, William A., Palmer, Brian D.
Published in Bioorganic & medicinal chemistry (01.04.2019)
Published in Bioorganic & medicinal chemistry (01.04.2019)
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Journal Article
Structure-activity relationships for analogs of the tuberculosis drug bedaquiline with the naphthalene unit replaced by bicyclic heterocycles
Sutherland, Hamish S., Tong, Amy S.T., Choi, Peter J., Conole, Daniel, Blaser, Adrian, Franzblau, Scott G., Cooper, Christopher B., Upton, Anna M., Lotlikar, Manisha U., Denny, William A., Palmer, Brian D.
Published in Bioorganic & medicinal chemistry (01.05.2018)
Published in Bioorganic & medicinal chemistry (01.05.2018)
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Journal Article
Structure-activity relationships for unit C pyridyl analogues of the tuberculosis drug bedaquiline
Blaser, Adrian, Sutherland, Hamish S., Tong, Amy S.T., Choi, Peter J., Conole, Daniel, Franzblau, Scott G., Cooper, Christopher B., Upton, Anna M., Lotlikar, Manisha, Denny, William A., Palmer, Brian D.
Published in Bioorganic & medicinal chemistry (01.04.2019)
Published in Bioorganic & medicinal chemistry (01.04.2019)
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Journal Article
Synthesis and structure–activity relationships of soluble 8-substituted 4-(2-chlorophenyl)-9-hydroxypyrrolo[3,4- c]carbazole-1,3(2 H,6 H)-diones as inhibitors of the Wee1 and Chk1 checkpoint kinases
Smaill, Jeff B., Lee, Ho H., Palmer, Brian D., Thompson, Andrew M., Squire, Christopher J., Baker, Edward N., Booth, R. John, Kraker, Alan, Hook, Ken, Denny, William A.
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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Journal Article
Parallel discovery of selective and dual inhibitors of tryptophan dioxygenases IDO1 and TDO2 with a newly-modified enzymatic assay
Capochiani de Iudicibus, Rossella, Tomek, Petr, Palmer, Brian D., Tijono, Sofian M., Flanagan, Jack U., Ching, Lai-Ming
Published in Bioorganic & medicinal chemistry (01.06.2021)
Published in Bioorganic & medicinal chemistry (01.06.2021)
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Journal Article
Variations in the C-unit of bedaquiline provides analogues with improved biology and pharmacology
Sutherland, Hamish S., Tong, Amy S.T., Choi, Peter J., Blaser, Adrian, Franzblau, Scott G., Cooper, Christopher B., Upton, Anna M., Lotlikar, Manisha, Denny, William A., Palmer, Brian D.
Published in Bioorganic & medicinal chemistry (01.01.2020)
Published in Bioorganic & medicinal chemistry (01.01.2020)
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Journal Article
Thalidomide Pharmacokinetics and Metabolite Formation in Mice, Rabbits, and Multiple Myeloma Patients
CHUNG, Francisco, JUN LU, PALMER, Brian D, KESTELL, Philip, BROWETT, Peter, BAGULEY, Bruce C, TINGLE, Malcolm, CHING, Lai-Ming
Published in Clinical cancer research (01.09.2004)
Published in Clinical cancer research (01.09.2004)
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Journal Article
Synthetic studies towards isomeric pyrazolopyrimidines as potential ATP synthesis inhibitors of Mycobacterium tuberculosis. Structural correction of reported N-(6-(2-(dimethylamino)ethoxy)-5-fluoropyridin-3-yl)-2-(4-fluorophenyl)-5-(trifluoromethyl)pyrazolo[1,5-α]pyrimidin-7-amine
Choi, Peter J., Lu, Guo-Liang, Sutherland, Hamish S., Giddens, Anna C., Franzblau, Scott G., Cooper, Christopher B., Denny, William A., Palmer, Brian D.
Published in Tetrahedron letters (02.02.2022)
Published in Tetrahedron letters (02.02.2022)
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Journal Article
Labeling of Oxidizable Proteins with a Photoactivatable Analog of the Antitumor Agent DMXAA: Evidence for Redox Signaling in Its Mode of Action
Brauer, Romy, Wang, Liang-Chuan S., Woon, See-Tarn, Bridewell, David J.A., Henare, Kimiora, Malinger, Dieter, Palmer, Brian D., Vogel, Stefanie N., Kieda, Claudine, Tijono, Sofian M., Ching, Lai-Ming
Published in Neoplasia (New York, N.Y.) (01.09.2010)
Published in Neoplasia (New York, N.Y.) (01.09.2010)
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