Structure‐Metabolism Relationships of Benzimidazole Derivatives with anti‐Trypanosoma cruzi Activity for Chagas Disease
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Published in ChemMedChem (16.10.2024)
Published in ChemMedChem (16.10.2024)
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Synthesis, Design, and Structure‐Activity Relationship of a Benzenesulfonylpiperazine Series against Trypanosoma cruzi
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Published in ChemMedChem (06.10.2022)
Published in ChemMedChem (06.10.2022)
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The in vitro activity of fatty diamines and amino alcohols against mixed amastigote and trypomastigote Trypanosoma cruzi forms
Júnior, Policarpo Ademar Sales, Júnior, Celso Oliveira Rezende, Le Hyaric, Mireille, de Almeida, Mauro Vieira, Romanha, Alvaro José
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Published in Memórias do Instituto Oswaldo Cruz (01.06.2014)
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Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum
Lapierre, Thibault Joseph William Jacques Dit, Farago, Danilo Nascimento, de Moura Lodi Cruz, Mariza Gabriela Faleiro, de Melo Resende, Daniela, de Oliveira, Adriane Cristina Rosa, Dos Santos, Brenda Rosa Macedo, de Oliveira Souza, Felipe, Michelan-Duarte, Simone, Chelucci, Rafael C, Andricopulo, Adriano D, Ferreira, Leonardo L G, Pilau, Eduardo Jorge, Murta, Silvane Maria Fonseca, de Oliveira Rezende Júnior, Celso
Published in Chemical biology & drug design (01.04.2024)
Published in Chemical biology & drug design (01.04.2024)
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A Novel Compound from the Phenylsulfonylpiperazine Class: Evaluation of In Vitro Activity on Luminal Breast Cancer Cells
da Silva, Fernanda Cardoso, Martinho, Ana Clara Cassiano, Ferreira, Helen Soares Valença, Siqueira, Raoni Pais, Arruda, Vinicius Marques, Guerra, Joyce Ferreira da Costa, de Souza, Maria Laura Dos Reis, Landin, Emanuelly Silva, Rezende Júnior, Celso de Oliveira, de Araújo, Thaise Gonçalves
Published in Molecules (Basel, Switzerland) (20.09.2024)
Published in Molecules (Basel, Switzerland) (20.09.2024)
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Structure-based discovery of thiosemicarbazones as SARS-CoV-2 main protease inhibitors
Maltarollo, Vinícius Gonçalves, da Silva, Elany Barbosa, Kronenberger, Thales, Sena Andrade, Marina Mol, de Lima Marques, Gabriel V, Cândido Oliveira, Nereu J, Santos, Lucianna H, Oliveira Rezende Júnior, Celso de, Cassiano Martinho, Ana C, Skinner, Danielle, Fajtová, Pavla, M Fernandes, Thaís H, Silveira Dos Santos, Eduardo da, Rodrigues Gazolla, Poliana A, Martins de Souza, Ana P, da Silva, Milene Lopes, Dos Santos, Fabíola S, Lavorato, Stefânia N, Oliveira Bretas, Ana C, Carvalho, Diogo Teixeira, Franco, Lucas Lopardi, Luedtke, Stephanie, Giardini, Miriam A, Poso, Antti, Dias, Luiz C, Podust, Larissa M, Alves, Ricardo J, McKerrow, James, Andrade, Saulo F, Teixeira, Róbson R, Siqueira-Neto, Jair L, O'Donoghue, Anthony, de Oliveira, Renata B, Ferreira, Rafaela S
Published in Future medicinal chemistry (01.06.2023)
Published in Future medicinal chemistry (01.06.2023)
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New Palladium(II) Complexes Containing Methyl Gallate and Octyl Gallate: Effect against Mycobacterium tuberculosis and Campylobacter jejuni
Silva, Raphael Tristão Cruvinel, Guidotti-Takeuchi, Micaela, Peixoto, Jéssica Laura Miranda, Demarqui, Fernanda Manaia, Mori, Ananda Paula, Dumont, Carolyne Ferreira, Ferreira, Gabriella Rayane Aparecida, Pereira, Gabriele de Menezes, Rossi, Daise Aparecida, Corbi, Pedro Paulo, Pavan, Fernando Rogério, Rezende Júnior, Celso de Oliveira, Melo, Roberta Torres de, Guerra, Wendell
Published in Molecules (Basel, Switzerland) (05.05.2023)
Published in Molecules (Basel, Switzerland) (05.05.2023)
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Quinic acid derivatives inhibit dengue virus replication in vitro
Zanello, Paula Rodrigues, Koishi, Andrea Cristine, Rezende Júnior, Celso de Oliveira, Oliveira, Larissa Albuquerque, Pereira, Adriane Antonia, de Almeida, Mauro Vieira, Duarte dos Santos, Claudia Nunes, Bordignon, Juliano
Published in Virology journal (22.12.2015)
Published in Virology journal (22.12.2015)
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Optimization of benzenesulfonyl derivatives as anti-Trypanosomatidae agents: Structural design, synthesis, and pharmacological assessment against Trypanosoma cruzi and Leishmania infantum
Freitas de Lima Hercos, Guilherme, Gabriela Faleiro de Moura Lodi Cruz, Mariza, Clara Cassiano Martinho, Ana, de Melo Resende, Daniela, Farago Nascimento, Danilo, Derksen Macruz, Paula, Jorge Pilau, Eduardo, Maria Fonseca Murta, Silvane, de Oliveira Rezende Júnior, Celso
Published in Bioorganic & medicinal chemistry (01.05.2024)
Published in Bioorganic & medicinal chemistry (01.05.2024)
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Hit-to-lead optimization of a pyrazinylpiperazine series against Leishmania infantum and Leishmania braziliensis
Jacques Dit Lapierre, Thibault Joseph William, Cruz, Mariza Gabriela Faleiro de Moura Lodi, Brito, Nícolas Peterson Ferreira, Resende, Daniela de Melo, Souza, Felipe de Oliveira, Pilau, Eduardo Jorge, da Silva, Meryck Felipe Brito, Neves, Bruno Junior, Murta, Silvane Maria Fonseca, Rezende Júnior, Celso de Oliveira
Published in European journal of medicinal chemistry (05.08.2023)
Published in European journal of medicinal chemistry (05.08.2023)
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Synthesis, design, and optimization of a potent and selective series of pyridylpiperazines as promising antimalarial agents
da Silva Oliveira, Douglas Davison, Paz, Franciarli, Brito, Nícolas Peterson Ferreira, Krüger, Arne, Martinho, Ana Clara Cassiano, Lapierre, Thibault Joseph William Jacques Dit, de Oliveira Souza, Felipe, Maltarollo, Vinícius G., Kronenberger, Thales, Mendes, Marina Sena, Nonato, Maria Cristina, Pilau, Eduardo Jorge, Wrenger, Carsten, Wunderlich, Gerhard, Rezende Júnior, Celso de Oliveira
Published in European journal of medicinal chemistry (05.09.2024)
Published in European journal of medicinal chemistry (05.09.2024)
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Chemoinformatics Studies on a Series of Imidazoles as Cruzain Inhibitors
Medeiros, Alex R, Ferreira, Leonardo L G, de Souza, Mariana L, de Oliveira Rezende Junior, Celso, Espinoza-Chávez, Rocío Marisol, Dias, Luiz Carlos, Andricopulo, Adriano D
Published in Biomolecules (Basel, Switzerland) (15.04.2021)
Published in Biomolecules (Basel, Switzerland) (15.04.2021)
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2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling
Ferreira, Rafael Augusto Alves, Junior, Celso de Oliveira Rezende, Martinez, Pablo David Grigol, Koovits, Paul John, Soares, Bruna Miranda, Ferreira, Leonardo L G, Michelan-Duarte, Simone, Chelucci, Rafael Consolin, Andricopulo, Adriano D, Galuppo, Mariana K, Uliana, Silvia R B, Matheeussen, An, Caljon, Guy, Maes, Louis, Campbell, Simon, Kratz, Jadel M, Mowbray, Charles E, Dias, Luiz Carlos
Published in PLoS neglected tropical diseases (22.02.2021)
Published in PLoS neglected tropical diseases (22.02.2021)
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Discovery of Potent, Reversible, and Competitive Cruzain Inhibitors with Trypanocidal Activity: A Structure-Based Drug Design Approach
de Souza, Mariana L, de Oliveira Rezende Junior, Celso, Ferreira, Rafaela S, Espinoza Chávez, Rocio Marisol, Ferreira, Leonardo L. G, Slafer, Brian W, Magalhães, Luma G, Krogh, Renata, Oliva, Glaucius, Cruz, Fabio Cardoso, Dias, Luiz Carlos, Andricopulo, Adriano D
Published in Journal of chemical information and modeling (24.02.2020)
Published in Journal of chemical information and modeling (24.02.2020)
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Crystal structure and in vitro biological studies of a Pt(II) complex based on gallic acid and triphenylphosphine
Tristão Cruvinel Silva, Raphael, Pereira Silva-Caldeira, Priscila, Manaia Demarqui, Fernanda, Duque Lopes, Carla, de Albuquerque, Sérgio, Rogério Pavan, Fernando, Cristina Pereira-Maia, Elene, Diniz, Renata, de Oliveira, Alberto, de Oliveira Rezende Júnior, Celso, Guerra, Wendell
Published in Inorganica Chimica Acta (01.09.2024)
Published in Inorganica Chimica Acta (01.09.2024)
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Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease
de Oliveira Rezende Júnior, Celso, Martinez, Pablo David Grigol, Ferreira, Rafael Augusto Alves, Koovits, Paul John, Miranda Soares, Bruna, Ferreira, Leonardo L.G., Michelan-Duarte, Simone, Chelucci, Rafael Consolin, Andricopulo, Adriano D., Matheeussen, An, Van Pelt, Natascha, Caljon, Guy, Maes, Louis, Campbell, Simon, Kratz, Jadel M., Mowbray, Charles E., Dias, Luiz Carlos
Published in European journal of medicinal chemistry (15.01.2023)
Published in European journal of medicinal chemistry (15.01.2023)
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Discovery and structural optimization of a new series of N-acyl-2-aminobenzothiazole as inhibitors of Zika virus
Flávia Clemente Dias, Renieidy, Murta Rezende Moraes Ribeiro, Beatriz, Marques Cassani, Natasha, Nascimento Farago, Danilo, André Antoniucci, Giovanna, Eduardo de Oliveira Rocha, Rafael, de Oliveira Souza, Felipe, Jorge Pilau, Eduardo, Carolina Gomes Jardim, Ana, Salgado Ferreira, Rafaela, de Oliveira Rezende Júnior, Celso
Published in Bioorganic & medicinal chemistry (15.11.2023)
Published in Bioorganic & medicinal chemistry (15.11.2023)
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Discovery of Arylpiperazines with Broad-Spectrum Antimicrobial Activity and Favorable Pharmacokinetic Profiles
Oliveira, Douglas Davison da Silva, Silva, Nagela Bernadelli Sousa, Lapierre, Thibault Joseph William Jacques Dit, de Souza, Sara Lemes, Brito, Nícolas Peterson Ferreira, Martinho, Ana Clara Cassiano, Clemente Dias, Renieidy Flávia, Farago, Danilo Nascimento, Michelan-Duarte, Simone, Chelucci, Rafael Consolin, Cruz, Mariza Gabriela Faleiro de Moura Lodi, de Melo Resende, Daniela, Andricopulo, Adriano D, Murta, Silvane Maria Fonseca, Ferreira, Leonardo L G, Gomes Martins, Carlos Henrique, de Oliveira Rezende Júnior, Celso
Published in Chemistry & biodiversity (26.09.2024)
Published in Chemistry & biodiversity (26.09.2024)
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New drug discovery strategies for the treatment of benznidazole-resistance in Trypanosoma cruzi , the causative agent of Chagas disease
Murta, Silvane Maria Fonseca, Lemos Santana, Pedro Augusto, Jacques Dit Lapierre, Thibault Joseph William, Penteado, André Berndt, El Hajje, Marissa, Navarro Vinha, Thabata Corazza, Liarte, Daniel Barbosa, de Souza, Mariana Laureano, Goulart Trossini, Gustavo Henrique, de Oliveira Rezende Júnior, Celso, de Oliveira, Renata Barbosa, Ferreira, Rafaela Salgado
Published in Expert opinion on drug discovery (01.06.2024)
Published in Expert opinion on drug discovery (01.06.2024)
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