GPR55: A therapeutic target for Parkinson's disease?
Celorrio, Marta, Rojo-Bustamante, Estefanía, Fernández-Suárez, Diana, Sáez, Elena, Estella-Hermoso de Mendoza, Ander, Müller, Christa E., Ramírez, María J., Oyarzábal, Julen, Franco, Rafael, Aymerich, María S.
Published in Neuropharmacology (01.10.2017)
Published in Neuropharmacology (01.10.2017)
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Published in Hepatology (Baltimore, Md.) (01.06.2021)
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Repurposing ciclopirox as a pharmacological chaperone in a model of congenital erythropoietic porphyria
Urquiza, Pedro, Laín, Ana, Sanz-Parra, Arantza, Moreno, Jorge, Bernardo-Seisdedos, Ganeko, Dubus, Pierre, González, Esperanza, Gutiérrez-de-Juan, Virginia, García, Sandra, Eraña, Hasier, San Juan, Itxaso, Macías, Iratxe, Ben Bdira, Fredj, Pluta, Paula, Ortega, Gabriel, Oyarzábal, Julen, González-Muñiz, Rosario, Rodríguez-Cuesta, Juan, Anguita, Juan, Díez, Emilio, Blouin, Jean-Marc, de Verneuil, Hubert, Mato, José M, Richard, Emmanuel, Falcón-Pérez, Juan M, Castilla, Joaquín, Millet, Oscar
Published in Science translational medicine (19.09.2018)
Published in Science translational medicine (19.09.2018)
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Inhibition of FOXP3/NFAT Interaction Enhances T Cell Function after TCR Stimulation
Lozano, Teresa, Villanueva, Lorea, Durántez, Maika, Gorraiz, Marta, Ruiz, Marta, Belsúe, Virginia, Riezu-Boj, José I, Hervás-Stubbs, Sandra, Oyarzábal, Julen, Bandukwala, Hozefa, Lourenço, Ana R, Coffer, Paul J, Sarobe, Pablo, Prieto, Jesús, Casares, Noelia, Lasarte, Juan J
Published in The Journal of immunology (1950) (01.10.2015)
Published in The Journal of immunology (1950) (01.10.2015)
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Fatty acid amide hydrolase inhibition for the symptomatic relief of Parkinson’s disease
Celorrio, Marta, Fernández-Suárez, Diana, Rojo-Bustamante, Estefanía, Echeverry-Alzate, Víctor, Ramírez, María J, Hillard, Cecilia J, López-Moreno, José A, Maldonado, Rafael, Oyarzábal, Julen, Franco, Rafael, Aymerich, María S
Published in Brain, behavior, and immunity (01.10.2016)
Published in Brain, behavior, and immunity (01.10.2016)
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Information Retrieval and Text Mining Technologies for Chemistry
Krallinger, Martin, Rabal, Obdulia, Lourenço, Anália, Oyarzabal, Julen, Valencia, Alfonso
Published in Chemical reviews (28.06.2017)
Published in Chemical reviews (28.06.2017)
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Cid, Jose María, Duvey, Guillaume, Cluzeau, Philippe, Nhem, Vanthea, Macary, Karim, Raux, Alexandre, Poirier, Nicolas, Muller, Jessica, Boléa, Christelle, Finn, Terry, Poli, Sonia, Epping-Jordan, Mark, Chamelot, Emilie, Derouet, Francis, Girard, Francoise, Macdonald, Gregor J, Vega, Juan Antonio, de Lucas, Ana Isabel, Matesanz, Encarnación, Lavreysen, Hilde, Linares, María Lourdes, Oehlrich, Daniel, Oyarzábal, Julen, Tresadern, Gary, Trabanco, Andrés A, Andrés, Jose Ignacio, Le Poul, Emmanuel, Imogai, Hassan, Lutjens, Robert, Rocher, Jean-Philippe
Published in ACS chemical neuroscience (15.12.2010)
Published in ACS chemical neuroscience (15.12.2010)
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Inhibition of a G9a/DNMT network triggers immune-mediated bladder cancer regression
Segovia, Cristina, San José-Enériz, Edurne, Munera-Maravilla, Ester, Martínez-Fernández, Mónica, Garate, Leire, Miranda, Estíbaliz, Vilas-Zornoza, Amaia, Lodewijk, Iris, Rubio, Carolina, Segrelles, Carmen, Valcárcel, Luis Vitores, Rabal, Obdulia, Casares, Noelia, Bernardini, Alejandra, Suarez-Cabrera, Cristian, López-Calderón, Fernando F, Fortes, Puri, Casado, José A, Dueñas, Marta, Villacampa, Felipe, Lasarte, Juan José, Guerrero-Ramos, Félix, de Velasco, Guillermo, Oyarzabal, Julen, Castellano, Daniel, Agirre, Xabier, Prósper, Felipe, Paramio, Jesús M
Published in Nature medicine (01.07.2019)
Published in Nature medicine (01.07.2019)
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Targeting aberrant DNA methylation in mesenchymal stromal cells as a treatment for myeloma bone disease
Garcia-Gomez, Antonio, Li, Tianlu, de la Calle-Fabregat, Carlos, Rodríguez-Ubreva, Javier, Ciudad, Laura, Català-Moll, Francesc, Godoy-Tena, Gerard, Martín-Sánchez, Montserrat, San-Segundo, Laura, Muntión, Sandra, Morales, Xabier, Ortiz-de-Solórzano, Carlos, Oyarzabal, Julen, San José-Enériz, Edurne, Esteller, Manel, Agirre, Xabier, Prosper, Felipe, Garayoa, Mercedes, Ballestar, Esteban
Published in Nature communications (18.01.2021)
Published in Nature communications (18.01.2021)
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Dual Targeting of Histone Methyltransferase G9a and DNA‐Methyltransferase 1 for the Treatment of Experimental Hepatocellular Carcinoma
Bárcena‐Varela, Marina, Caruso, Stefano, Llerena, Susana, Álvarez‐Sola, Gloria, Uriarte, Iker, Latasa, M. Ujue, Urtasun, Raquel, Rebouissou, Sandra, Alvarez, Laura, Jimenez, Maddalen, Santamaría, Eva, Rodriguez‐Ortigosa, Carlos, Mazza, Giuseppe, Rombouts, Krista, San José‐Eneriz, Edurne, Rabal, Obdulia, Agirre, Xabier, Iraburu, Maria, Santos‐Laso, Alvaro, Banales, Jesus M., Zucman‐Rossi, Jessica, Prósper, Felipe, Oyarzabal, Julen, Berasain, Carmen, Ávila, Matías A., Fernández‐Barrena, Maite G.
Published in Hepatology (Baltimore, Md.) (01.02.2019)
Published in Hepatology (Baltimore, Md.) (01.02.2019)
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Discovery of first-in-class reversible dual small molecule inhibitors against G9a and DNMTs in hematological malignancies
San José-Enériz, Edurne, Agirre, Xabier, Rabal, Obdulia, Vilas-Zornoza, Amaia, Sanchez-Arias, Juan A, Miranda, Estibaliz, Ugarte, Ana, Roa, Sergio, Paiva, Bruno, Estella-Hermoso de Mendoza, Ander, Alvarez, Rosa María, Casares, Noelia, Segura, Victor, Martín-Subero, José I, Ogi, François-Xavier, Soule, Pierre, Santiveri, Clara M, Campos-Olivas, Ramón, Castellano, Giancarlo, de Barrena, Maite Garcia Fernandez, Rodriguez-Madoz, Juan Roberto, García-Barchino, Maria José, Lasarte, Juan Jose, Avila, Matias A, Martinez-Climent, Jose Angel, Oyarzabal, Julen, Prosper, Felipe
Published in Nature communications (26.05.2017)
Published in Nature communications (26.05.2017)
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Binding and Signaling Studies Disclose a Potential Allosteric Site for Cannabidiol in Cannabinoid CB2 Receptors
Martínez-Pinilla, Eva, Varani, Katia, Reyes-Resina, Irene, Angelats, Edgar, Vincenzi, Fabrizio, Ferreiro-Vera, Carlos, Oyarzabal, Julen, Canela, Enric I., Lanciego, José L., Nadal, Xavier, Navarro, Gemma, Borea, Pier Andrea, Franco, Rafael
Published in Frontiers in pharmacology (23.10.2017)
Published in Frontiers in pharmacology (23.10.2017)
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Targeting CB1 and GPR55 Endocannabinoid Receptors as a Potential Neuroprotective Approach for Parkinson’s Disease
Martínez-Pinilla, Eva, Aguinaga, David, Navarro, Gemma, Rico, Alberto J., Oyarzábal, Julen, Sánchez-Arias, Juan A., Lanciego, José Luis, Franco, Rafael
Published in Molecular neurobiology (01.08.2019)
Published in Molecular neurobiology (01.08.2019)
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A novel FTY720 analogue targets SET-PP2A interaction and inhibits growth of acute myeloid leukemia cells without inducing cardiac toxicity
Vicente, Carmen, Arriazu, Elena, Martínez-Balsalobre, Elena, Peris, Irene, Marcotegui, Nerea, García-Ramírez, Patricia, Pippa, Raffaella, Rabal, Obdulia, Oyarzábal, Julen, Guruceaga, Elizabeth, Prósper, Felipe, Mateos, María C., Cayuela, María L., Odero, María D.
Published in Cancer letters (01.01.2020)
Published in Cancer letters (01.01.2020)
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Tadalafil crosses the blood–brain barrier and reverses cognitive dysfunction in a mouse model of AD
García-Barroso, Carolina, Ricobaraza, Ana, Pascual-Lucas, María, Unceta, Nora, Rico, Alberto J., Goicolea, Maria Aranzazu, Sallés, Joan, Lanciego, José Luis, Oyarzabal, Julen, Franco, Rafael, Cuadrado-Tejedor, Mar, García-Osta, Ana
Published in Neuropharmacology (01.01.2013)
Published in Neuropharmacology (01.01.2013)
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Identification of LAG3 high affinity aptamers by HT-SELEX and Conserved Motif Accumulation (CMA)
Soldevilla, Mario Martínez, Hervas, Sandra, Villanueva, Helena, Lozano, Teresa, Rabal, Obdulia, Oyarzabal, Julen, Lasarte, Juan José, Bendandi, Maurizio, Inoges, Susana, López-Díaz de Cerio, Ascensión, Pastor, Fernando
Published in PloS one (21.09.2017)
Published in PloS one (21.09.2017)
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Epigenetic-based differentiation therapy for Acute Myeloid Leukemia
San José-Enériz, Edurne, Gimenez-Camino, Naroa, Rabal, Obdulia, Garate, Leire, Miranda, Estibaliz, Gómez-Echarte, Nahia, García, Fernando, Charalampopoulou, Stella, Sáez, Elena, Vilas-Zornoza, Amaia, San Martín-Uriz, Patxi, Valcárcel, Luis V, Barrena, Naroa, Alignani, Diego, Tamariz-Amador, Luis Esteban, Pérez-Ruiz, Ana, Hilscher, Sebastian, Schutkowski, Mike, Alfonso-Pierola, Ana, Martinez-Calle, Nicolás, Larrayoz, María José, Paiva, Bruno, Calasanz, María José, Muñoz, Javier, Isasa, Marta, Martin-Subero, José Ignacio, Pineda-Lucena, Antonio, Oyarzabal, Julen, Agirre, Xabier, Prósper, Felipe
Published in Nature communications (02.07.2024)
Published in Nature communications (02.07.2024)
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Novel pharmacological maps of protein lysine methyltransferases: key for target deorphanization
Rabal, Obdulia, Castellar, Andrea, Oyarzabal, Julen
Published in Journal of cheminformatics (21.07.2018)
Published in Journal of cheminformatics (21.07.2018)
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