Rh(III)-Catalyzed C–H Activation and Double Directing Group Strategy for the Regioselective Synthesis of Naphthyridinones
Huckins, John R, Bercot, Eric A, Thiel, Oliver R, Hwang, Tsang-Lin, Bio, Matthew M
Published in Journal of the American Chemical Society (02.10.2013)
Published in Journal of the American Chemical Society (02.10.2013)
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Journal Article
An Efficient and Scalable Ritter Reaction for the Synthesis of tert-Butyl Amides
Baum, Jean C, Milne, Jacqueline E, Murry, Jerry A, Thiel, Oliver R
Published in Journal of organic chemistry (06.03.2009)
Published in Journal of organic chemistry (06.03.2009)
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Journal Article
DYKAT of Baylis−Hillman Adducts: Concise Total Synthesis of Furaquinocin E
Trost, Barry M, Thiel, Oliver R, Tsui, Hon-Chung
Published in Journal of the American Chemical Society (02.10.2002)
Published in Journal of the American Chemical Society (02.10.2002)
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Journal Article
Selection of a Suitable Physical Form and Development of a Crystallization Process for a PDE10A Inhibitor Exhibiting Enantiotropic Polymorphism
Kiang, Y.-H, Bercot, Eric A, Wu, Qiong, Liu, Jodi, Milburn, Robert R, Cohen, Dawn E, Borths, Christopher J, Saw, Robert E, Staples, Richard J, Davis, Carl, Thiel, Oliver R
Published in Organic process research & development (18.12.2015)
Published in Organic process research & development (18.12.2015)
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Journal Article
Palladium-Catalyzed Coupling of Aldehyde-Derived Hydrazones: Practical Synthesis of Triazolopyridines and Related Heterocycles
Thiel, Oliver R., Achmatowicz, Michal M., Reichelt, Andreas, Larsen, Robert D.
Published in Angewandte Chemie International Edition (02.11.2010)
Published in Angewandte Chemie International Edition (02.11.2010)
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Journal Article
Development of a Practical Synthesis of a p38 MAP Kinase Inhibitor
Thiel, Oliver R, Achmatowicz, Michal, Bernard, Charles, Wheeler, Philip, Savarin, Cecile, Correll, Tiffany L, Kasparian, Annie, Allgeier, Alan, Bartberger, Michael D, Tan, Helming, Larsen, Robert D
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Journal Article
Synthesis of Substituted Pyridines via Formal (3+3) Cycloaddition of Enamines with Unsaturated Aldehydes and Ketones
Dai, Xi-Jie, Krolikowski, Paul, Murray, James I., Wei, Carolyn S., Dornan, Peter K., Rötheli, Andreas R., Caille, Seb, Thiel, Oliver R., Smith, Austin G., Parsons, Andrew T.
Published in Journal of organic chemistry (01.07.2022)
Published in Journal of organic chemistry (01.07.2022)
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Journal Article
Accelerated Development of a Scalable Ring-Closing Metathesis to Manufacture AMG 176 Using a Combined High-Throughput Experimentation and Computational Modeling Approach
St-Pierre, Gabrielle, Cherney, Alan H, Chen, Wencan, Dong, Xiaofei, Dornan, Peter K, Griffin, Daniel J, Houk, K. N, Lin, Janice B, Osgood, Stephen, Silva Elipe, Maria V, Timmons, Heath C, Xie, Yong, Tedrow, Jason S, Thiel, Oliver R, Smith, Austin G
Published in Organic process research & development (19.03.2021)
Published in Organic process research & development (19.03.2021)
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Journal Article
Palladium-Catalyzed Chemoselective Monoarylation of Hydrazides for the Synthesis of [1,2,4]Triazolo[4,3-a]pyridines
Reichelt, Andreas, Falsey, James R, Rzasa, Robert M, Thiel, Oliver R, Achmatowicz, Michal M, Larsen, Robert D, Zhang, Dawei
Published in Organic letters (19.02.2010)
Published in Organic letters (19.02.2010)
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Journal Article
Green Chemistry as a Driver for Innovation in the Pharmaceutical Industry
Beaver, Matthew G., Caille, Seb, Içten, Elçin, Michalak, Sharon E., St‐Pierre, Gabrielle, Thiel, Oliver R.
Published in Israel journal of chemistry (01.07.2021)
Published in Israel journal of chemistry (01.07.2021)
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Journal Article
Synthesis of a Ring-Expanded Bryostatin Analogue
Trost, Barry M, Yang, Hanbiao, Thiel, Oliver R, Frontier, Alison J, Brindle, Cheyenne S
Published in Journal of the American Chemical Society (28.02.2007)
Published in Journal of the American Chemical Society (28.02.2007)
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Journal Article
An Improved Process for the Preparation of a Covalent Kinase Inhibitor through a C–N Bond-Forming SNAr Reaction
Parsons, Andrew T, Kubryk, Michele, Hedley, Simon J, Thiel, Oliver R, Bauer, David, Potter-Racine, Matthew S, Lin, Zhenxin
Published in Organic process research & development (20.07.2018)
Published in Organic process research & development (20.07.2018)
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Journal Article
Development of a Factory Process for Omecamtiv Mecarbil, a Novel Cardiac Myosin Activator
Caille, Seb, Allgeier, Alan M, Bernard, Charles, Correll, Tiffany L, Cosbie, Andrew, Crockett, Richard D, Cui, Sheng, Faul, Margaret M, Hansen, Karl B, Huggins, Seth, Langille, Neil, Mennen, Steven M, Morgan, Bradley P, Morrison, Henry, Muci, Alexander, Nagapudi, Karthik, Quasdorf, Kyle, Ranganathan, Krishnakumar, Roosen, Philipp, Shi, Xianqing, Thiel, Oliver R, Wang, Fang, Tvetan, Justin T, Woo, Jacqueline C. S, Wu, Steven, Walker, Shawn D
Published in Organic process research & development (16.08.2019)
Published in Organic process research & development (16.08.2019)
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Journal Article