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Published in Scientific reports (12.01.2018)
Published in Scientific reports (12.01.2018)
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Late-stage lipidation of fully elaborated tryptophan-containing peptides for improved pharmacokinetics
Huang, Chunhui, Wille, Cannon B., He, Huaibing, Reddy, Vijay Bhasker Gangula, Nargund, Ravi P., Lin, Songnian, Palani, Anandan
Published in Tetrahedron letters (22.03.2017)
Published in Tetrahedron letters (22.03.2017)
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Development of a New Structural Class of Broadly Acting HCV Non‐Nucleoside Inhibitors Leading to the Discovery of MK‐8876
McComas, Casey C., Palani, Anandan, Chang, Wei, Holloway, M. Katharine, Lesburg, Charles A., Li, Peng, Liverton, Nigel, Meinke, Peter T., Olsen, David B., Peng, Xuanjia, Soll, Richard M., Ummat, Ajay, Wu, Jie, Wu, Jin, Zorn, Nicolas, Ludmerer, Steven W.
Published in ChemMedChem (07.09.2017)
Published in ChemMedChem (07.09.2017)
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A general approach to access 5,6-dihydroindolo-naphthyridine ring system
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Published in Tetrahedron letters (05.04.2017)
Published in Tetrahedron letters (05.04.2017)
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The Discovery of Potent Antitumor Agent C11-Deoxypsymberin/irciniastatin A: Total Synthesis and Biology of Advanced Psymberin Analogs
Huang, Xianhai, Shao, Ning, Huryk, Robert, Palani, Anandan, Aslanian, Robert, Seidel-Dugan, Cynthia
Published in Organic letters (19.02.2009)
Published in Organic letters (19.02.2009)
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Discovery of a novel series of potent MK2 non-ATP competitive inhibitors using 1,2-substituted azoles as cis-amide isosteres
Xiao, Dong, Zhu, Xiaohong, Sofolarides, Michael, Degrado, Sylvia, Shao, Ning, Rao, Ashwin, Chen, Xiao, Aslanian, Robert, Fossetta, James, Tian, Fang, Trivedi, Prashant, Lundell, Daniel, Palani, Anandan
Published in Bioorganic & medicinal chemistry letters (01.08.2014)
Published in Bioorganic & medicinal chemistry letters (01.08.2014)
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HIV-1 Escape from a Small Molecule, CCR5-Specific Entry Inhibitor Does Not Involve CXCR4 Use
Trkola, Alexandra, Kuhmann, Shawn E., Strizki, Julie M., Maxwell, Elizabeth, Ketas, Tom, Morgan, Tom, Pugach, Pavel, Xu, Serena, Wojcik, Lisa, Tagat, Jayaram, Palani, Anandan, Shapiro, Sherry, Clader, John W., McCombie, Stuart, Reyes, Gregory R., Baroudy, Bahige M., Moore, John P.
Published in Proceedings of the National Academy of Sciences - PNAS (08.01.2002)
Published in Proceedings of the National Academy of Sciences - PNAS (08.01.2002)
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Discovery of SCH 900271, a Potent Nicotinic Acid Receptor Agonist for the Treatment of Dyslipidemia
Palani, Anandan, Rao, Ashwin U, Chen, Xiao, Huang, Xianhai, Su, Jing, Tang, Haiqun, Huang, Ying, Qin, Jun, Xiao, Dong, Degrado, Sylvia, Sofolarides, Michael, Zhu, Xiaohong, Liu, Zhidan, McKittrick, Brian, Zhou, Wei, Aslanian, Robert, Greenlee, William J, Senior, Mary, Cheewatrakoolpong, Boonlert, Zhang, Hongtao, Farley, Constance, Cook, John, Kurowski, Stan, Li, Qiu, van Heek, Margaret, Wang, Gangfeng, Hsieh, Yunsheng, Li, Fangbiao, Greenfeder, Scott, Chintala, Madhu
Published in ACS medicinal chemistry letters (12.01.2012)
Published in ACS medicinal chemistry letters (12.01.2012)
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Discovery of 4-[(Z)-(4-Bromophenyl)- (ethoxyimino)methyl]-1‘-[(2,4-dimethyl-3- pyridinyl)carbonyl]-4‘-methyl-1,4‘- bipiperidine N-Oxide (SCH 351125): An Orally Bioavailable Human CCR5 Antagonist for the Treatment of HIV Infection
Palani, Anandan, Shapiro, Sherry, Clader, John W, Greenlee, William J, Cox, Kathleen, Strizki, Julie, Endres, Michael, Baroudy, Bahige M
Published in Journal of medicinal chemistry (11.10.2001)
Published in Journal of medicinal chemistry (11.10.2001)
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Concise Formation of 4-Benzyl Piperidines and Related Derivatives Using a Suzuki Protocol
Vice, Susan, Bara, Tom, Bauer, Annette, Evans, C. Anderson, Ford, Jennifer, Josien, Hubert, McCombie, Stuart, Miller, Michael, Nazareno, Dennis, Palani, Anandan, Tagat, Jay
Published in Journal of organic chemistry (06.04.2001)
Published in Journal of organic chemistry (06.04.2001)
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Multi-step parallel synthesis enabled optimization of benzofuran derivatives as pan-genotypic non-nucleoside inhibitors of HCV NS5B
Xiao, Dong, Dai, Xing, Liu, Hong, He, Shuwen, Shi, Zhi-Cai, Ludmerer, Steven W., Li, Fangbiao, Nargund, Ravi, Palani, Anandan
Published in Bioorganic & medicinal chemistry letters (01.04.2020)
Published in Bioorganic & medicinal chemistry letters (01.04.2020)
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Discovery of MK-1084: An Orally Bioavailable and Low-Dose KRAS G12C Inhibitor
Ma, Xiaoshen, Sloman, David L., Duggal, Ruchia, Anderson, Kenneth D., Ballard, Jeanine E., Bharathan, Indu, Brynczka, Christopher, Gathiaka, Symon, Henderson, Timothy J., Lyons, Thomas W., Miller, Richard, Munsell, Erik V., Orth, Peter, Otte, Ryan D., Palani, Anandan, Rankic, Danica A., Robinson, Michelle R., Sather, Aaron C., Solban, Nicolas, Song, Xuelei Sherry, Wen, Xin, Xu, Zangwei, Yang, Yi, Yang, Ruojing, Day, Phil J., Stoeck, Alexander, Bennett, David Jonathan, Han, Yongxin
Published in Journal of medicinal chemistry (11.07.2024)
Published in Journal of medicinal chemistry (11.07.2024)
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Generation of Leads for γ‑Secretase Modulation
Mandal, Mihirbaran, Buevich, Alexei, Caldwell, John P, Hyde, Lynn, Huang, Xianhai, Liu, Xiaoxiang, McKittrick, Brian, Mazzola, Robert D, Pissarnitski, Dmitri, Palani, Anandan, Zhang, Lili, Parker, Eric, Xiao, Li, Rindgen, Diane, Zhu, Zhaoning
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Ligand-Dependent Site-Selective Suzuki Cross-Coupling of 3,5-Dichloropyridazines
Dai, Xing, Chen, Yonggang, Garrell, Stephanie, Liu, Hong, Zhang, Li-Kang, Palani, Anandan, Hughes, Gregory, Nargund, Ravi
Published in Journal of organic chemistry (02.08.2013)
Published in Journal of organic chemistry (02.08.2013)
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Discovery of MK-1084: An Orally Bioavailable and Low-Dose KRASG12C Inhibitor
Ma, Xiaoshen, Sloman, David L., Duggal, Ruchia, Anderson, Kenneth D., Ballard, Jeanine E., Bharathan, Indu, Brynczka, Christopher, Gathiaka, Symon, Henderson, Timothy J., Lyons, Thomas W., Miller, Richard, Munsell, Erik V., Orth, Peter, Otte, Ryan D., Palani, Anandan, Rankic, Danica A., Robinson, Michelle R., Sather, Aaron C., Solban, Nicolas, Song, Xuelei Sherry, Wen, Xin, Xu, Zangwei, Yang, Yi, Yang, Ruojing, Day, Phil J., Stoeck, Alexander, Bennett, David Jonathan, Han, Yongxin
Published in Journal of medicinal chemistry (11.07.2024)
Published in Journal of medicinal chemistry (11.07.2024)
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The Total Synthesis of Psymberin
Huang, Xianhai, Shao, Ning, Palani, Anandan, Aslanian, Robert, Buevich, Alexei
Published in Organic letters (21.06.2007)
Published in Organic letters (21.06.2007)
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Discovery of Insulin/GLP-1/Glucagon Triagonists for the Treatment of Diabetes and Obesity
Huang, Chunhui, Palani, Anandan, Yang, Zhiqiang, Deng, Qiaolin, Reddy, Vijay, Nargund, Ravi P., Lin, Songnian, Altezza, Simona, Bianchi, Elisabetta, Orvieto, Federica, Carrington, Paul
Published in ACS medicinal chemistry letters (11.08.2022)
Published in ACS medicinal chemistry letters (11.08.2022)
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