Comparative Investigation of Ruthenium-Based Metathesis Catalysts Bearing N-Heterocyclic Carbene (NHC) Ligands
Fürstner, Alois, Ackermann, Lutz, Gabor, Barbara, Goddard, Richard, Lehmann, Christian W., Mynott, Richard, Stelzer, Frank, Thiel, Oliver R.
Published in Chemistry : a European journal (03.08.2001)
Published in Chemistry : a European journal (03.08.2001)
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Journal Article
Telescoped Process to Manufacture 6,6,6-Trifluorofucose via Diastereoselective Transfer Hydrogenation: Scalable Access to an Inhibitor of Fucosylation Utilized in Monoclonal Antibody Production
Achmatowicz, Michal M, Allen, John G, Bio, Matthew M, Bartberger, Michael D, Borths, Christopher J, Colyer, John T, Crockett, Richard D, Hwang, Tsang-Lin, Koek, Jan. N, Osgood, Stephen A, Roberts, Scott W, Swietlow, Aleksander, Thiel, Oliver R, Caille, Seb
Published in Journal of organic chemistry (03.06.2016)
Published in Journal of organic chemistry (03.06.2016)
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Journal Article
AMG 580: a novel small molecule phosphodiesterase 10A (PDE10A) positron emission tomography tracer
Chen, Hang, Lester-Zeiner, Dianna, Shi, Jianxia, Miller, Silke, Glaus, Charlie, Hu, Essa, Chen, Ning, Able, Jessica, Biorn, Christopher, Wong, Jamie, Ma, Ji, Michelsen, Klaus, Hill Della Puppa, Geraldine, Kazules, Tim, Dou, Hui Hannah, Talreja, Santosh, Zhao, Xiaoning, Chen, Ada, Rumfelt, Shannon, Kunz, Roxanne K, Ye, Hu, Thiel, Oliver R, Williamson, Toni, Davis, Carl, Porter, Amy, Immke, David, Allen, Jennifer R, Treanor, James
Published in The Journal of pharmacology and experimental therapeutics (01.02.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2015)
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Journal Article
Total Syntheses of Furaquinocin A, B, and E
Trost, Barry M, Thiel, Oliver R, Tsui, Hon-Chung
Published in Journal of the American Chemical Society (29.10.2003)
Published in Journal of the American Chemical Society (29.10.2003)
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Journal Article
Total Synthesis of Bryostatins: The Development of Methodology for the Atom-Economic and Stereoselective Synthesis of the Ring C Subunit
Trost, Barry M., Frontier, Alison J., Thiel, Oliver R., Yang, Hanbiao, Dong, Guangbin
Published in Chemistry : a European journal (22.08.2011)
Published in Chemistry : a European journal (22.08.2011)
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Journal Article
Practical Synthesis of a Vanilloid Receptor-1 Antagonist
Thiel, Oliver R, Bernard, Charles, King, Tony, Dilmeghani-Seran, Mina, Bostick, Tracy, Larsen, Robert D, Faul, Margaret M
Published in Journal of organic chemistry (02.05.2008)
Published in Journal of organic chemistry (02.05.2008)
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Journal Article
Hydrolysis of Phosphoryl Trichloride (POCl3): Characterization, in Situ Detection, and Safe Quenching of Energetic Metastable Intermediates
Achmatowicz, Michał M, Thiel, Oliver R, Colyer, John T, Hu, Jack, Elipe, Maria Victoria Silva, Tomaskevitch, Joe, Tedrow, Jason S, Larsen, Robert D
Published in Organic process research & development (19.11.2010)
Published in Organic process research & development (19.11.2010)
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Journal Article
Total Syntheses of (S)-(−)-Zearalenone and Lasiodiplodin Reveal Superior Metathesis Activity of Ruthenium Carbene Complexes with Imidazol-2-ylidene Ligands
Fürstner, Alois, Thiel, Oliver R, Kindler, Nicole, Bartkowska, Beata
Published in Journal of organic chemistry (17.11.2000)
Published in Journal of organic chemistry (17.11.2000)
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Journal Article
Oxopyrido[2,3‑d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors
Wurz, Ryan P, Pettus, Liping H, Ashton, Kate, Brown, James, Chen, Jian Jeffrey, Herberich, Brad, Hong, Fang-Tsao, Hu-Harrington, Essa, Nguyen, Tom, St. Jean, David J, Tadesse, Seifu, Bauer, David, Kubryk, Michele, Zhan, Jinghui, Cooke, Keegan, Mitchell, Petia, Andrews, Kristin L, Hsieh, Faye, Hickman, Dean, Kalyanaraman, Nataraj, Wu, Tian, Reid, Darren L, Lobenhofer, Edward K, Andrews, Dina A, Everds, Nancy, Guzman, Roberto, Parsons, Andrew T, Hedley, Simon J, Tedrow, Jason, Thiel, Oliver R, Potter, Matthew, Radinsky, Robert, Beltran, Pedro J, Tasker, Andrew S
Published in ACS medicinal chemistry letters (10.09.2015)
Published in ACS medicinal chemistry letters (10.09.2015)
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Journal Article
METHOD OF CONJUGATION OF CYS-MAB
DANTE ROMANINI, BRADLEY J HERBERICH, MICHAL ACHMATOWICZ, JAMES R FALSEY, OLIVER R THIEL
Year of Publication 10.07.2024
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Year of Publication 10.07.2024
Patent
Practical Synthesis of a p38 MAP Kinase Inhibitor
Achmatowicz, Michał, Thiel, Oliver R, Wheeler, Philip, Bernard, Charles, Huang, Jinkun, Larsen, Robert D, Faul, Margaret M
Published in Journal of organic chemistry (16.01.2009)
Published in Journal of organic chemistry (16.01.2009)
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Journal Article
Mechanistic Insights and Safety Evaluation of the Ritter Reaction Utilizing tert-Butyl Acetate as the tert-Butyl Cation Source
Roberts, Scott W, Shaw, Stephen M, Milne, Jacqueline E, Cohen, Dawn E, Tvetan, Justin T, Tomaskevitch, Joseph, Thiel, Oliver R
Published in Organic process research & development (21.12.2012)
Published in Organic process research & development (21.12.2012)
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Journal Article
Development of a Practical Synthesis of a Pyrazolopyridinone-Based p38 MAP Kinase Inhibitor
Milburn, Robert R, Thiel, Oliver R, Achmatowicz, Michal, Wang, Xiang, Zigterman, Jamie, Bernard, Charles, Colyer, John T, DiVirgilio, Evan, Crockett, Rich, Correll, Tiffany L, Nagapudi, Karthik, Ranganathan, Kumar, Hedley, Simon J, Allgeier, Alan, Larsen, Robert D
Published in Organic process research & development (21.01.2011)
Published in Organic process research & development (21.01.2011)
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Journal Article
Leveraging ICH M7 Control Options 3 and 4: Discussion and Clarification Using Industrial Case Studies
Urquhart, Michael W., Burns, Michael J., Clark, Hugh F., Crochard, Jean-Philippe, Dirat, Olivier, Hildbrand, Stefan, Moessner, Christian, Pascoe, David D., Roberts, Alastair J., Teasdale, Andrew, Thiel, Oliver R.
Published in Organic process research & development (16.08.2024)
Published in Organic process research & development (16.08.2024)
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Journal Article
PAT-Enabled Automated Feedforward Control: An Application to the Continuous Manufacture of Apremilast
Hsieh, Hsiao-Wu, Griffin, Daniel J., Nambiar, Anirudh M. K., Sarkar, Nandini, Youssef Ismail, Hamza, Saigal, Kartik, Shen, Dongying Erin, Goudas-Salomon, Nicole, Wimalasinghe, Rasangi, Zeng, Alicia, Thiel, Oliver R., Beaver, Matthew G.
Published in Organic process research & development (19.07.2024)
Published in Organic process research & development (19.07.2024)
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Journal Article
Development of a scalable route to a complex cyclobutane linchpin via a diastereoselective CuI-catalyzed vinylation of a cyclobutanyl aldehyde
Corbett, Michael T., Baucom, Kyle, Cui, Sheng, Dornan, Peter K., Jiao, Fangxia, Han, Jun, Langille, Neil F., Osgood, Steve, Parsons, Andrew T., Quasdorf, Kyle W., Rötheli, Andreas R., Elipe, Maria Victoria Silva, Sangodkar, Rahul P., Smith, Austin G., Spada, Simone, Stahl, Amanda E., St-Pierre, Gabrielle, Thiel, Oliver R., Walker, Shawn D., Xie, Yong, Yang, Ning
Published in Tetrahedron (10.09.2024)
Published in Tetrahedron (10.09.2024)
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Journal Article