Synthesis and multiparametric evaluation of thiadiazoles and oxadiazoles as diacylglycerol acyltransferase type 1 inhibitors
Mougenot, Patrick, Namane, Claudie, Fett, Eykmar, Goumy, Florence, Dadji-Faïhun, Rommel, Langot, Gwladys, Monseau, Catherine, Onofri, Bénédicte, Pacquet, François, Pascal, Cécile, Crespin, Olivier, Ben-Hassine, Majdi, Ragot, Jean-Luc, Van-Pham, Thao, Philippo, Christophe, Chatelain-Egger, Florence, Péron, Philippe, Le Bail, Jean-Christophe, Guillot, Etienne, Chamiot-Clerc, Philippe, Chabanaud, Marie-Aude, Pruniaux, Marie-Pierre, Ménegotto, Jérôme, Schmidt, Friedemann, Venier, Olivier, Viviani, Fabrice, Nicolai, Eric
Published in Bioorganic & medicinal chemistry letters (01.01.2016)
Published in Bioorganic & medicinal chemistry letters (01.01.2016)
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Thiadiazoles as new inhibitors of diacylglycerol acyltransferase type 1
Mougenot, Patrick, Namane, Claudie, Fett, Eykmar, Camy, Florence, Dadji-Faïhun, Rommel, Langot, Gwladys, Monseau, Catherine, Onofri, Bénédicte, Pacquet, François, Pascal, Cécile, Crespin, Olivier, Ben-Hassine, Majdi, Ragot, Jean-Luc, Van-Pham, Thao, Philippo, Christophe, Chatelain-Egger, Florence, Péron, Philippe, Le Bail, Jean-Christophe, Guillot, Etienne, Chamiot-Clerc, Philippe, Chabanaud, Marie-Aude, Pruniaux, Marie-Pierre, Schmidt, Friedemann, Venier, Olivier, Nicolaï, Eric, Viviani, Fabrice
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Discovery of SAR184841, a potent and long-lasting inhibitor of 11β-hydroxysteroid dehydrogenase type 1, active in a physiopathological animal model of T2D
Venier, Olivier, Pascal, Cécile, Braun, Alain, Namane, Claudie, Mougenot, Patrick, Crespin, Olivier, Pacquet, François, Mougenot, Cécile, Monseau, Catherine, Onofri, Bénédicte, Dadji-Faïhun, Rommel, Leger, Céline, Ben-Hassine, Majdi, Van-Pham, Thao, Ragot, Jean-Luc, Philippo, Christophe, Farjot, Géraldine, Noah, Lionel, Maniani, Karima, Boutarfa, Asma, Nicolaï, Eric, Guillot, Etienne, Pruniaux, Marie-Pierre, Güssregen, Stefan, Engel, Christian, Coutant, Anne-Laure, de Miguel, Beatriz, Castro, Antonio
Published in Bioorganic & medicinal chemistry letters (15.04.2013)
Published in Bioorganic & medicinal chemistry letters (15.04.2013)
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Journal Article
Pyrrolidine-pyrazole ureas as potent and selective inhibitors of 11β-hydroxysteroid-dehydrogenase type 1
Venier, Olivier, Pascal, Cécile, Braun, Alain, Namane, Claudie, Mougenot, Patrick, Crespin, Olivier, Pacquet, François, Mougenot, Cécile, Monseau, Catherine, Onofri, Bénédicte, Dadji-Faïhun, Rommel, Leger, Céline, Ben-Hassine, Majdi, Van-Pham, Thao, Ragot, Jean-Luc, Philippo, Christophe, Güssregen, Stefan, Engel, Christian, Farjot, Géraldine, Noah, Lionel, Maniani, Karima, Nicolaï, Eric
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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Journal Article
Discovery of SAR184841, a potent and long-lasting inhibitor of 11[beta]-hydroxysteroid dehydrogenase type 1, active in a physiopathological animal model of T2D
Venier, Olivier, Pascal, Cecile, Braun, Alain, Namane, Claudie, Mougenot, Patrick, Crespin, Olivier, Pacquet, Francois, Mougenot, Cecile, Monseau, Catherine, Onofri, Benedicte, Dadji-Faiehun, Rommel, Leger, Celine, Ben-Hassine, Majdi, Van-Pham, Thao, Ragot, Jean-Luc, Philippo, Christophe, Farjot, Geraldine, Noah, Lionel, Maniani, Karima, Boutarfa, Asma, Nicolaie, Eric, Guillot, Etienne, Pruniaux, Marie-Pierre, Guessregen, Stefan, Engel, Christian, Coutant, Anne-Laure, de Miguel, Beatriz, Castro, Antonio
Published in Bioorganic & medicinal chemistry letters (15.04.2013)
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Published in Bioorganic & medicinal chemistry letters (15.04.2013)
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