TP0586532, a non-hydroxamate LpxC inhibitor, has in vitro and in vivo antibacterial activities against Enterobacteriaceae
Fujita, Kiyoko, Takata, Iichiro, Yoshida, Ippei, Okumura, Hirotoshi, Otake, Katsumasa, Takashima, Hajime, Sugiyama, Hiroyuki
Published in Journal of antibiotics (01.02.2022)
Published in Journal of antibiotics (01.02.2022)
Get full text
Journal Article
Pharmacodynamic target assessment and prediction of clinically effective dosing regimen of TP0586532, a novel non-hydroxamate LpxC inhibitor, using a murine lung infection model
Fujita, Kiyoko, Takata, Iichiro, Yoshida, Ippei, Honma, Yusuke, Okumura, Hirotoshi, Otake, Katsumasa, Takashima, Hajime, Sugiyama, Hiroyuki
Published in Journal of infection and chemotherapy : official journal of the Japan Society of Chemotherapy (01.05.2022)
Published in Journal of infection and chemotherapy : official journal of the Japan Society of Chemotherapy (01.05.2022)
Get full text
Journal Article
Metabolic Activation of Benzodiazepines by CYP3A4
MIZUNO, Katsuhiko, KATOH, Miki, OKUMURA, Hirotoshi, NAKAGAWA, Nao, NEGISHI, Toru, HASHIZUME, Takanori, NAKAJIMA, Miki, YOKOI, Tsuyoshi
Published in Drug metabolism and disposition (01.02.2009)
Published in Drug metabolism and disposition (01.02.2009)
Get full text
Journal Article
EXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVER
KATOH, Miki, MATSUI, Tomohito, OKUMURA, Hirotoshi, NAKAJIMA, Miki, NISHIMURA, Masuhiro, NAITO, Shinsaku, TATENO, Chise, YOSHIZATO, Katsutoshi, YOKOI, Tsuyoshi
Published in Drug metabolism and disposition (01.09.2005)
Published in Drug metabolism and disposition (01.09.2005)
Get full text
Journal Article
Change of drug excretory pathway by CCl4-induced liver dysfunction in rat
Okumura, Hirotoshi, Katoh, Miki, Minami, Keiichi, Nakajima, Miki, Yokoi, Tsuyoshi
Published in Biochemical pharmacology (01.08.2007)
Published in Biochemical pharmacology (01.08.2007)
Get full text
Journal Article
In Vitro and In Vivo Activities of TP0480066, a Novel Topoisomerase Inhibitor, against Neisseria gonorrhoeae
Masuko, Aiko, Takata, Iichiro, Fujita, Kiyoko, Okumura, Hirotoshi, Ushiyama, Fumihito, Amada, Hideaki, Sugiyama, Hiroyuki
Published in Antimicrobial agents and chemotherapy (18.03.2021)
Published in Antimicrobial agents and chemotherapy (18.03.2021)
Get full text
Journal Article
Lead optimization of 2-hydroxymethyl imidazoles as non-hydroxamate LpxC inhibitors: Discovery of TP0586532
Ushiyama, Fumihito, Takashima, Hajime, Matsuda, Yohei, Ogata, Yuya, Sasamoto, Naoki, Kurimoto-Tsuruta, Risa, Ueki, Kaori, Tanaka-Yamamoto, Nozomi, Endo, Mayumi, Mima, Masashi, Fujita, Kiyoko, Takata, Iichiro, Tsuji, Satoshi, Yamashita, Haruhiro, Okumura, Hirotoshi, Otake, Katsumasa, Sugiyama, Hiroyuki
Published in Bioorganic & medicinal chemistry (15.01.2021)
Published in Bioorganic & medicinal chemistry (15.01.2021)
Get full text
Journal Article
Humanization of Excretory Pathway in Chimeric Mice with Humanized Liver
Okumura, Hirotoshi, Katoh, Miki, Sawada, Toshiro, Nakajima, Miki, Soeno, Yoshinori, Yabuuchi, Hikaru, Ikeda, Toshihiko, Tateno, Chise, Yoshizato, Katsutoshi, Yokoi, Tsuyoshi
Published in Toxicological sciences (01.06.2007)
Published in Toxicological sciences (01.06.2007)
Get full text
Journal Article
IMAGE PROCESSING DEVICE, IMAGE PROCESSING METHOD, AND PROGRAM
OKUMURA HIROTOSHI, YOSHIDA HIROYUKI, OKAMOTO TAKUYA, ISHIHARA RIEKO, TAKEUCHI TOMOYOSHI, KAWADA YUKI
Year of Publication 23.03.2017
Get full text
Year of Publication 23.03.2017
Patent
IMAGE PROCESSING DEVICE, IMAGE PROCESSING METHOD, AND PROGRAM
OKUMURA HIROTOSHI, YOSHIDA HIROYUKI, OKAMOTO TAKUYA, ISHIHARA RIEKO, TAKEUCHI TOMOYOSHI, KAWADA YUKI
Year of Publication 23.03.2017
Get full text
Year of Publication 23.03.2017
Patent
Image processing device, image processing method, and recording medium
Okumura, Hirotoshi, Takeuchi, Tomoyoshi, Ishihara, Rieko, Yoshida, Hiroyuki, Okamoto, Takuya, Kawata, Yuki
Year of Publication 25.02.2020
Get full text
Year of Publication 25.02.2020
Patent
IMAGE PROCESSING DEVICE, IMAGE PROCESSING METHOD, AND RECORDING MEDIUM
YOSHIDA Hiroyuki, OKUMURA Hirotoshi, ISHIHARA Rieko, TAKEUCHI Tomoyoshi, KAWATA Yuki, OKAMOTO Takuya
Year of Publication 23.03.2017
Get full text
Year of Publication 23.03.2017
Patent