Small-molecule agonists and antagonists of the opioid receptor-like receptor (ORL1, NOP): ligand-based analysis of structural factors influencing intrinsic activity at NOP
Zaveri, Nurulain, Jiang, Faming, Olsen, Cris, Polgar, Willma, Toll, Lawrence
Published in The AAPS journal (05.10.2005)
Published in The AAPS journal (05.10.2005)
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A Novel Series of Piperidin-4-yl-1,3-Dihydroindol-2-ones as Agonist and Antagonist Ligands at the Nociceptin Receptor
Zaveri, Nurulain T, Jiang, Faming, Olsen, Cris M, Deschamps, Jeffrey R, Parrish, Damon, Polgar, Willma, Toll, Lawrence
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Novel alpha 3 beta 4 Nicotinic Acetylcholine Receptor-Selective Ligands. Discovery, Structure-Activity Studies, and Pharmacological Evaluation
Zaveri, Nurulain, Jiang, Faming, Olsen, Cris, Polgar, Willma, Toll, Lawrence
Published in Journal of medicinal chemistry (25.11.2010)
Published in Journal of medicinal chemistry (25.11.2010)
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Comparison of the antinociceptive and antirewarding profiles of novel bifunctional nociceptin receptor/mu-opioid receptor ligands: implications for therapeutic applications
Toll, Lawrence, Khroyan, Taline V, Polgar, Willma E, Jiang, Faming, Olsen, Cris, Zaveri, Nurulain T
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
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SR 16435 [1-(1-(bicyclo[3.3.1]nonan-9-yl)piperidin-4-yl)indolin-2-one], a novel mixed nociceptin/orphanin FQ/mu-opioid receptor partial agonist: analgesic and rewarding properties in mice
Khroyan, Taline V, Zaveri, Nurulain T, Polgar, Willma E, Orduna, Juan, Olsen, Cris, Jiang, Faming, Toll, Lawrence
Published in The Journal of pharmacology and experimental therapeutics (01.02.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2007)
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Novel alpha3beta4 nicotinic acetylcholine receptor-selective ligands. Discovery, structure-activity studies and pharmacological evaluation
Zaveri, Nurulain, Jiang, Faming, Olsen, Cris, Polgar, Willma, Toll, Lawrence
Published in Journal of medicinal chemistry (27.10.2010)
Published in Journal of medicinal chemistry (27.10.2010)
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Comparison of the Antinociceptive and Antirewarding Profiles of Novel Bifunctional Nociceptin Receptor/μ-Opioid Receptor Ligands: Implications for Therapeutic Applications
Lawrence Toll, Taline V. Khroyan, Willma E. Polgar, Faming Jiang, Cris Olsen, Nurulain T. Zaveri
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
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Activity of new NOP receptor ligands in a rat peripheral mononeuropathy model: Potentiation of morphine
Khroyan, Taline V, Polgar, Willma E, Orduna, Juan, Jiang, Faming, Olsen, Cris, Toll, Lawrence, Zaveri, Nurulain T
Published in European journal of pharmacology (01.05.2009)
Published in European journal of pharmacology (01.05.2009)
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Activity of new NOP receptor ligands in a rat peripheral mononeuropathy model: Potentiation of morphine anti-allodynic activity by NOP receptor antagonists
Khroyan, Taline V., Polgar, Willma E., Orduna, Juan, Jiang, Faming, Olsen, Cris, Toll, Lawrence, Zaveri, Nurulain T.
Published in European journal of pharmacology (21.05.2009)
Published in European journal of pharmacology (21.05.2009)
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Journal Article
SR 16435 [1-(1-(Bicyclo[3.3.1]nonan-9-yl)piperidin-4-yl)indolin-2-one], a Novel Mixed Nociceptin/Orphanin FQ/μ-Opioid Receptor Partial Agonist: Analgesic and Rewarding Properties in Mice
Taline V. Khroyan, Nurulain T. Zaveri, Willma E. Polgar, Juan Orduna, Cris Olsen, Faming Jiang, Lawrence Toll
Published in The Journal of pharmacology and experimental therapeutics (01.02.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2007)
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Replacement of the peptide-backbone amides connecting Tyr-Gly and Gly-Gly in leucine-enkephalin with ketomethylene groups: synthesis and biological activity
Almquist, Ronald G, Olsen, Cris M, Uyeno, Edward T, Toll, Lawrence
Published in Journal of medicinal chemistry (01.02.1984)
Published in Journal of medicinal chemistry (01.02.1984)
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The synthesis and biological activity of two analogs of the anti-HIV alkaloid michellamine B
Upender, Pollart, DJ, Liu, J, Hobbs, PD, Olsen, C, Chao, WR, Bowden, B, Crase, JL, Thomas, DW, Pandey, A, Lawson, JA, Dawson, MI
Published in Journal of heterocyclic chemistry (01.07.1996)
Published in Journal of heterocyclic chemistry (01.07.1996)
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Nicotinic acetylcholine receptor modulators
KHROYAN TALINE, POLGAR WILLMA E, ZAVERI NURULAIN T, JIANG FAMING, OLSEN CRIS M, TOLL LAWRENCE R
Year of Publication 15.04.2014
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Year of Publication 15.04.2014
Patent
NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS
JIANG, FAMING, OLSEN, CRIS, M, ZAVERI, NURULAIN, T, KHROYAN, TALINE, POLGAR, WILLMA, E, TOLL, LAWRENCE, R
Year of Publication 07.05.2009
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Year of Publication 07.05.2009
Patent
Nicotinic Acetylcholine Receptor Modulators
KHROYAN TALINE, POLGAR WILLMA E, ZAVERI NURULAIN T, JIANG FAMING, OLSEN CRIS M, TOLL LAWRENCE R
Year of Publication 07.05.2009
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Year of Publication 07.05.2009
Patent
Structure of a Bovine Thrombin-Hirudin51−65 Complex Determined by a Combination of Molecular Replacement and Graphics. Incorporation of Known Structural Information in Molecular Replacement
Vitali, J., Martin, P. D., Malkowski, M. G., Olsen, C. M., Johnson, P. H., Edwards, B. F. P.
Published in Acta crystallographica. Section D, Biological crystallography. (01.05.1996)
Published in Acta crystallographica. Section D, Biological crystallography. (01.05.1996)
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