QSAR without borders
Muratov, Eugene N, Bajorath, Jürgen, Sheridan, Robert P, Tetko, Igor V, Filimonov, Dmitry, Poroikov, Vladimir, Oprea, Tudor I, Baskin, Igor I, Varnek, Alexandre, Roitberg, Adrian, Isayev, Olexandr, Curtalolo, Stefano, Fourches, Denis, Cohen, Yoram, Aspuru-Guzik, Alan, Winkler, David A, Agrafiotis, Dimitris, Cherkasov, Artem, Tropsha, Alexander
Published in Chemical Society reviews (07.06.2020)
Published in Chemical Society reviews (07.06.2020)
Get full text
Journal Article
Therapies for rare diseases: therapeutic modalities, progress and challenges ahead
Tambuyzer, Erik, Vandendriessche, Benjamin, Austin, Christopher P., Brooks, Philip J., Larsson, Kristina, Miller Needleman, Katherine I., Valentine, James, Davies, Kay, Groft, Stephen C., Preti, Robert, Oprea, Tudor I., Prunotto, Marco
Published in Nature reviews. Drug discovery (01.02.2020)
Published in Nature reviews. Drug discovery (01.02.2020)
Get full text
Journal Article
The significance of acid/base properties in drug discovery
Manallack, David T, Prankerd, Richard J, Yuriev, Elizabeth, Oprea, Tudor I, Chalmers, David K
Published in Chemical Society reviews (21.01.2013)
Published in Chemical Society reviews (21.01.2013)
Get full text
Journal Article
TCRD and Pharos 2021: mining the human proteome for disease biology
Sheils, Timothy K, Mathias, Stephen L, Kelleher, Keith J, Siramshetty, Vishal B, Nguyen, Dac-Trung, Bologa, Cristian G, Jensen, Lars Juhl, Vidović, Dušica, Koleti, Amar, Schürer, Stephan C, Waller, Anna, Yang, Jeremy J, Holmes, Jayme, Bocci, Giovanni, Southall, Noel, Dharkar, Poorva, Mathé, Ewy, Simeonov, Anton, Oprea, Tudor I
Published in Nucleic Acids Research (08.01.2021)
Published in Nucleic Acids Research (08.01.2021)
Get full text
Journal Article
Web Resource
Pharos: Collating protein information to shed light on the druggable genome
Nguyen, Dac-Trung, Mathias, Stephen, Bologa, Cristian, Brunak, Soren, Fernandez, Nicolas, Gaulton, Anna, Hersey, Anne, Holmes, Jayme, Jensen, Lars Juhl, Karlsson, Anneli, Liu, Guixia, Ma'ayan, Avi, Mandava, Geetha, Mani, Subramani, Mehta, Saurabh, Overington, John, Patel, Juhee, Rouillard, Andrew D, Schürer, Stephan, Sheils, Timothy, Simeonov, Anton, Sklar, Larry A, Southall, Noel, Ursu, Oleg, Vidovic, Dusica, Waller, Anna, Yang, Jeremy, Jadhav, Ajit, Oprea, Tudor I, Guha, Rajarshi
Published in Nucleic acids research (04.01.2017)
Published in Nucleic acids research (04.01.2017)
Get full text
Journal Article
DrugCentral 2023 extends human clinical data and integrates veterinary drugs
Avram, Sorin, Wilson, Thomas B, Curpan, Ramona, Halip, Liliana, Borota, Ana, Bora, Alina, Bologa, Cristian G, Holmes, Jayme, Knockel, Jeffrey, Yang, Jeremy J, Oprea, Tudor I
Published in Nucleic acids research (06.01.2023)
Published in Nucleic acids research (06.01.2023)
Get full text
Journal Article
Pharos 2023: an integrated resource for the understudied human proteome
Kelleher, Keith J, Sheils, Timothy K, Mathias, Stephen L, Yang, Jeremy J, Metzger, Vincent T, Siramshetty, Vishal B, Nguyen, Dac-Trung, Jensen, Lars Juhl, Vidović, Dušica, Schürer, Stephan C, Holmes, Jayme, Sharma, Karlie R, Pillai, Ajay, Bologa, Cristian G, Edwards, Jeremy S, Mathé, Ewy A, Oprea, Tudor I
Published in Nucleic acids research (06.01.2023)
Published in Nucleic acids research (06.01.2023)
Get full text
Journal Article
QSAR Modeling of the Blood–Brain Barrier Permeability for Diverse Organic Compounds
Zhang, Liying, Zhu, Hao, Oprea, Tudor I., Golbraikh, Alexander, Tropsha, Alexander
Published in Pharmaceutical research (01.08.2008)
Published in Pharmaceutical research (01.08.2008)
Get full text
Journal Article
Distribution and characterization of estrogen receptor G protein-coupled receptor 30 in the rat central nervous system
Brailoiu, Eugen, Dun, Siok L, Brailoiu, G Cristina, Mizuo, Keisuke, Sklar, Larry A, Oprea, Tudor I, Prossnitz, Eric R, Dun, Nae J
Published in Journal of endocrinology (01.05.2007)
Published in Journal of endocrinology (01.05.2007)
Get full text
Journal Article
GLUT3 inhibitor discovery through in silico ligand screening and in vivo validation in eukaryotic expression systems
Iancu, Cristina V., Bocci, Giovanni, Ishtikhar, Mohd, Khamrai, Moumita, Oreb, Mislav, Oprea, Tudor I., Choe, Jun-yong
Published in Scientific reports (26.01.2022)
Published in Scientific reports (26.01.2022)
Get full text
Journal Article
Microbial efflux pump inhibition: tactics and strategies
Tegos, George P, Haynes, Mark, Strouse, J Jacob, Khan, Mohiuddin Md T, Bologa, Cristian G, Oprea, Tudor I, Sklar, Larry A
Published in Current pharmaceutical design (01.05.2011)
Published in Current pharmaceutical design (01.05.2011)
Get more information
Journal Article
The G Protein-Coupled Receptor GPR30 Inhibits Proliferation of Estrogen Receptor-Positive Breast Cancer Cells
ARIAZI, Eric A, BRAILOIU, Eugen, PROSSNITZ, Eric R, DUN, Nae J, JORDAN, V. Craig, YERRUM, Smitha, SHUPP, Heather A, SLIFKER, Michael J, CUNLIFFE, Heather E, BLACK, Michael A, DONATO, Anne L, ARTERBURN, Jeffrey B, OPREA, Tudor I
Published in Cancer research (Chicago, Ill.) (01.02.2010)
Published in Cancer research (Chicago, Ill.) (01.02.2010)
Get full text
Journal Article
A machine learning platform to estimate anti-SARS-CoV-2 activities
KC, Govinda B., Bocci, Giovanni, Verma, Srijan, Hassan, Md Mahmudulla, Holmes, Jayme, Yang, Jeremy J., Sirimulla, Suman, Oprea, Tudor I.
Published in Nature machine intelligence (01.06.2021)
Published in Nature machine intelligence (01.06.2021)
Get full text
Journal Article
Modulation of Bitter Taste Perception by a Small Molecule hTAS2R Antagonist
Slack, Jay P., Brockhoff, Anne, Batram, Claudia, Menzel, Susann, Sonnabend, Caroline, Born, Stephan, Galindo, Maria Mercedes, Kohl, Susann, Thalmann, Sophie, Ostopovici-Halip, Liliana, Simons, Christopher T., Ungureanu, Ioana, Duineveld, Kees, Bologa, Cristian G., Behrens, Maik, Furrer, Stefan, Oprea, Tudor I., Meyerhof, Wolfgang
Published in Current biology (22.06.2010)
Published in Current biology (22.06.2010)
Get full text
Journal Article