Visible‐Light‐Mediated Metal‐Free Difunctionalization of Alkenes with CO2 and Silanes or C(sp3)−H Alkanes
Hou, Jing, Ee, Aloysius, Cao, Hui, Ong, Han‐Wee, Xu, Jin‐Hui, Wu, Jie
Published in Angewandte Chemie International Edition (21.12.2018)
Published in Angewandte Chemie International Edition (21.12.2018)
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Journal Article
Strategic Fluorination to Achieve a Potent, Selective, Metabolically Stable, and Orally Bioavailable Inhibitor of CSNK2
Ong, Han Wee, Yang, Xuan, Smith, Jeffery L., Taft-Benz, Sharon, Howell, Stefanie, Dickmander, Rebekah J., Havener, Tammy M., Sanders, Marcia K., Brown, Jason W., Couñago, Rafael M., Chang, Edcon, Krämer, Andreas, Moorman, Nathaniel J., Heise, Mark, Axtman, Alison D., Drewry, David H., Willson, Timothy M.
Published in Molecules (Basel, Switzerland) (02.09.2024)
Published in Molecules (Basel, Switzerland) (02.09.2024)
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Discovery and characterization of a specific inhibitor of serine-threonine kinase cyclin-dependent kinase-like 5 (CDKL5) demonstrates role in hippocampal CA1 physiology
Castano, Anna, Silvestre, Margaux, Wells, Carrow I, Sanderson, Jennifer L, Ferrer, Carla A, Ong, Han Wee, Lang, Yi, Richardson, William, Silvaroli, Josie A, Bashore, Frances M, Smith, Jeffery L, Genereux, Isabelle M, Dempster, Kelvin, Drewry, David H, Pabla, Navlot S, Bullock, Alex N, Benke, Tim A, Ultanir, Sila K, Axtman, Alison D
Published in eLife (25.07.2023)
Published in eLife (25.07.2023)
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Journal Article
Optimization of 3‑Cyano-7-cyclopropylamino-pyrazolo[1,5‑a]pyrimidines toward the Development of an In Vivo Chemical Probe for CSNK2A
Yang, Xuan, Ong, Han Wee, Dickmander, Rebekah J., Smith, Jeffery L., Brown, Jason W., Tao, William, Chang, Edcon, Moorman, Nathaniel J., Axtman, Alison D., Willson, Timothy M.
Published in ACS omega (24.10.2023)
Published in ACS omega (24.10.2023)
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Journal Article
Visible‐Light‐Induced Selective Defluoroborylation of Polyfluoroarenes, gem‐Difluoroalkenes, and Trifluoromethylalkenes
Xu, Wengang, Jiang, Heming, Leng, Jing, Ong, Han‐Wee, Wu, Jie
Published in Angewandte Chemie (02.03.2020)
Published in Angewandte Chemie (02.03.2020)
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Journal Article
Visible‐Light‐Mediated Metal‐Free Difunctionalization of Alkenes with CO2 and Silanes or C(sp3)−H Alkanes
Hou, Jing, Ee, Aloysius, Cao, Hui, Ong, Han‐Wee, Xu, Jin‐Hui, Wu, Jie
Published in Angewandte Chemie (21.12.2018)
Published in Angewandte Chemie (21.12.2018)
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Journal Article
A Potent and Selective CDKL5/GSK3 Chemical Probe is Neuroprotective
Han Wee Ong, Liang, Yi, Richardson, William, Lowry, Emily R, Wells, Carrow I, Chen, Xiangrong, Silvestre, Margaux, Dempster, Kelvin, Silvaroli, Josie A, Smith, Jeffery L, Wichterle, Hynek, Pabla, Navjot S, Ultanir, Sila K, Bullock, Alex N, Drewry, David, Alison Donnelly Axtman
Published in bioRxiv (10.02.2023)
Published in bioRxiv (10.02.2023)
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Journal Article
How many kinases are druggable? A review of our current understanding
Anderson, Brian, Rosston, Peter, Ong, Han Wee, Hossain, Mohammad Anwar, Davis-Gilbert, Zachary W, Drewry, David H
Published in Biochemical journal (30.08.2023)
Published in Biochemical journal (30.08.2023)
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Journal Article
Parasite and host kinases as targets for antimalarials
Ong, Han Wee, Adderley, Jack, Tobin, Andrew B., Drewry, David H., Doerig, Christian
Published in Expert opinion on therapeutic targets (01.02.2023)
Published in Expert opinion on therapeutic targets (01.02.2023)
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Journal Article
CK2 Chemical Probes: Past, Present, and Future
Ong, Han Wee, Drewry, David H., Axtman, Alison D.
Published in Kinases and Phosphatases (01.11.2023)
Published in Kinases and Phosphatases (01.11.2023)
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Journal Article
More than an Amide Bioisostere: Discovery of 1,2,4-Triazole-containing Pyrazolo1,5-apyrimidine Host CSNK2 Inhibitors for Combatting β-Coronavirus Replication
Ong, Han Wee, Yang, Xuan, Smith, Jeffery L, Dickmander, Rebekah J, Brown, Jason W, Havener, Tammy M, Taft-Benz, Sharon, Howell, Stefanie, Sanders, Marcia K, Capener, Jacob L, Couñago, Rafael M, Chang, Edcon, Krämer, Andreas, Moorman, Nathaniel J, Heise, Mark, Axtman, Alison D, Drewry, David H, Willson, Timothy M
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Journal Article
More than an Amide Bioisostere: Discovery of 1,2,4-Triazole-containing Pyrazolo[1,5‑a]pyrimidine Host CSNK2 Inhibitors for Combatting β‑Coronavirus Replication
Ong, Han Wee, Yang, Xuan, Smith, Jeffery L., Dickmander, Rebekah J., Brown, Jason W., Havener, Tammy M., Taft-Benz, Sharon, Howell, Stefanie, Sanders, Marcia K., Capener, Jacob L., Couñago, Rafael M., Chang, Edcon, Krämer, Andreas, Moorman, Nathaniel J., Heise, Mark, Axtman, Alison D., Drewry, David H., Willson, Timothy M.
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Journal Article
Identification of Novel 2,4,5-Trisubstituted Pyrimidines as Potent Dual Inhibitors of Plasmodial Pf GSK3/ Pf PK6 with Activity against Blood Stage Parasites In Vitro
Galal, Kareem A., Truong, Anna, Kwarcinski, Frank, de Silva, Chandi, Avalani, Krisha, Havener, Tammy M., Chirgwin, Michael E., Merten, Eric, Ong, Han Wee, Willis, Caleb, Abdelwaly, Ahmad, Helal, Mohamed A., Derbyshire, Emily R., Zutshi, Reena, Drewry, David H.
Published in Journal of medicinal chemistry (13.10.2022)
Published in Journal of medicinal chemistry (13.10.2022)
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Journal Article
Discovery of potent Plasmodium falciparum protein kinase 6 (PfPK6) inhibitors with a type II inhibitor pharmacophore
Ong, Han Wee, Truong, Anna, Kwarcinski, Frank, de Silva, Chandi, Avalani, Krisha, Havener, Tammy M., Chirgwin, Michael, Galal, Kareem A., Willis, Caleb, Krämer, Andreas, Liu, Shubin, Knapp, Stefan, Derbyshire, Emily R., Zutshi, Reena, Drewry, David H.
Published in European journal of medicinal chemistry (05.03.2023)
Published in European journal of medicinal chemistry (05.03.2023)
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Journal Article
Identification of Novel 2,4,5-Trisubstituted Pyrimidines as Potent Dual Inhibitors of Plasmodial PfGSK3/PfPK6 with Activity against Blood Stage Parasites In Vitro
Galal, Kareem A., Truong, Anna, Kwarcinski, Frank, de Silva, Chandi, Avalani, Krisha, Havener, Tammy M., Chirgwin, Michael E., Merten, Eric, Ong, Han Wee, Willis, Caleb, Abdelwaly, Ahmad, Helal, Mohamed A., Derbyshire, Emily R., Zutshi, Reena, Drewry, David H.
Published in Journal of medicinal chemistry (13.10.2022)
Published in Journal of medicinal chemistry (13.10.2022)
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Journal Article
PROTAC Linkerology Leads to an Optimized Bivalent Chemical Degrader of Polycomb Repressive Complex 2 (PRC2) Components
Bashore, Frances M., Foley, Caroline A., Ong, Han Wee, Rectenwald, Justin M., Hanley, Ronan P., Norris-Drouin, Jacqueline L., Cholensky, Stephanie H., Mills, Christine A., Pearce, Kenneth H., Herring, Laura E., Kireev, Dmitri, Frye, Stephen V., James, Lindsey I.
Published in ACS chemical biology (17.03.2023)
Published in ACS chemical biology (17.03.2023)
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Journal Article
Characterization of 2,4-Dianilinopyrimidines Against Five P. falciparum Kinases PfARK1, PfARK3, PfNEK3, PfPK9, and PfPKB
Ong, Han Wee, de Silva, Chandi, Avalani, Krisha, Kwarcinski, Frank, Mansfield, Christopher R., Chirgwin, Michael, Truong, Anna, Derbyshire, Emily R., Zutshi, Reena, Drewry, David H.
Published in ACS medicinal chemistry letters (14.12.2023)
Published in ACS medicinal chemistry letters (14.12.2023)
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Journal Article
Coordination of the Hemilabile Ligand Diphenylvinylphosphine to Ru4(µ-H)4(CO)12: Synthesis, Stability and Structural Studies
Neo, Ren Kai Edward, Ong, Han Wee, Wong, Zhen Xuan, Kumaran, Elumalai, Ganguly, Rakesh, Leong, Weng Kee, Tan, Yong Leng Kelvin
Published in Journal of cluster science (01.09.2022)
Published in Journal of cluster science (01.09.2022)
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