Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation
Peauger, Ludovic, Azzouz, Rabah, Gembus, Vincent, Ţînţaş, Mihaela-Liliana, Sopková-de Oliveira Santos, Jana, Bohn, Pierre, Papamicaël, Cyril, Levacher, Vincent
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
Get full text
Journal Article
Drug Repurposing: Deferasirox Inhibits the Anti-Apoptotic Activity of Mcl-1
Bourafai-Aziez, Asma, Benabderrahmane, Mohammed, Paysant, Hippolyte, Weiswald, Louis-Bastien, Poulain, Laurent, Carlier, Ludovic, Ravault, Delphine, Jouanne, Marie, Coadou, Gaël, Oulyadi, Hassan, Voisin-Chiret, Anne-Sophie, Sopková-de Oliveira Santos, Jana, Sebban, Muriel
Published in Drug design, development and therapy (01.01.2021)
Published in Drug design, development and therapy (01.01.2021)
Get full text
Journal Article
Development of Novel Potential Pleiotropic Compounds of Interest in Alzheimer's Disease Treatment through Rigidification Strategy
Lecoutey, Cédric, Legay, Rémi, Davis, Audrey, Sopková-de Oliveira Santos, Jana, Dallemagne, Patrick, Rochais, Christophe
Published in Molecules (Basel, Switzerland) (26.04.2021)
Published in Molecules (Basel, Switzerland) (26.04.2021)
Get full text
Journal Article
A Three-Site Mechanism for Agonist/Antagonist Selective Binding to Vasopressin Receptors
Saleh, Noureldin, Saladino, Giorgio, Gervasio, Francesco L., Haensele, Elke, Banting, Lee, Whitley, David C., Sopkova-de Oliveira Santos, Jana, Bureau, Ronan, Clark, Timothy
Published in Angewandte Chemie (International ed.) (04.07.2016)
Published in Angewandte Chemie (International ed.) (04.07.2016)
Get full text
Journal Article
One-pot synthesis of new aza- and diaza-aminophenanthrenes
Rochais, Christophe, Yougnia, Rodrigue, Cailly, Thomas, Sopková-de Oliveira Santos, Jana, Rault, Sylvain, Dallemagne, Patrick
Published in Tetrahedron (12.08.2011)
Published in Tetrahedron (12.08.2011)
Get full text
Journal Article
Room-Temperature ortho-Alkoxylation and -Halogenation of N-Tosylbenzamides by Using Palladium(II)-Catalyzed CH Activation
Péron, Florent, Fossey, Christine, Sopkova-de Oliveira Santos, Jana, Cailly, Thomas, Fabis, Frédéric
Published in Chemistry : a European journal (10.06.2014)
Published in Chemistry : a European journal (10.06.2014)
Get full text
Journal Article
Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core
Ţînţaş, Mihaela-Liliana, Peauger, Ludovic, Alix, Florent, Papamicaël, Cyril, Besson, Thierry, Sopková-de Oliveira Santos, Jana, Gembus, Vincent, Levacher, Vincent
Published in Molecules (Basel, Switzerland) (01.01.2023)
Published in Molecules (Basel, Switzerland) (01.01.2023)
Get full text
Journal Article
Effect of oral exposure to the acaricide pirimicarb, a new varroacide candidate, on Apis mellifera feeding rate
Riva, Clémence, Sokolowski, Michel BC, Normand, Julien, Santos, Jana Sopkova‐de Oliveira, Halm‐Lemeille, Marie‐Pierre
Published in Pest management science (01.08.2018)
Published in Pest management science (01.08.2018)
Get full text
Journal Article
Synthesis and Physicochemical Properties of Cryptophazane—A Soluble and Functionalizable C1‐Symmetrical Cryptophane
Vigier, Clément, Fayolle, Dimitri, El Siblani, Hussein, Sopkova ‐ de Oliveira Santos, Jana, Fabis, Frederic, Cailly, Thomas, Dubost, Emmanuelle
Published in Angewandte Chemie International Edition (14.11.2022)
Published in Angewandte Chemie International Edition (14.11.2022)
Get full text
Journal Article
Selecting the first chemical molecule inhibitor of HSP110 for colorectal cancer therapy
Gozzi, Gustavo J., Gonzalez, Daniel, Boudesco, Christophe, Dias, Alexandre M. M., Gotthard, Guillaume, Uyanik, Burhan, Dondaine, Lucile, Marcion, Guillaume, Hermetet, François, Denis, Camille, Hardy, Laurianne, Suzanne, Peggy, Douhard, Romain, Jego, Gaetan, Dubrez, Laurence, Demidov, Oleg N., Neiers, Fabrice, Briand, Loïc, Sopková-de Oliveira Santos, Jana, Voisin-Chiret, Anne-Sophie, Garrido, Carmen
Published in Cell death and differentiation (01.01.2020)
Published in Cell death and differentiation (01.01.2020)
Get full text
Journal Article
Web Resource
Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer's Disease
Toublet, François-Xavier, Lecoutey, Cédric, Lalut, Julien, Hatat, Bérénice, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopkova de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in Molecules (Basel, Switzerland) (31.07.2019)
Published in Molecules (Basel, Switzerland) (31.07.2019)
Get full text
Journal Article
Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5‑HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers
Dubost, Emmanuelle, Dumas, Noé, Fossey, Christine, Magnelli, Rosa, Butt-Gueulle, Sabrina, Ballandonne, Céline, Caignard, Daniel H, Dulin, Fabienne, Sopkova de-Oliveira Santos, Jana, Millet, Philippe, Charnay, Yves, Rault, Sylvain, Cailly, Thomas, Fabis, Frederic
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
Get full text
Journal Article
Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A/CLK1 kinases
în a, Mihaela-Liliana, Peauger, Ludovic, Barré, Anaïs, Papamicaël, Cyril, Besson, Thierry, Sopkovà-de Oliveira Santos, Jana, Gembus, Vincent, Levacher, Vincent
Published in MedChemComm (20.03.2024)
Published in MedChemComm (20.03.2024)
Get full text
Journal Article
An Efficient and Straightforward Access to Sulfur Substituted [2.2]Paracyclophanes: Application to Stereoselective Sulfenate Salt Alkylation
Lohier, Jean-François, Foucoin, Florian, Jaffrès, Paul-Alain, Garcia, José I, Sopková−de Oliveira Santos, Jana, Perrio, Stéphane, Metzner, Patrick
Published in Organic letters (20.03.2008)
Published in Organic letters (20.03.2008)
Get full text
Journal Article
Quinoline derivatives: potential antiparasitic and antiviral agents
Sopková-de Oliveira Santos, Jana, Verhaeghe, Pierre, Lohier, Jean-François, Rathelot, Pascal, Vanelle, Patrice, Rault, Sylvain
Published in Acta crystallographica. Section C, Crystal structure communications (01.11.2007)
Published in Acta crystallographica. Section C, Crystal structure communications (01.11.2007)
Get full text
Journal Article
Structure-guided design of pyridoclax derivatives based on Noxa / Mcl-1 interaction mode
Hedir, Siham, De Giorgi, Marcella, Fogha, Jade, De Pascale, Martina, Weiswald, Louis-Bastien, Brotin, Emilie, Marekha, Bogdan, Denoyelle, Christophe, Denis, Camille, Suzanne, Peggy, Gautier, Fabien, Juin, Philippe, Ligat, Laetitia, Lopez, Frédéric, Carlier, Ludovic, Legay, Rémi, Bureau, Ronan, Rault, Sylvain, Poulain, Laurent, Oliveira Santos, Jana Sopková-de, Voisin-Chiret, Anne Sophie
Published in European journal of medicinal chemistry (05.11.2018)
Published in European journal of medicinal chemistry (05.11.2018)
Get full text
Journal Article
Design and synthesis of thienylpyridyl garlands as non-peptidic alpha helix mimetics and potential protein–protein interactions disruptors
De Giorgi, Marcella, Voisin-Chiret, Anne Sophie, Sopková-de Oliveira Santos, Jana, Corbo, Filomena, Franchini, Carlo, Rault, Sylvain
Published in Tetrahedron (26.08.2011)
Published in Tetrahedron (26.08.2011)
Get full text
Journal Article
One-pot synthesis of novel poly-substituted phenanthrenes
Yougnia, Rodrigue, Rochais, Christophe, Oliveira Santos, Jana Sopkovà-de, Dallemagne, Patrick, Rault, Sylvain
Published in Tetrahedron (10.04.2010)
Published in Tetrahedron (10.04.2010)
Get full text
Journal Article