Mathematical Models in the Description of Pregnane X Receptor (PXR)-Regulated Cytochrome P450 Enzyme Induction
Tebbens, Jurjen Duintjer, Azar, Malek, Friedmann, Elfriede, Lanzendörfer, Martin, Pávek, Petr
Published in International journal of molecular sciences (15.06.2018)
Published in International journal of molecular sciences (15.06.2018)
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Real-time monitoring of Metridia luciferase release from cells upon interaction with model toxic substances by a fully automatic flow setup – A proof of concept
Aguinaga Martínez, Maite V., Jozičová, Natali, Dušek, Jan, Horstkotte, Burkhard, Pávek, Petr, Miró, Manuel, Sklenářová, Hana
Published in Talanta (Oxford) (01.08.2022)
Published in Talanta (Oxford) (01.08.2022)
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2-Substituted quinazolines: Partial agonistic and antagonistic ligands of the constitutive androstane receptor (CAR)
Brožová, Zuzana Rania, Dušek, Jan, Palša, Norbert, Maixnerová, Jana, Kamaraj, Rajamanikkam, Smutná, Lucie, Matouš, Petr, Braeuning, Albert, Pávek, Petr, Kuneš, Jiří, Gathergood, Nicholas, Špulák, Marcel, Pour, Milan, Carazo, Alejandro
Published in European journal of medicinal chemistry (05.11.2023)
Published in European journal of medicinal chemistry (05.11.2023)
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S-substituted 3,5-dinitrophenyl 1,3,4-oxadiazole-2-thiols and tetrazole-5-thiols as highly efficient antitubercular agents
Karabanovich, Galina, Němeček, Jan, Valášková, Lenka, Carazo, Alejandro, Konečná, Klára, Stolaříková, Jiřina, Hrabálek, Alexandr, Pavliš, Oto, Pávek, Petr, Vávrová, Kateřina, Roh, Jaroslav, Klimešová, Věra
Published in European journal of medicinal chemistry (27.01.2017)
Published in European journal of medicinal chemistry (27.01.2017)
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Journal Article
Teriflunomide Is an Indirect Human Constitutive Androstane Receptor (CAR) Activator Interacting With Epidermal Growth Factor (EGF) Signaling
Carazo, Alejandro, Dusek, Jan, Holas, Ondrej, Skoda, Josef, Hyrsova, Lucie, Smutny, Tomas, Soukup, Tomas, Dosedel, Martin, Pávek, Petr
Published in Frontiers in pharmacology (11.10.2018)
Published in Frontiers in pharmacology (11.10.2018)
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Comparison of HepaRG and HepG2 cell lines to model mitochondrial respiratory adaptations in non‑alcoholic fatty liver disease
Maseko, Tumisang Edward, Elkalaf, Moustafa, Peterová, Eva, Lotková, Halka, Staňková, Pavla, Melek, Jan, Dušek, Jan, Žádníková, Petra, Čížková, Dana, Bezrouk, Aleš, Pávek, Petr, Červinková, Zuzana, Kučera, Otto
Published in International journal of molecular medicine (01.02.2024)
Published in International journal of molecular medicine (01.02.2024)
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Development of water-soluble 3,5-dinitrophenyl tetrazole and oxadiazole antitubercular agents
Roh, Jaroslav, Karabanovich, Galina, Vlčková, Hana, Carazo, Alejandro, Němeček, Jan, Sychra, Pavel, Valášková, Lenka, Pavliš, Oto, Stolaříková, Jiřina, Klimešová, Věra, Vávrová, Kateřina, Pávek, Petr, Hrabálek, Alexandr
Published in Bioorganic & medicinal chemistry (15.10.2017)
Published in Bioorganic & medicinal chemistry (15.10.2017)
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Higher Risk of Cardiovascular Diseases in Rheumatoid Arthritis Patients Without Methotrexate Treatment
Hloch, Karel, Doseděl, Martin, Duintjer Tebbens, Jurjen, Žaloudková, Lenka, Medková, Helena, Vlček, Jiří, Soukup, Tomáš, Pávek, Petr
Published in Frontiers in pharmacology (05.11.2021)
Published in Frontiers in pharmacology (05.11.2021)
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Journal Article
The influence of coffee intake and genetics on adenosine pathway in rheumatoid arthritis
Soukup, Tomáš, Hloch, Karel, Doseděl, Martin, Tebbens, Jurjen Duintjer, Nekvindová, Jana, Šembera, Štěpán, Veleta, Tomáš, Pávek, Petr, Barvík, Ivan
Published in Pharmacogenomics (01.07.2020)
Published in Pharmacogenomics (01.07.2020)
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1-Substituted-5-[(3,5-dinitrobenzyl)sulfanyl]-1H-tetrazoles and their isosteric analogs: A new class of selective antitubercular agents active against drug-susceptible and multidrug-resistant mycobacteria
Karabanovich, Galina, Roh, Jaroslav, Smutný, Tomáš, Němeček, Jan, Vicherek, Petr, Stolaříková, Jiřina, Vejsová, Marcela, Dufková, Ida, Vávrová, Kateřina, Pávek, Petr, Klimešová, Věra, Hrabálek, Alexandr
Published in European journal of medicinal chemistry (23.07.2014)
Published in European journal of medicinal chemistry (23.07.2014)
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Novel derivatives of nitro-substituted salicylic acids: Synthesis, antimicrobial activity and cytotoxicity
Paraskevopoulos, Georgios, Krátký, Martin, Mandíková, Jana, Trejtnar, František, Stolaříková, Jiřina, Pávek, Petr, Besra, Gurdyal, Vinšová, Jarmila
Published in Bioorganic & medicinal chemistry (15.11.2015)
Published in Bioorganic & medicinal chemistry (15.11.2015)
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Modulation of xenobiotic conjugation enzymes by dihydromyricetin in rats
Bebová, Michaela, Boštíková, Zdislava, Moserová, Michaela, Pávek, Petr, Anzenbacherová, Eva, Stiborová, Marie, Hodek, Petr
Published in Monatshefte für Chemie (01.11.2017)
Published in Monatshefte für Chemie (01.11.2017)
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Bisamidate Prodrugs of 2-Substituted 9-[2-(Phosphonomethoxy)ethyl]adenine (PMEA, adefovir) as Selective Inhibitors of Adenylate Cyclase Toxin from Bordetella pertussis
Česnek, Michal, Jansa, Petr, Šmídková, Markéta, Mertlíková-Kaiserová, Helena, Dračínský, Martin, Brust, Tarsis F., Pávek, Petr, Trejtnar, František, Watts, Val J., Janeba, Zlatko
Published in ChemMedChem (01.08.2015)
Published in ChemMedChem (01.08.2015)
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In vitro platelet antiaggregatory properties of 4-methylcoumarins
Macáková, Kateřina, Řeháková, Zuzana, Mladěnka, Přemysl, Karlíčková, Jana, Filipský, Tomáš, Říha, Michal, Prasad, Ashok K., Parmar, Virinder S., Jahodář, Luděk, Pávek, Petr, Hrdina, Radomír, Saso, Luciano
Published in Biochimie (01.12.2012)
Published in Biochimie (01.12.2012)
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