Synthesis, molecular modeling, quantum mechanical calculations and ADME estimation studies of benzimidazole-oxadiazole derivatives as potent antifungal agents
Çevik, Ulviye Acar, Celik, Ismail, Işık, Ayşen, Pillai, Renjith Raveendran, Tallei, Trina Ekawati, Yadav, Rohitash, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Journal of molecular structure (15.03.2022)
Published in Journal of molecular structure (15.03.2022)
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Metabolic engineering of Saccharomyces cerevisiae for enhanced taxadiene production
Karaca, Hulya, Kaya, Murat, Kapkac, Handan Açelya, Levent, Serkan, Ozkay, Yusuf, Ozan, Secil Deniz, Nielsen, Jens, Krivoruchko, Anastasia
Published in Microbial cell factories (06.09.2024)
Published in Microbial cell factories (06.09.2024)
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Synthesis and Anticandidal Activity of New Imidazole-Chalcones
Osmaniye, Derya, Kaya Çavuşoğlu, Betül, Sağlık, Begüm Nurpelin, Levent, Serkan, Acar Çevik, Ulviye, Atlı, Özlem, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Molecules (Basel, Switzerland) (04.04.2018)
Published in Molecules (Basel, Switzerland) (04.04.2018)
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Synthesis of New Fluoro-Benzimidazole Derivatives as an Approach towards the Discovery of Novel Intestinal Antiseptic Drug Candidates
Cevik, Ulviye Acar, Saglik, Begum Nurpelin, Ozkay, Yusuf, Canturk, Zerrin, Bueno, Juan, Demirci, Fatih, Koparal, Ali Savas
Published in Current pharmaceutical design (01.01.2017)
Published in Current pharmaceutical design (01.01.2017)
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Novel 1,3,4-thiadiazole compounds as potential MAO-A inhibitors - design, synthesis, biological evaluation and molecular modelling
Sa l k, Begüm Nurpelin, Kaya Çavu o lu, Betül, Acar Çevik, Ulviye, Osmaniye, Derya, Levent, Serkan, Özkay, Yusuf, Kaplanc kl, Zafer As m
Published in MedChemComm (01.09.2020)
Published in MedChemComm (01.09.2020)
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Design, synthesis, molecular modeling, DFT, ADME and biological evaluation studies of some new 1,3,4-oxadiazole linked benzimidazoles as anticancer agents and aromatase inhibitors
Acar Çevik, Ulviye, Celik, Ismail, Işık, Ayşen, Ahmad, Iqrar, Patel, Harun, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Journal of biomolecular structure & dynamics (24.03.2023)
Published in Journal of biomolecular structure & dynamics (24.03.2023)
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Synthesis and biological evaluation of new pyrazolone Schiff bases as monoamine oxidase and cholinesterase inhibitors
Tok, Fatih, Koçyiğit-Kaymakçıoğlu, Bedia, Sağlık, Begüm Nurpelin, Levent, Serkan, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Bioorganic chemistry (01.03.2019)
Published in Bioorganic chemistry (01.03.2019)
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Synthesis, characterization, biological evaluation and in silico studies of novel 1,3,4-thiadiazole derivatives as aromatase inhibitors
Demiraran, Sena, Osmaniye, Derya, Özkay, Yusuf, Kaplancıklı, Zafer Asım, Koçyiğit-Kaymakçıoğlu, Bedia, Tok, Fatih
Published in Journal of molecular structure (15.01.2024)
Published in Journal of molecular structure (15.01.2024)
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Selective in vitro Synergistic Evaluation of Probiotic Tolerant morpholinyl- and 4-ethylpiperazinyl-Imidazole-chalcone Derivatives on Gastrointestinal System Pathogens
Söylemez, Tuncay, Kaplancıklı, Zafer Asım, Osmaniye, Derya, Özkay, Yusuf, Demirci, Fatih
Published in Current microbiology (01.08.2024)
Published in Current microbiology (01.08.2024)
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Design, synthesis, and biological activity of novel dithiocarbamate‐methylsulfonyl hybrids as carbonic anhydrase inhibitors
Osmaniye, Derya, Türkeş, Cüneyt, Demir, Yeliz, Özkay, Yusuf, Beydemir, Şükrü, Kaplancıklı, Zafer A.
Published in Archiv der Pharmazie (Weinheim) (01.08.2022)
Published in Archiv der Pharmazie (Weinheim) (01.08.2022)
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Development and assessment of novel pyrazole–thiadiazol hybrid derivatives as VEGFR-2 inhibitors: design, synthesis, anticancer activity evaluation, molecular docking, and molecular dynamics simulation
Halimi, Gresa, Osmaniye, Derya, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Zeitschrift für Naturforschung C. A journal of biosciences (25.09.2024)
Published in Zeitschrift für Naturforschung C. A journal of biosciences (25.09.2024)
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Design, synthesis, molecular docking and molecular dynamics studies of novel triazolothiadiazine derivatives containing furan or thiophene rings as anticancer agents
Osmaniye, Derya, Karaca, Şevval, Kurban, Berkant, Baysal, Merve, Ahmad, Iqrar, Patel, Harun, Özkay, Yusuf, Asım Kaplancıklı, Zafer
Published in Bioorganic chemistry (01.05.2022)
Published in Bioorganic chemistry (01.05.2022)
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Journal Article
Synthesis, Docking Studies and Biological Activity of New Benzimidazole- Triazolothiadiazine Derivatives as Aromatase Inhibitor
Acar Çevik, Ulviye, Kaya Çavuşoğlu, Betül, Sağlık, Begüm Nurpelin, Osmaniye, Derya, Levent, Serkan, Ilgın, Sinem, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Molecules (Basel, Switzerland) (02.04.2020)
Published in Molecules (Basel, Switzerland) (02.04.2020)
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Design, Synthesis, and Evaluation of Novel 2H-Benzo[b][1,4]thiazin-3(4H)-one Derivatives as New Acetylcholinesterase Inhibitors
Haji Ali, Sazan, Osmaniye, Derya, Sağlık, Begüm Nurpelin, Levent, Serkan, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Molecules (Basel, Switzerland) (25.03.2022)
Published in Molecules (Basel, Switzerland) (25.03.2022)
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Journal Article
Synthesis and Biological Evaluation of New Cholinesterase Inhibitors for Alzheimer's Disease
Hussein, Weiam, Sağlık, Begüm Nurpelin, Levent, Serkan, Korkut, Büşra, Ilgın, Sinem, Özkay, Yusuf, Kaplancıklı, Zafer Asım
Published in Molecules (Basel, Switzerland) (14.08.2018)
Published in Molecules (Basel, Switzerland) (14.08.2018)
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