Lignans as Pharmacological Agents in Disorders Related to Oxidative Stress and Inflammation: Chemical Synthesis Approaches and Biological Activities
Osmakov, Dmitry I, Kalinovskii, Aleksandr P, Belozerova, Olga A, Andreev, Yaroslav A, Kozlov, Sergey A
Published in International journal of molecular sciences (27.05.2022)
Published in International journal of molecular sciences (27.05.2022)
Get full text
Journal Article
Opioid Analgesic as a Positive Allosteric Modulator of Acid-Sensing Ion Channels
Osmakov, Dmitry I, Onoprienko, Lyudmila V, Kalinovskii, Aleksandr P, Koshelev, Sergey G, Stepanenko, Vasiliy N, Andreev, Yaroslav A, Kozlov, Sergey A
Published in International journal of molecular sciences (01.02.2024)
Published in International journal of molecular sciences (01.02.2024)
Get full text
Journal Article
Dual Modulator of ASIC Channels and GABAA Receptors from Thyme Alters Fear-Related Hippocampal Activity
Kalinovskii, Aleksandr P., Pushkarev, Anton P., Mikhailenko, Anastasia D., Kudryavtsev, Denis S., Belozerova, Olga A., Shmygarev, Vladimir I., Yatskin, Oleg N., Korolkova, Yuliya V., Kozlov, Sergey A., Osmakov, Dmitry I., Popov, Alexander, Andreev, Yaroslav A.
Published in International journal of molecular sciences (01.09.2023)
Published in International journal of molecular sciences (01.09.2023)
Get full text
Journal Article
Retinoic Acid-Differentiated Neuroblastoma SH-SY5Y Is an Accessible In Vitro Model to Study Native Human Acid-Sensing Ion Channels 1a (ASIC1a)
Kalinovskii, Aleksandr P, Osmakov, Dmitry I, Koshelev, Sergey G, Lubova, Kseniya I, Korolkova, Yuliya V, Kozlov, Sergey A, Andreev, Yaroslav A
Published in Biology (Basel, Switzerland) (20.01.2022)
Published in Biology (Basel, Switzerland) (20.01.2022)
Get full text
Journal Article
Analgesic Activity of Acid-Sensing Ion Channel 3 (ASIС3) Inhibitors: Sea Anemones Peptides Ugr9-1 and APETx2 versus Low Molecular Weight Compounds
Andreev, Yaroslav A, Osmakov, Dmitry I, Koshelev, Sergey G, Maleeva, Ekaterina E, Logashina, Yulia A, Palikov, Victor A, Palikova, Yulia A, Dyachenko, Igor A, Kozlov, Sergey A
Published in Marine drugs (12.12.2018)
Published in Marine drugs (12.12.2018)
Get full text
Journal Article
Anxiolytic, Analgesic and Anti-Inflammatory Effects of Peptides Hmg 1b-2 and Hmg 1b-4 from the Sea Anemone Heteractis magnifica
Gladkikh, Irina N, Klimovich, Anna A, Kalina, Rimma S, Kozhevnikova, Yulia V, Khasanov, Timur A, Osmakov, Dmitry I, Koshelev, Sergey G, Monastyrnaya, Margarita M, Andreev, Yaroslav A, Leychenko, Elena V, Kozlov, Sergey A
Published in Toxins (15.05.2023)
Published in Toxins (15.05.2023)
Get full text
Journal Article
Alkaloid Lindoldhamine Inhibits Acid-Sensing Ion Channel 1a and Reveals Anti-Inflammatory Properties
Osmakov, Dmitry I, Koshelev, Sergey G, Palikov, Victor A, Palikova, Yulia A, Shaykhutdinova, Elvira R, Dyachenko, Igor A, Andreev, Yaroslav A, Kozlov, Sergey A
Published in Toxins (18.09.2019)
Published in Toxins (18.09.2019)
Get full text
Journal Article
Endogenous Isoquinoline Alkaloids Agonists of Acid-Sensing Ion Channel Type 3
Osmakov, Dmitry I, Koshelev, Sergey G, Andreev, Yaroslav A, Kozlov, Sergey A
Published in Frontiers in molecular neuroscience (13.09.2017)
Published in Frontiers in molecular neuroscience (13.09.2017)
Get full text
Journal Article
Multiple Modulation of Acid-Sensing Ion Channel 1a by the Alkaloid Daurisoline
Osmakov, Dmitry I, Koshelev, Sergey G, Lyukmanova, Ekaterina N, Shulepko, Mikhail A, Andreev, Yaroslav A, Illes, Peter, Kozlov, Sergey A
Published in Biomolecules (Basel, Switzerland) (02.08.2019)
Published in Biomolecules (Basel, Switzerland) (02.08.2019)
Get full text
Journal Article
Sevanol and Its Analogues: Chemical Synthesis, Biological Effects and Molecular Docking
Belozerova, Olga A., Osmakov, Dmitry I., Vladimirov, Andrey, Koshelev, Sergey G., Chugunov, Anton O., Andreev, Yaroslav A., Palikov, Victor A., Palikova, Yulia A., Shaykhutdinova, Elvira R., Gvozd, Artem N., Dyachenko, Igor A., Efremov, Roman G., Kublitski, Vadim S., Kozlov, Sergey A.
Published in Pharmaceuticals (Basel, Switzerland) (24.07.2020)
Published in Pharmaceuticals (Basel, Switzerland) (24.07.2020)
Get full text
Journal Article
A Diterpenoid of the Medicinal Plant Andrographis paniculata Targets Cutaneous TRPV3 Channel and Relieves Itch
Kalinovskii, Aleksandr P., Logashina, Yulia A., Palikova, Yulia A., Palikov, Victor A., Osmakov, Dmitry I., Mineev, Konstantin S., Belozerova, Olga A., Shmygarev, Vladimir I., Kozlov, Sergey A., Dyachenko, Igor A., Korolkova, Yuliya V., Andreev, Yaroslav A.
Published in Journal of natural products (Washington, D.C.) (26.07.2024)
Published in Journal of natural products (Washington, D.C.) (26.07.2024)
Get full text
Journal Article
Nocistatin and Products of Its Proteolysis Are Dual Modulators of Type 3 Acid-Sensing Ion Channels (ASIC3) with Algesic and Analgesic Properties
Osmakov, Dmitry I., Tarasova, Nadezhda V., Nedorubov, Andrey A., Palikov, Victor A., Palikova, Yulia A., Dyachenko, Igor A., Andreev, Yaroslav A., Kozlov, Sergey A.
Published in Biochemistry (Moscow) (01.12.2023)
Published in Biochemistry (Moscow) (01.12.2023)
Get full text
Journal Article
Proton‐independent activation of acid‐sensing ion channel 3 by an alkaloid, lindoldhamine, from Laurus nobilis
Osmakov, Dmitry I, Koshelev, Sergey G, Andreev, Yaroslav A, Dubinnyi, Maxim A, Kublitski, Vadim S, Efremov, Roman G, Sobolevsky, Alexander I, Kozlov, Sergey A
Published in British journal of pharmacology (01.03.2018)
Published in British journal of pharmacology (01.03.2018)
Get full text
Journal Article
Sea Anemone Peptide with Uncommon β-Hairpin Structure Inhibits Acid-sensing Ion Channel 3 (ASIC3) and Reveals Analgesic Activity
Osmakov, Dmitry I., Kozlov, Sergey A., Andreev, Yaroslav A., Koshelev, Sergey G., Sanamyan, Nadezhda P., Sanamyan, Karen E., Dyachenko, Igor A., Bondarenko, Dmitry A., Murashev, Arkadii N., Mineev, Konstantin S., Arseniev, Alexander S., Grishin, Eugene V.
Published in The Journal of biological chemistry (09.08.2013)
Published in The Journal of biological chemistry (09.08.2013)
Get full text
Journal Article
Conversed mutagenesis of an inactive peptide to ASIC3 inhibitor for active sites determination
Osmakov, Dmitry I., Koshelev, Sergey G., Andreev, Yaroslav A., Dyachenko, Igor A., Bondarenko, Dmitry A., Murashev, Arkadii N., Grishin, Eugene V., Kozlov, Sergey A.
Published in Toxicon (Oxford) (15.06.2016)
Published in Toxicon (Oxford) (15.06.2016)
Get full text
Journal Article
Lignan from Thyme Possesses Inhibitory Effect on ASIC3 Channel Current
Dubinnyi, Maxim A., Osmakov, Dmitry I., Koshelev, Sergey G., Kozlov, Sergey A., Andreev, Yaroslav A., Zakaryan, Naira A., Dyachenko, Igor A., Bondarenko, Dmitry A., Arseniev, Alexander S., Grishin, Eugene V.
Published in The Journal of biological chemistry (21.09.2012)
Published in The Journal of biological chemistry (21.09.2012)
Get full text
Journal Article
Dual Modulator of ASIC Channels and GABA[sub.A] Receptors from Thyme Alters Fear-Related Hippocampal Activity
Kalinovskii, Aleksandr P, Pushkarev, Anton P, Mikhailenko, Anastasia D, Kudryavtsev, Denis S, Belozerova, Olga A, Shmygarev, Vladimir I, Yatskin, Oleg N, Korolkova, Yuliya V, Kozlov, Sergey A, Osmakov, Dmitry I, Popov, Alexander, Andreev, Yaroslav A
Published in International journal of molecular sciences (01.08.2023)
Published in International journal of molecular sciences (01.08.2023)
Get full text
Journal Article