Large-amplitude 5-HT1A receptor activation: a new mechanism of profound, central analgesia
Colpaert, F C, Tarayre, J P, Koek, W, Pauwels, P J, Bardin, L, Xu, X-J, Wiesenfeld-Hallin, Z, Cosi, C, Carilla-Durand, E, Assié, M B, Vacher, B
Published in Neuropharmacology (01.11.2002)
Published in Neuropharmacology (01.11.2002)
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In vitro and in vivo receptor binding and effects on monoamine turnover in rat brain regions of the novel antipsychotics risperidone and ocaperidone
LEYSEN, J. E, JANSSEN, P. M. F, GOMMEREN, W, WYNANTS, J, PAUWELS, P. J, JANSSEN, P. A. J
Published in Molecular pharmacology (01.03.1992)
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Published in Molecular pharmacology (01.03.1992)
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Stimulated [35S]GTP gamma S binding by 5-HT1A receptor agonists in recombinant cell lines. Modulation of apparent efficacy by G-protein activation state
Pauwels, P J, Tardif, S, Wurch, T, Colpaert, F C
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.1997)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.1997)
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Sign-reversal during Persistent Activation in μ -Opioid Signal Transduction
BRUINS SLOT, L.A., PAUWELS, P.J., COLPAERT, F.C.
Published in Journal of theoretical biology (21.03.2002)
Published in Journal of theoretical biology (21.03.2002)
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Differentiation between Partial Agonists and Neutral 5-HT1B Antagonists by Chemical Modulation of 3-[3-(N,N-Dimethylamino)propyl]-4-hydroxy- N-[4-(pyridin-4-yl)phenyl]benzamide (GR-55562)
Lamothe, Marie, Pauwels, Petrus J, Belliard, Karine, Schambel, Philippe, Halazy, Serge
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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Neurotoxic action of veratridine in rat brain neuronal cultures: mechanism of neuroprotection by Ca++ antagonists nonselective for slow Ca++ channels
PAUWELS, P. J, VAN ASSOUW, H. P, PEETERS, L, LEYSEN, J. E
Published in The Journal of pharmacology and experimental therapeutics (01.12.1990)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1990)
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Dimerization of sumatriptan as an efficient way to design a potent, centrally and orally active 5-HT1B agonist
PEREZ, M, PAUWELS, P. J, FOURRIER, C, CHOPIN, P, VALENTIN, J.-P, JOHN, G. W, MARIEN, M, HALAZY, S
Published in Bioorganic & medicinal chemistry letters (17.03.1998)
Published in Bioorganic & medicinal chemistry letters (17.03.1998)
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Sequence and Functional Analysis of Cloned Guinea Pig and Rat Serotonin 5‐HT1D Receptors: Common Pharmacological Features Within the 5‐HT1D Receptor Subfamily
Wurch, Thierry, Palmier, Christiane, Colpaert, Francis C., Pauwels, Petrus J.
Published in Journal of neurochemistry (01.01.1997)
Published in Journal of neurochemistry (01.01.1997)
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Design and synthesis of new potent, silent 5-HT1A antagonists by covalent coupling of aminopropanol derivatives with selective serotonin reuptake inhibitors
PEREZ, M, PAUWELS, P. J, PALLARD-SIGOGNEAU, I, FOURRIER, C, CHOPIN, P, PALMIER, C, COLOVRAY, V, HALAZY, S
Published in Bioorganic & medicinal chemistry letters (01.12.1998)
Published in Bioorganic & medicinal chemistry letters (01.12.1998)
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