Synthesis and evaluation of diphenylphosphinic amides and diphenylphosphine oxides as inhibitors of Kv1.5
Olsson, Roine I., Jacobson, Ingemar, Boström, Jonas, Fex, Tomas, Björe, Annika, Olsson, Christina, Sundell, Johan, Gran, Ulrik, Öhrn, Anna, Nordin, Andreas, Gyll, Jonna, Thorstensson, Maria, Hayen, Ahlke, Aplander, Karolina, Hidestål, Olle, Jiang, Fanyi, Linhardt, Gunilla, Forsström, Elin, Collins, Teresa, Sundqvist, Monika, Lindhardt, Emma, Åstrand, Annika, Löfberg, Boel
Published in Bioorganic & medicinal chemistry letters (01.02.2013)
Published in Bioorganic & medicinal chemistry letters (01.02.2013)
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AZD0284, a Potent, Selective, and Orally Bioavailable Inverse Agonist of Retinoic Acid Receptor-Related Orphan Receptor C2
Narjes, Frank, Llinas, Antonio, von Berg, Stefan, Jirholt, Johan, Lever, Sarah, Pehrson, Rikard, Collins, Mia, Malmberg, Anna, Svanberg, Petter, Xue, Yafeng, Olsson, Roine I, Malmberg, Jesper, Hughes, Glyn, Hossain, Nafizal, Grindebacke, Hanna, Leffler, Agnes, Krutrök, Nina, Bäck, Elisabeth, Ramnegård, Marie, Lepistö, Matti, Thunberg, Linda, Aagaard, Anna, McPheat, Jane, Hansson, Eva L, Chen, Rongfeng, Xiong, Yao, Hansson, Thomas G
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
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Discovery of a Novel Oral Glucocorticoid Receptor Modulator (AZD9567) with Improved Side Effect Profile
Ripa, Lena, Edman, Karl, Dearman, Matthew, Edenro, Goran, Hendrickx, Ramon, Ullah, Victoria, Chang, Hui-Fang, Lepistö, Matti, Chapman, Dave, Geschwindner, Stefan, Wissler, Lisa, Svanberg, Petter, Lawitz, Karolina, Malmberg, Jesper, Nikitidis, Antonios, Olsson, Roine I, Bird, James, Llinas, Antoni, Hegelund-Myrbäck, Tove, Berger, Markus, Thorne, Philip, Harrison, Richard, Köhler, Christian, Drmota, Tomas
Published in Journal of medicinal chemistry (08.03.2018)
Published in Journal of medicinal chemistry (08.03.2018)
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Potent and Orally Bioavailable Inverse Agonists of RORγt Resulting from Structure-Based Design
Narjes, Frank, Xue, Yafeng, von Berg, Stefan, Malmberg, Jesper, Llinas, Antonio, Olsson, Roine I, Jirholt, Johan, Grindebacke, Hanna, Leffler, Agnes, Hossain, Nafizal, Lepistö, Matti, Thunberg, Linda, Leek, Hanna, Aagaard, Anna, McPheat, Jane, Hansson, Eva L, Bäck, Elisabeth, Tångefjord, Stefan, Chen, Rongfeng, Xiong, Yao, Hongbin, Ge, Hansson, Thomas G
Published in Journal of medicinal chemistry (13.09.2018)
Published in Journal of medicinal chemistry (13.09.2018)
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Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (TH17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor RORγ
Olsson, Roine I., Xue, Yafeng, von Berg, Stefan, Aagaard, Anna, McPheat, Jane, Hansson, Eva L., Bernström, Jenny, Hansson, Pia, Jirholt, Johan, Grindebacke, Hanna, Leffler, Agnes, Chen, Rongfeng, Xiong, Yao, Ge, Hongbin, Hansson, Thomas G., Narjes, Frank
Published in ChemMedChem (19.01.2016)
Published in ChemMedChem (19.01.2016)
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Structure–Affinity Relationships and Structure–Kinetic Relationships of 1,2-Diarylimidazol-4-carboxamide Derivatives as Human Cannabinoid 1 Receptor Antagonists
Xia, Lizi, de Vries, Henk, Lenselink, Eelke B., Louvel, Julien, Waring, Michael J., Cheng, Leifeng, Pahlén, Sara, Petersson, Maria J., Schell, Peter, Olsson, Roine I., Heitman, Laura H., Sheppard, Robert J., IJzerman, Adriaan P.
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Discovery of Potent and Orally Bioavailable Inverse Agonists of the Retinoic Acid Receptor-Related Orphan Receptor C2
von Berg, Stefan, Xue, Yafeng, Collins, Mia, Llinas, Antonio, Olsson, Roine I, Halvarsson, Torbjörn, Lindskog, Maria, Malmberg, Jesper, Jirholt, Johan, Krutrök, Nina, Ramnegård, Marie, Brännström, Marie, Lundqvist, Anders, Lepistö, Matti, Aagaard, Anna, McPheat, Jane, Hansson, Eva L, Chen, Rongfeng, Xiong, Yao, Hansson, Thomas G, Narjes, Frank
Published in ACS medicinal chemistry letters (13.06.2019)
Published in ACS medicinal chemistry letters (13.06.2019)
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Journal Article
Isoindolinone compounds active as Kv1.5 blockers identified using a multicomponent reaction approach
Kajanus, Johan, Jacobson, Ingemar, Åstrand, Annika, Olsson, Roine I., Gran, Ulrik, Björe, Annika, Fjellström, Ola, Davidsson, Öjvind, Emtenäs, Hans, Dahlén, Anders, Löfberg, Boel, Yuan, Zhong-Qing, Sundell, Johan, Cassel, Johan, Gyll, Jonna, Iliefski, Tommy, Högberg, Ågot, Lindhardt, Emma, Malmberg, Jesper
Published in Bioorganic & medicinal chemistry letters (15.04.2016)
Published in Bioorganic & medicinal chemistry letters (15.04.2016)
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Journal Article
Lactam sulfonamides as potent inhibitors of the Kv1.5 potassium ion channel
Olsson, Roine I., Jacobson, Ingemar, Iliefski, Tommy, Bostrom, Jonas, Davidsson, Ojvind, Fjellstrom, Ola, Bjore, Annika, Olsson, Christina, Sundell, Johan, Gran, Ulrik, Gyll, Jonna, Malmberg, Jesper, Hidestal, Olle, Emtenas, Hans, Svensson, Tor, Yuan, Zhong-Qing, Strandlund, Gert, Astrand, Annika, Lindhardt, Emma, Linhardt, Gunilla, Forsstrom, Elin, Hogberg, Agot, Persson, Frida, Andersson, Birgit, Ronnborg, Anna, Lofberg, Boel
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
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Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (T(H)17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor ROR gamma
Olsson, Roine I., Xue, Yafeng, von Berg, Stefan, Aagaard, Anna, McPheat, Jane, Hansson, Eva L., Bernstrom, Jenny, Hansson, Pia, Jirholt, Johan, Grindebacke, Hanna, Leffler, Agnes, Chen, Rongfeng, Xiong, Yao, Ge, Hongbin, Hansson, Thomas G., Narjes, Frank
Published in ChemMedChem (19.01.2016)
Published in ChemMedChem (19.01.2016)
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Journal Article
Back Cover: Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper17 (TH17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor ROR[gamma]
Olsson, Roine I, Xue, Yafeng, vonBerg, Stefan, Aagaard, Anna, McPheat, Jane, Hansson, Eva L, Bernstrom, Jenny, Hansson, Pia, Jirholt, Johan, Grindebacke, Hanna, Leffler, Agnes, Chen, Rongfeng, Xiong, Yao, Ge, Hongbin, Hansson, Thomas G, Narjes, Frank
Published in ChemMedChem (01.01.2016)
Published in ChemMedChem (01.01.2016)
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Journal Article
Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper17 (TH17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor ROR[gamma]
Olsson, Roine I, Xue, Yafeng, vonBerg, Stefan, Aagaard, Anna, McPheat, Jane, Hansson, Eva L, Bernstrom, Jenny, Hansson, Pia, Jirholt, Johan, Grindebacke, Hanna, Leffler, Agnes, Chen, Rongfeng, Xiong, Yao, Ge, Hongbin, Hansson, Thomas G, Narjes, Frank
Published in ChemMedChem (01.01.2016)
Published in ChemMedChem (01.01.2016)
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Back Cover: Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (TH17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor RORγ (ChemMedChem 2/2016)
Olsson, Roine I., Xue, Yafeng, von Berg, Stefan, Aagaard, Anna, McPheat, Jane, Hansson, Eva L., Bernström, Jenny, Hansson, Pia, Jirholt, Johan, Grindebacke, Hanna, Leffler, Agnes, Chen, Rongfeng, Xiong, Yao, Ge, Hongbin, Hansson, Thomas G., Narjes, Frank
Published in ChemMedChem (01.01.2016)
Published in ChemMedChem (01.01.2016)
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