Synthesis of cyclic hydropyran oligolides with convergent amine, amide, phosphonate and furan appendages
Burke, Steven D., O'Donnell, Christopher J., Hans, Jeremy J., Moon, Choong Woon, Ng, Raymond A., Adkins, Thomas W., Packard, Garrick K.
Published in Tetrahedron letters (14.04.1997)
Published in Tetrahedron letters (14.04.1997)
Get full text
Journal Article
EIF4-A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO
TRAN, Chinh, PACKARD, Garrick, Kenneth, REICH, Siegfried, H, NILEWSKI, Christian, XIANG, Alan, Xin, ERNST, Justin, T, MICHELS, Theodore, SPRENGELER, Paul, A
Year of Publication 01.06.2017
Get full text
Year of Publication 01.06.2017
Patent
EIF4A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO
MICHELS, THEODORE, ERNST, JUSTIN T, PACKARD, GARRICK KENNETH, REICH, SIEGFRIED H, NILEWSKI, CHRISTIAN, SPRENGELER, PAUL A, XIANG, ALAN XIN, TRAN, CHINH
Year of Publication 01.06.2017
Get full text
Year of Publication 01.06.2017
Patent
EIF4A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO
TRAN Chinh Viet, PACKARD Garrick Kenneth, XIANG Alan X, MICHELS Theo, ERNST Justin T, NILEWSKI Christian, REICH Siegfried H, SPRENGELER Paul A
Year of Publication 25.05.2017
Get full text
Year of Publication 25.05.2017
Patent
TREX1 inhibitors and uses thereof
DUBENSKY, THOMAS WALTER JR, CLARK, RYAN C, ERNST, JUSTIN, PACKARD, GARRICK K, KALITA, BISWAJIT, DURAISWAMY, ATHISAYAMANI JEYARAJ, BUSCH, BRETT, NAGAMIZO, JOE FRED
Year of Publication 01.05.2022
Get full text
Year of Publication 01.05.2022
Patent
Synthesis of Rimocidinolide Methyl Ester, the Aglycone of (+)‐Rimocidin
Packard, Garrick K., Hu, Yueqing, Vescovi, Andrea, Rychnovsky, Scott D.
Published in Angewandte Chemie (17.05.2004)
Published in Angewandte Chemie (17.05.2004)
Get full text
Journal Article
METHODS OF SYNTHESIS AND PURIFICATION OF HETEROARYL COMPOUNDS
MORTENSEN, DEBORAH, PERRIN-NINKOVIC, SOPHIE, PYE, PHILIP, ZHAO, JINGJING, CHOUDHURY, ANUSUYA, SHEVLIN, GRAZIELLA, BEAUCHAMPS, MARIE GEORGES, KREILEIN, MATTHEW MICHAEL, PACKARD, GARRICK, KOTHARE, MOHIT ATUL, SAPIENZA, JOHN, LEONG, WILLIAM WEI-HWA, LEE, BRANDEN GINGSEE, ELSNER, JAN, HARRIS, ROY L, JOKIEL, PATRICK ANTHONY, RIGGS, JENNIFER, PAPA, PATRICK, GAMBOA, JUAN ANTONIO
Year of Publication 23.04.2019
Get full text
Year of Publication 23.04.2019
Patent
MTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE MTOR/P13K/AKT PATHWAY
MORTENSEN, DEBORAH, PERRIN-NINKOVIC, SOPHIE, ZHAO, JINGJING, SHEVLIN, GRAZIELLA, NARLA, RAMA K, TEHRANI, LIDA, MADAKAMUTIL, LOUI, PACKARD, GARRICK, SAPIENZA, JOHN, PARNES, JASON, XU, WEIMING, SANKAR, SABITA, ELSNER, JAN, HARRIS, ROY L, FULTZ, KIMBERLY, RIGGS, JENNIFER, PAPA, PATRICK, LEE, BRANDEN
Year of Publication 20.03.2018
Get full text
Year of Publication 20.03.2018
Patent
INTERMEDIATES FOR THE SYNTHESIS OF MTOR KINASE INHIBITORS
PAPA, Patrick, SHEVLIN, Graziella I, PACKARD, Garrick, HARRIS, Roy L, LEE, Branden, ZHAO, Jingjing, SAPIENZA, John, MORTENSEN, Deborah, PARNES, Jason, PERRIN-NINKOVIC, Sophie, RIGGS, Jennifer, ELSNER, Jan
Year of Publication 14.12.2016
Get full text
Year of Publication 14.12.2016
Patent
PYRAZINO[2,3-b]PYRAZINE mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY
MORTENSEN Deborah, SAPIENZA John, TEHRANI Lida, PERRIN-NINKOVIC Sophie, HARRIS Roy L, PARNES Jason, ZHAO Jingjing, ELSNER Jan, PAPA Patrick, RIGGS Jennifer, LEE Branden Gingsee, SHEVLIN Graziella I, PACKARD Garrick K
Year of Publication 30.11.2017
Get full text
Year of Publication 30.11.2017
Patent
MTOR kinase inhibitors for oncology indications and diseases associated with the MTOR/P13K/AKT pathway
Sankar, Sabita, Riggs, Jennifer, Sapienza, John, Papa, Patrick, Parnes, Jason, Shevlin, Graziella I, Perrin-Ninkovic, Sophie, Harris, Roy, Elsner, Jan, Tehrani, Lida, Xu, Weiming, Zhao, Jingjing, Fultz, Kimberly Elizabeth, Narla, Rama K, Mortensen, Deborah, Madakamutil, Loui, Lee, Branden, Packard, Garrick K
Year of Publication 25.10.2017
Get full text
Year of Publication 25.10.2017
Patent
MTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE MTOR/P13K/AKT PATHWAY
Sankar, Sabita, Riggs, Jennifer, Sapienza, John, Papa, Patrick, Parnes, Jason, Shevlin, Graziella I, Perrin-Ninkovic, Sophie, Harris, Roy, Elsner, Jan, Tehrani, Lida, Xu, Weiming, Zhao, Jingjing, Fultz, Kimberly Elizabeth, Narla, Rama K, Mortensen, Deborah, Madakamutil, Loui, Lee, Branden, Packard, Garrick K
Year of Publication 06.10.2017
Get full text
Year of Publication 06.10.2017
Patent
MTOR kinase inhibitors for oncology indications and diseases associated with the MTOR/P13K/AKT pathway
Madakamutil Loui, Fultz Kimberly Elizabeth, Mortensen Deborah, Packard Garrick K, Shevlin Graziella I, Zhao Jingjing, Narla Rama K, Perrin-Ninkovic Sophie, Tehrani Lida, Harris Roy, Sankar Sabita, Sapienza John, Parnes Jason, Riggs Jennifer, Elsner Jan, Lee Branden, Papa Patrick, Xu Weiming
Year of Publication 29.09.2017
Get full text
Year of Publication 29.09.2017
Patent
MTOR kinase inhibitors for oncology indications and diseases associated with the MTOR/P13K/AKT pathway
PERRIN-NINKOVIC SOPHIE, ZHAO JINGJING, LEE BRANDEN, SANKAR SABITA, HARRIS ROY, RIGGS JENNIFER, SHEVLIN GRAZIELLA I, NARLA RAMA K, MADAKAMUTIL LOUI, PAPA PATRICK, ELSNER JAN, MORTENSEN DEBORAH, PARNES JASON, XU WEIMING, FULTZ KIMBERLY ELIZABETH, PACKARD GARRICK K, TEHRANI LIDA
Year of Publication 29.09.2017
Get full text
Year of Publication 29.09.2017
Patent
Substituted pyrazino[2,3-b]pyrazines as mTOR kinase inhibitors
Mortensen Deborah, Packard Garrick K, Shevlin Graziella I, Zhao Jingjing, Perrin-Ninkovic Sophie, Tehrani Lida, Parnes Jason, Sapienza John, Riggs Jennifer, Elsner Jan, Harris Roy L, Lee Branden Gingsee, Papa Patrick
Year of Publication 26.09.2017
Get full text
Year of Publication 26.09.2017
Patent
Compuestos y métodos que inhiben eif4e
ERNST, Justin T, URKALAN, Kaveri, SPRENGELER, Paul A, NILEWSKI, Christian, SPERRY, Samuel, TRAN, Chinh Viet, SHAGHAFI, Mike, PACKARD, Garrick Kenneth, XIANG, Alan X, MICHELS, Theo, REICH, Siegfried H, MUKAIYAMA, Takasuke, GRUBBS, Alan
Year of Publication 12.08.2022
Get full text
Year of Publication 12.08.2022
Patent
Eif4a-inhibiting compounds and methods related thereto
MICHELS, THEODORE, ERNST, JUSTIN T, PACKARD, GARRICK KENNETH, REICH, SIEGFRIED H, NILEWSKI, CHRISTIAN, SPRENGELER, PAUL A, XIANG, ALAN XIN, TRAN, CHINH
Year of Publication 01.07.2021
Get full text
Year of Publication 01.07.2021
Patent
MTOR kinase inhibitors for oncology indications and diseases associated with the MTOR/P13K/AKT pathway
Sankar, Sabita, Riggs, Jennifer, Sapienza, John, Papa, Patrick, Parnes, Jason, Shevlin, Graziella I, Perrin-Ninkovic, Sophie, Harris, Roy, Elsner, Jan, Tehrani, Lida, Xu, Weiming, Zhao, Jingjing, Fultz, Kimberly Elizabeth, Narla, Rama K, Mortensen, Deborah, Madakamutil, Loui, Lee, Branden, Packard, Garrick K
Year of Publication 17.05.2017
Get full text
Year of Publication 17.05.2017
Patent
EIF4A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO
ERNST, Justin T, SPRENGELER, Paul A, TRAN, Chinh, NILEWSKI, Christian, REICH, Siegfried H, XIANG, Alan Xin, MICHELS, Theodore, PACKARD, Garrick Kenneth
Year of Publication 19.03.2021
Get full text
Year of Publication 19.03.2021
Patent
MTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE MTOR/P13K/AKT PATHWAY
PAPA, Patrick, HARRIS, Roy, L, MADAKAMUTIL Loui, PACKARD, Garrick, LEE, Branden, TEHRANI, Lida, ZHAO, Jingjing, MORTENSEN, Deborah, SANKAR, Sabita, SAPIENZA, John, SHEVLIN, Graziella, PARNES, Jason, XU, Weiming, FULTZ Kimberly, ELSNER, Jan, PERRIN-NINKOVIC, Sophie, RIGGS, Jennifer, NARLA, Rama K
Year of Publication 18.01.2017
Get full text
Year of Publication 18.01.2017
Patent