A new class of non-C2-symmetric ligands for oxidative and redox-neutral palladium-catalyzed asymmetric allylic alkylations of 1,3-diketones
Trost, Barry M, Donckele, Etienne J, Thaisrivongs, David A, Osipov, Maksim, Masters, James T
Published in Journal of the American Chemical Society (25.02.2015)
Published in Journal of the American Chemical Society (25.02.2015)
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Journal Article
Acetoxy Meldrum’s Acid: A Versatile Acyl Anion Equivalent in the Pd-Catalyzed Asymmetric Allylic Alkylation
Trost, Barry M, Osipov, Maksim, Kaib, Philip S. J, Sorum, Mark T
Published in Organic letters (17.06.2011)
Published in Organic letters (17.06.2011)
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Journal Article
Palladium-Catalyzed Dynamic Kinetic Asymmetric Transformations of Vinyl Aziridines with Nitrogen Heterocycles: Rapid Access to Biologically Active Pyrroles and Indoles
Trost, Barry M, Osipov, Maksim, Dong, Guangbin
Published in Journal of the American Chemical Society (10.11.2010)
Published in Journal of the American Chemical Society (10.11.2010)
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Journal Article
Synthesis of deep-cavity fluorous calix[4]arenes as molecular recognition scaffolds
Osipov, Maksim, Chu, Qianli, Geib, Steven J, Curran, Dennis P, Weber, Stephen G
Published in Beilstein journal of organic chemistry (20.10.2008)
Published in Beilstein journal of organic chemistry (20.10.2008)
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Journal Article
A New Class of Non‑C 2‑Symmetric Ligands for Oxidative and Redox-Neutral Palladium-Catalyzed Asymmetric Allylic Alkylations of 1,3-Diketones
Trost, Barry M, Donckele, Etienne J, Thaisrivongs, David A, Osipov, Maksim, Masters, James T
Published in Journal of the American Chemical Society (25.02.2015)
Published in Journal of the American Chemical Society (25.02.2015)
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Journal Article
Discovery of Potent, Selective, and Orally Bioavailable Inhibitors of USP7 with In Vivo Antitumor Activity
Leger, Paul R, Hu, Dennis X, Biannic, Berenger, Bui, Minna, Han, Xinping, Karbarz, Emily, Maung, Jack, Okano, Akinori, Osipov, Maksim, Shibuya, Grant M, Young, Kyle, Higgs, Christopher, Abraham, Betty, Bradford, Delia, Cho, Cynthia, Colas, Christophe, Jacobson, Scott, Ohol, Yamini M, Pookot, Deepa, Rana, Payal, Sanchez, Jerick, Shah, Niket, Sun, Michael, Wong, Steve, Brockstedt, Dirk G, Kassner, Paul D, Schwarz, Jacob B, Wustrow, David J
Published in Journal of medicinal chemistry (28.05.2020)
Published in Journal of medicinal chemistry (28.05.2020)
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Discovery of DNL343: A Potent, Selective, and Brain-Penetrant eIF2B Activator Designed for the Treatment of Neurodegenerative Diseases
Craig, Robert A., De Vicente, Javier, Estrada, Anthony A., Feng, Jianwen A., Lexa, Katrina W., Canet, Mark J., Dowdle, William E., Erickson, Rebecca I., Flores, Brittany N., Haddick, Patrick C. G., Kane, Lesley A., Lewcock, Joseph W., Moerke, Nathan J., Poda, Suresh B., Sweeney, Zachary, Takahashi, Ryan H., Tong, Vincent, Wang, Jing, Yulyaningsih, Ernie, Solanoy, Hilda, Scearce-Levie, Kimberly, Sanchez, Pascal E., Tang, Liwei, Xu, Musheng, Zhang, Rui, Osipov, Maksim
Published in Journal of medicinal chemistry (11.04.2024)
Published in Journal of medicinal chemistry (11.04.2024)
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Discovery of Potent and Selective Dual Leucine Zipper Kinase/Leucine Zipper-Bearing Kinase Inhibitors with Neuroprotective Properties in In Vitro and In Vivo Models of Amyotrophic Lateral Sclerosis
Craig, Robert A., Fox, Brian M., Hu, Cheng, Lexa, Katrina W., Osipov, Maksim, Thottumkara, Arun P., Larhammar, Martin, Miyamoto, Takashi, Rana, Anil, Kane, Lesley A., Yulyaningsih, Ernie, Solanoy, Hilda, Nguyen, Hoang, Chau, Roni, Earr, Timothy, Kajiwara, Yuji, Fleck, Daniel, Lucas, Anthony, Haddick, Patrick C. G., Takahashi, Ryan H., Tong, Vincent, Wang, Jing, Canet, Mark J., Poda, Suresh B., Scearce-Levie, Kimberly, Srivastava, Ankita, Sweeney, Zachary K., Xu, Musheng, Zhang, Rui, He, Jianrong, Lei, Yanan, Zhuo, Zheng, de Vicente, Javier
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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DNL343 is an investigational CNS penetrant eukaryotic initiation factor 2B activator that prevents and reverses the effects of neurodegeneration caused by the integrated stress response
Yulyaningsih, Ernie, Suh, Jung H, Fanok, Melania, Chau, Roni, Solanoy, Hilda, Takahashi, Ryan, Bakardjiev, Anna I, Becerra, Isabel, Benitez, N Butch, Chiu, Chi-Lu, Davis, Sonnet S, Dowdle, William E, Earr, Timothy, Estrada, Anthony A, Gill, Audrey, Ha, Connie, Haddick, Patrick CG, Henne, Kirk R, Larhammar, Martin, Leung, Amy W-S, Maciuca, Romeo, Memarzadeh, Bahram, Nguyen, Hoang N, Nugent, Alicia A, Osipov, Maksim, Ran, Yingqing, Rebadulla, Kevin, Roche, Elysia, Sandman, Thomas, Wang, Jing, Lewcock, Joseph W, Scearce-Levie, Kimberly, Kane, Lesley A, Sanchez, Pascal E
Published in eLife (17.09.2024)
Published in eLife (17.09.2024)
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화합물, 조성물 및 방법
CRAIG II ROBERT A, HU CHENG, OSIPOV MAKSIM, ESTRADA ANTHONY A, THOTTUMKARA ARUN, BUCHER CYRIL, FOX BRIAN M, DE VICENTE FIDALGO JAVIER, NILEWSKI LIZANNE G, BAGDASARIAN ALEX L, HUFFMAN BENJAMIN J, LEXA KATRINA W
Year of Publication 23.08.2023
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Year of Publication 23.08.2023
Patent
화합물, 조성물 및 방법
CRAIG II ROBERT A, HU CHENG, OSIPOV MAKSIM, ESTRADA ANTHONY A, THOTTUMKARA ARUN, FOX BRIAN M, DE VICENTE FIDALGO JAVIER, NILEWSKI LIZANNE G, BAGDASARIAN ALEX L, HUFFMAN BENJAMIN J, LEXA KATRINA W
Year of Publication 18.04.2023
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Year of Publication 18.04.2023
Patent
화합물, 조성물 및 방법
CRAIG II ROBERT A, HU CHENG, OSIPOV MAKSIM, ESTRADA ANTHONY A, THOTTUMKARA ARUN, FOX BRIAN M, DE VICENTE FIDALGO JAVIER, NILEWSKI LIZANNE G, LEXA KATRINA W
Year of Publication 10.03.2023
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Year of Publication 10.03.2023
Patent
화합물, 조성물 및 방법
OSIPOV MAKSIM, CRAIG ROBERT A. II, ESTRADA ANTHONY A, THOTTUMKARA ARUN, FOX BRIAN M, DE VICENTE FIDALGO JAVIER, FENG JIANWEN A
Year of Publication 19.10.2021
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Year of Publication 19.10.2021
Patent
Abstract 4290: Potent and selective next generation inhibitors of indoleamine-2,3-dioxygenase (IDO1) for the treatment of cancer
Powers, Jay P., Walters, Matthew J., Noubade, Rajkumar, Young, Stephen W., Marshall, Lisa, Melom, Jan, Park, Adam, Shah, Nick, Bjork, Pia, Fridman, Jordan S., Beck, Hilary P., Chian, David, McKinnell, Jenny V., Osipov, Maksim, Reilly, Maureen K., Shunatona, Hunter P., Walker, James R., Zibinsky, Mikhail, Jaen, Juan C.
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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